4gsw:A (MET4) to (GLU55) CRYSTAL STRUCTURE OF UBIQUITIN FROM ENTAMOEBA HISTOLYTICA TO 2.15 ANGSTROM | UBIQUITIN, UBIQUITIN-LIKE MODIFIER, UBIQUITIN FOLD, POST- TRANSLATIONAL MODIFICATION, EHUBC5, EHUBA1, UBIQUITINATION, ISOPEPTIDE BOND, PROTEIN BINDING
3e7s:B (TYR250) to (VAL303) STRUCTURE OF BOVINE ENOS OXYGENASE DOMAIN WITH INHIBITOR AR- C95791 | NITRIC OXIDE SYNTHASE, NOS, HEME, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE CALMODULIN-BINDING, FAD, FMN, IRON, METAL- BINDING, NADP, OXIDOREDUCTASE, POLYMORPHISM, ZINC
3eah:A (TYR217) to (LEU270) STRUCTURE OF INHIBITED HUMAN ENOS OXYGENASE DOMAIN | NITRIC OXIDE SYNTHASE, NOS, HEME, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE CALMODULIN-BINDING, FAD, FMN, IRON, METAL- BINDING, NADP, OXIDOREDUCTASE, POLYMORPHISM, ZINC
3eah:B (TYR217) to (LEU270) STRUCTURE OF INHIBITED HUMAN ENOS OXYGENASE DOMAIN | NITRIC OXIDE SYNTHASE, NOS, HEME, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE CALMODULIN-BINDING, FAD, FMN, IRON, METAL- BINDING, NADP, OXIDOREDUCTASE, POLYMORPHISM, ZINC
2al6:A (ARG35) to (LEU98) FERM DOMAIN OF FOCAL ADHESION KINASE | FOCAL ADHESION KINASE FERM DOMAIN AUTOPHOSPHORYLATION SITE SRC SH3 BINDING SITE, TRANSFERASE
2al6:B (MET33) to (LEU98) FERM DOMAIN OF FOCAL ADHESION KINASE | FOCAL ADHESION KINASE FERM DOMAIN AUTOPHOSPHORYLATION SITE SRC SH3 BINDING SITE, TRANSFERASE
3rnb:C (ALA2) to (PHE83) STRUCTURE OF THE TOLUENE/O-XYLENE MONOOXYGENASE HYDROXYLASE T201S/F176W DOUBLE MUTANT | TOLUENE, HYDROXYLASE, FOUR-HELIX BUNDLE, DIIRON, OXYGEN PATHWAY, OXIDOREDUCTASE
3rqo:A (TYR253) to (VAL306) STRUCTURE OF THE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(((3R,4R)-4-(2-((1S,2R/1R,2S)-2-(3-CLOROPHENYL) CYCLOPROPYLAMINO)ETHOXY)PYRROLIDIN-3-YL)METHYL)-4-METHYLPYRIDIN-2- AMINE | OXIDOREDUCTASE, ENZYME-INHIBITOR COMPLEX, OXIDOREDUCTASE-INHIBITOR COMPLEX
3rqp:A (TYR253) to (VAL306) STRUCTURE OF THE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-{[(3R,4R)-4-(2-{[(2R/2S)-1-(3-FLUOROPHENYL)PROPAN-2- YL]AMINO}ETHOXY)PYRROLIDIN-3-YL]METHYL}-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, ENZYME-INHIBITOR COMPLEX, OXIDOREDUCTASE-INHIBITOR COMPLEX
4wjs:A (GLY35) to (GLN98) CRYSTAL STRUCTURE OF RSA4 FROM CHAETOMIUM THERMOPHILUM | RIBOSOME ASSEMBLY, RIBOSOME BIOGENESIS, BIOSYNTHETIC PROTEIN
2awt:A (ASN15) to (GLU69) SOLUTION STRUCTURE OF HUMAN SMALL UBIQUITIN-LIKE MODIFIER PROTEIN ISOFORM 2 (SUMO-2) | UBIQUITIN FOLD, HALF-OPEN BARREL, TWO HELICES, PROTEIN TRANSPORT
3egw:A (MET338) to (ALA385) THE CRYSTAL STRUCTURE OF THE NARGHI MUTANT NARH - C16A | OXIDOREDUCTASE, NITRATE REDUCTION, ELECTRON TRANSFER, MEMBRANE PROTEIN, 4FE-4S, CELL MEMBRANE, ELECTRON TRANSPORT, IRON, IRON-SULFUR, MEMBRANE, METAL-BINDING, MOLYBDENUM, NITRATE ASSIMILATION, TRANSPORT, 3FE-4S, CELL INNER MEMBRANE, FORMYLATION, HEME, TRANSMEMBRANE
3ehv:A (MET1) to (ASP52) X-RAY STRUCTURE OF HUMAN UBIQUITIN ZN(II) ADDUCT | HUMAN UBIQUITIN, ADDUCT, LIGASE
1nos:A (ALA262) to (GLU314) MURINE INDUCIBLE NITRIC OXIDE SYNTHASE OXYGENASE DOMAIN (DELTA 114), IMIDAZOLE COMPLEX | NITRIC OXIDE, L-ARGININE MONOOXYGENASE, HEME, IMIDAZOLE, NOS, NO, OXIDOREDUCTASE
4wph:A (ASP684) to (ILE746) CRYSTAL STRUCTURE OF USP7 UBIQUITIN-LIKE DOMAINS IN COMPACT CONFORMATION | DEUBIQUITINATING (DUB) ENZYME, UBIQUITIN-LIKE (UBL) DOMAINS, ICP0 BINDING SITE, HAUSP, HYDROLASE
4wph:B (ASP684) to (ILE746) CRYSTAL STRUCTURE OF USP7 UBIQUITIN-LIKE DOMAINS IN COMPACT CONFORMATION | DEUBIQUITINATING (DUB) ENZYME, UBIQUITIN-LIKE (UBL) DOMAINS, ICP0 BINDING SITE, HAUSP, HYDROLASE
2b3a:A (ASP11) to (GLU75) SOLUTION STRUCTURE OF THE RAS-BINDING DOMAIN OF THE RAL GUANOSINE DISSOCIATION STIMULATOR | RAS BINDING DOMAIN, UBIQUITIN FOLD, SIGNAL TRANSDUCTION, NMR, AUTOMATICALLY SOLVED, AUREMOL, SIGNALING PROTEIN
1nse:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE | NITRIC OXIDE SYNTHASE, ARGININE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
2bps:A (SER1) to (SER60) UBIQUITIN-LIKE PROTEIN YUKD OF BACILLUS SUBTILIS | YUKD, UBIQUITIN-LIKE PROTEIN, UBIQUITIN
2bps:B (SER1) to (SER60) UBIQUITIN-LIKE PROTEIN YUKD OF BACILLUS SUBTILIS | YUKD, UBIQUITIN-LIKE PROTEIN, UBIQUITIN
2bqq:A (ALA52) to (SER129) X-RAY STRUCTURE OF THE N-TERMINAL DOMAIN OF HUMAN DOUBLECORTIN | DCX DOMAIN, UBIQUITIN-LIKE FOLD, MICROTUBULE ASSOCIATED, SIGNALING PROTEIN, TRANSFERASE
3sdl:C (LEU82) to (ASP133) CRYSTAL STRUCTURE OF HUMAN ISG15 IN COMPLEX WITH NS1 N-TERMINAL REGION FROM INFLUENZA B VIRUS, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET IDS HX6481, HR2873, AND OR2 | STRUCTURAL GENOMICS, PSI-BIOLOGY, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, PROTEIN COMPLEX, VIRAL PROTEIN/ANTIVIRAL PROTEIN, VIRAL PROTEIN-ANTIVIRAL PROTEIN COMPLEX
2bye:A (HIS10) to (GLY81) NMR SOLUTION STRUCTURE OF PHOSPHOLIPASE C EPSILON RA 1 DOMAIN | PHOSPHOLIPASE C EPSILON, RAS ASSOCIATION DOMAIN, UBIQUITIN SUPERFOLD, LIPASE
2pph:A (SER2) to (LEU53) SOLUTION STRUCTURE OF HUMAN MEKK3 PB1 DOMAIN | KINASE SIGNALING DOMAIN, TRANSFERASE
4i6p:B (PHE1) to (ASP62) CRYSTAL STRUCTURE OF PAR3-NTD DOMAIN | PB1 LIKE MOTIF, DUF3534, CELL POLARITY PROTEIN, SIGNALING PROTEIN
2c60:A (ASP44) to (LEU93) CRYSTAL STRUCTURE OF HUMAN MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 3 ISOFORM 2 PHOX DOMAIN AT 1.25 A RESOLUTION | MAP3K3, MAP/ERK KINASE KINASE 3, MAPKKK3, MEKK3, SERINE THREONINE PHOSPHORYLATION, ATP-BINDING, KINASE, MAGNESIUM, METAL-BINDING, NUCLEOTIDE-BINDING, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE
2c7h:A (SER5) to (ASP64) SOLUTION NMR STRUCTURE OF THE DWNN DOMAIN FROM HUMAN RBBP6 | RBBP6, P53-ASSOCIATED, MRNA PROCESSING, SPLICING-ASSOCIATED, OESOPHAGEAL CANCER, UBIQUITIN-LIKE PROTEIN
3sua:D (GLU1745) to (ASP1819) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF PLEXIN-B1 IN COMPLEX WITH RAC1 | AXON GUIDANCE, SIGNAL TRANSDUCTION, APOPTOSIS-SIGNALING PROTEIN COMPLEX
3sua:E (GLU1745) to (ASP1819) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF PLEXIN-B1 IN COMPLEX WITH RAC1 | AXON GUIDANCE, SIGNAL TRANSDUCTION, APOPTOSIS-SIGNALING PROTEIN COMPLEX
3sua:F (GLU1745) to (ASP1819) CRYSTAL STRUCTURE OF THE INTRACELLULAR DOMAIN OF PLEXIN-B1 IN COMPLEX WITH RAC1 | AXON GUIDANCE, SIGNAL TRANSDUCTION, APOPTOSIS-SIGNALING PROTEIN COMPLEX
1d0c:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 3- BROMO-7-NITROINDAZOLE (H4B FREE) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1d0o:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 3- BROMO-7-NITROINDAZOLE (H4B PRESENT) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1d0o:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 3- BROMO-7-NITROINDAZOLE (H4B PRESENT) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1d1v:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH S- ETHYL-N-PHENYL-ISOTHIOUREA (H4B BOUND) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1d1w:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 2- AMINOTHIAZOLINE (H4B BOUND) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1d1x:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 1, 4-PBITU (H4B BOUND) | AHPHA-BETA FOLD, OXIDOREDUCTASE
4xol:B (MET1) to (ASP52) OBSERVING THE OVERALL ROCKING MOTION OF A PROTEIN IN A CRYSTAL - CUBIC UBIQUITIN CRYSTALS. | SIGNALING PROTEIN
4xok:A (MET1) to (ASP52) OBSERVING THE OVERALL ROCKING MOTION OF A PROTEIN IN A CRYSTAL. | UBIQUITIN, ZINC, SIGNALING PROTEIN
4xok:B (MET1) to (ASP52) OBSERVING THE OVERALL ROCKING MOTION OF A PROTEIN IN A CRYSTAL. | UBIQUITIN, ZINC, SIGNALING PROTEIN
1p6n:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NOS HEME DOMAIN WITH L-N(OMEGA)-NITROARGININE-(4R)- AMINO-L-PROLINE AMIDE BOUND | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE, HEME-ENZYME
1p6n:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NOS HEME DOMAIN WITH L-N(OMEGA)-NITROARGININE-(4R)- AMINO-L-PROLINE AMIDE BOUND | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE, HEME-ENZYME
2chx:A (ILE220) to (VAL282) A PHARMACOLOGICAL MAP OF THE PI3-K FAMILY DEFINES A ROLE FOR P110ALPHA IN SIGNALING: THE STRUCTURE OF COMPLEX OF PHOSPHOINOSITIDE 3-KINASE GAMMA WITH INHIBITOR PIK-90 | PHOSPHOINOSITIDE, KINASE, LIPID, INHIBITOR, 3-KINASE, SIGNALING, QUINAZOLINONE, TRANSFERASE
2chz:A (PHE221) to (VAL282) A PHARMACOLOGICAL MAP OF THE PI3-K FAMILY DEFINES A ROLE FOR P110ALPHA IN SIGNALING: THE STRUCTURE OF COMPLEX OF PHOSPHOINOSITIDE 3-KINASE GAMMA WITH INHIBITOR PIK-93 | PHOSPHOINOSITIDE, KINASE, LIPID, INHIBITOR, 3-KINASE, SIGNALING, PHENYLTHIAZOLE, QUINAZOLINONE, TRANSFERASE
2cjn:A (LYS4) to (ASP58) STRUCTURE OF FERREDOXIN, NMR, MINIMIZED AVERAGE STRUCTURE | FERREDOXIN, ELECTRON TRANSPORT, IRON-SULFUR PROTEIN
2cjo:A (ALA1) to (ASP58) STRUCTURE OF FERREDOXIN, NMR, 10 STRUCTURES | FERREDOXIN, ELECTRON TRANSPORT, IRON-SULFUR PROTEIN
4imx:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 3,5-BIS(2-(6-AMINO-4-METHYLPYRIDIN-2-YL)ETHYL) BENZONITRILE | OXIDOREDUCTASE NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4imx:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 3,5-BIS(2-(6-AMINO-4-METHYLPYRIDIN-2-YL)ETHYL) BENZONITRILE | OXIDOREDUCTASE NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
2cs4:A (SER6) to (HIS59) SOLUTION STRUCTURE OF N-TERMINAL DOMAIN OF CHROMOSOME 12 OPEN READING FRAME 2 | GTP BINDING, UBIQUITIN FOLD, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, SIGNALING PROTEIN
1dm6:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N- (4-CHLOROPHENYL)-N'-HYDROXYGUANIDINE (H4B FREE) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1dmi:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6S-H4B | ALPHA-BETA FOLD, OXIDOREDUCTASE
1dmj:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 5, 6-CYCLIC-TETRAHYDROPTERIDINE | ALPHA-BETA FOLD, OXIDOREDUCTASE
1dmj:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 5, 6-CYCLIC-TETRAHYDROPTERIDINE | ALPHA-BETA FOLD, OXIDOREDUCTASE
1dmk:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 4- AMINO-6-PHENYL-TETRAHYDROPTERIDINE | ALPHA-BETA FOLD, OXIDOREDUCTASE
2cu1:A (SER6) to (THR59) SOLUTION STRUCTURE OF THE PB1 DOMAIN OF HUMAN PROTEIN KINASE MEKK2B | PB1 DOMAIN, MITOGEN-ACTIVATED PROTEIN KINASE KINASE KINASE 2, MAPK/ERK KINASE KINASE 2, MEK KINASE 2, MEKK 2, SIGNALING PROTEIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
3t8m:A (ASN218) to (VAL282) RATIONAL DESIGN OF PI3K-ALPHA INHIBITORS THAT EXHIBIT SELECTIVITY OVER THE PI3K-BETA ISOFORM | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2r2o:A (ARG1747) to (ILE1816) CRYSTAL STRUCTURE OF THE EFFECTOR DOMAIN OF HUMAN PLEXIN B1 | PLEXIN, EFFECTOR DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, GLYCOPROTEIN, MEMBRANE, PHOSPHORYLATION, RECEPTOR, SECRETED, TRANSMEMBRANE, SIGNALING PROTEIN
2r2o:B (ARG1747) to (ASP1819) CRYSTAL STRUCTURE OF THE EFFECTOR DOMAIN OF HUMAN PLEXIN B1 | PLEXIN, EFFECTOR DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, GLYCOPROTEIN, MEMBRANE, PHOSPHORYLATION, RECEPTOR, SECRETED, TRANSMEMBRANE, SIGNALING PROTEIN
3gs2:C (GLU225) to (ASP306) RING1B C-TERMINAL DOMAIN/CBX7 CBOX COMPLEX | RING1B, CBOX, CBX7, POLYCOMB, E3-LIGASE, CHROMOSOMAL PROTEIN, TRANSCRIPTION REGULATION, CHROMATIN REGULATOR, TRANSCRIPTION REPRESSOR, LIGASE, METAL-BINDING, NUCLEUS, PHOSPHOPROTEIN, REPRESSOR, TRANSCRIPTION, UBL CONJUGATION PATHWAY, ZINC-FINGER
1q0w:B (MET1) to (ASP52) SOLUTION STRUCTURE OF VPS27 AMINO-TERMINAL UIM-UBIQUITIN COMPLEX | PROTEIN-PROTEIN COMPLEX, TRANSPORT PROTEIN
4j6i:A (ASN218) to (VAL282) DISCOVERY OF THIAZOLOBENZOXEPIN PI3-KINASE INHIBITORS THAT SPARE THE PI3-KINASE BETA ISOFORM | BETA-SPARING, SBDD, CATALYTIC SUBUNIT GAMMA, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1q16:A (MET338) to (ALA385) CRYSTAL STRUCTURE OF NITRATE REDUCTASE A, NARGHI, FROM ESCHERICHIA COLI | MEMBRANE PROTEIN, ELECTRON-TRANSFER, OXIDOREDUCTASE
1e7u:A (ASN218) to (VAL282) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, WORTMANNIN
1e8w:A (ASN218) to (VAL282) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, QUERCETIN
1q5w:B (MET101) to (ASP152) UBIQUITIN RECOGNITION BY NPL4 ZINC-FINGERS | UBIQUITIN, PROTEIN-PROTEIN COMPLEX, ZINC-FINGER, RUBREDOXIN KNUCKLE, NZF DOMAIN, PROTEIN BINDING
1ed6:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH L- NIO (H4B FREE) | NITRIC OXIDE SYNTHASE, HEME PROTEIN, ALPHA-BETA FOLD, OXIDOREDUCTASE
2dx5:B (MET1) to (ASP52) THE COMPLEX STRUCTURE BETWEEN THE MOUSE EAP45-GLUE DOMAIN AND UBIQUITIN | UBIQUITIN, PROTEIN-PROTEIN COMPLEX, PROTEIN TRANSPORT/SIGNALING PROTEIN COMPLEX
2rex:C (ARG1747) to (ASP1819) CRYSTAL STRUCTURE OF THE EFFECTOR DOMAIN OF PLXNB1 BOUND WITH RND1 GTPASE | COMPLEX, STRUCTURAL GENOMICS CONSORTIUM, SGC, GTPASE, GNP, PLEXIN, EFFECTOR DOMAIN, GLYCOPROTEIN, MEMBRANE, PHOSPHORYLATION, RECEPTOR, SECRETED, TRANSMEMBRANE, CYTOSKELETON, GTP-BINDING, LIPOPROTEIN, METHYLATION, NUCLEOTIDE-BINDING, PRENYLATION, SIGNALING PROTEIN- LIPOPROTEIN COMPLEX
4jps:A (GLY188) to (LEU262) CO-CRYSTAL STRUCTURES OF THE LIPID KINASE PI3K ALPHA WITH PAN AND ISOFORM SELECTIVE INHIBITORS | CLASS I PHOSPHATIDYLINOSITOL 3-KINASES, P85 ALPHA, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4jsk:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6,6'-(PENTANE-1,5-DIYL)BIS(4-METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4jsl:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6,6'-(HEPTANE-1,7-DIYL)BIS(4-METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4jsl:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6,6'-(HEPTANE-1,7-DIYL)BIS(4-METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4jsm:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(((5-(((3-FLUOROPHENETHYL)AMINO)METHYL)PYRIDIN-3-YL) OXY)METHYL)-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4jsm:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(((5-(((3-FLUOROPHENETHYL)AMINO)METHYL)PYRIDIN-3-YL) OXY)METHYL)-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3h8h:A (SER224) to (ASN306) STRUCTURE OF THE C-TERMINAL DOMAIN OF HUMAN RNF2/RING1B; | UBIQUITIN FOLD, LIGASE, RING1B, POLYCOMB, E3-LIGASE, NUCLEAR PROTEIN, CHROMOSOMAL PROTEIN, TRANSCRIPTION REGULATION, METAL-BINDING, PROTO- ONCOGENE, CHROMATIN REGULATOR, UBL CONJUGATION PATHWAY, REPRESSOR, TRANSCRIPTION, TRANSCRIPTION REGULATION COMPLEX, NUCLEUS, PHOSPHOPROTEIN, ZINC-FINGER, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
3u8z:A (LYS20) to (LEU75) HUMAN MERLIN FERM DOMAIN | NEUROFIBROMATOSIS, TUMOR SUPPRESSOR, SIGNALING PROTEIN
3u8z:B (LYS20) to (LEU75) HUMAN MERLIN FERM DOMAIN | NEUROFIBROMATOSIS, TUMOR SUPPRESSOR, SIGNALING PROTEIN
3u8z:D (LYS20) to (LEU75) HUMAN MERLIN FERM DOMAIN | NEUROFIBROMATOSIS, TUMOR SUPPRESSOR, SIGNALING PROTEIN
1r4n:I (MET101) to (ASP152) APPBP1-UBA3-NEDD8, AN E1-UBIQUITIN-LIKE PROTEIN COMPLEX WITH ATP | CELL CYCLE
1r4n:J (MET101) to (ASP152) APPBP1-UBA3-NEDD8, AN E1-UBIQUITIN-LIKE PROTEIN COMPLEX WITH ATP | CELL CYCLE
1r4n:K (MET101) to (ASP152) APPBP1-UBA3-NEDD8, AN E1-UBIQUITIN-LIKE PROTEIN COMPLEX WITH ATP | CELL CYCLE
1r4n:L (MET101) to (ASP152) APPBP1-UBA3-NEDD8, AN E1-UBIQUITIN-LIKE PROTEIN COMPLEX WITH ATP | CELL CYCLE
4yoc:C (LEU563) to (PRO635) CRYSTAL STRUCTURE OF HUMAN DNMT1 AND USP7/HAUSP COMPLEX | DNA METHYLATION, DEUBIQUITINATION, DNA METHYLTRANSFERASE, MODIFICATION, TRANSFERASE-HYDROLASE COMPLEX
4yoc:C (ASP684) to (ILE746) CRYSTAL STRUCTURE OF HUMAN DNMT1 AND USP7/HAUSP COMPLEX | DNA METHYLATION, DEUBIQUITINATION, DNA METHYLTRANSFERASE, MODIFICATION, TRANSFERASE-HYDROLASE COMPLEX
4yoc:C (CYS896) to (GLU955) CRYSTAL STRUCTURE OF HUMAN DNMT1 AND USP7/HAUSP COMPLEX | DNA METHYLATION, DEUBIQUITINATION, DNA METHYLTRANSFERASE, MODIFICATION, TRANSFERASE-HYDROLASE COMPLEX
2v4l:A (ASN218) to (VAL282) COMPLEX OF HUMAN PHOSPHOINOSITIDE 3-KINASE CATALYTIC SUBUNIT GAMMA (P110 GAMMA) WITH PIK-284 | TRANSFERASE, LIPID KINASE, PHOSPHOINOSITIDE, PYRAZOLOPYRIMIDINE, S1, KINASE, PIK-284, 3-KINASE, INHIBITOR, SIGNALING
4k5h:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (S)-1,2-BIS((2-AMINO-4-METHYLPYRIDIN-6-YL)-METHOXY)- PROPAN-3-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5h:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (S)-1,2-BIS((2-AMINO-4-METHYLPYRIDIN-6-YL)-METHOXY)- PROPAN-3-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5i:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (R)-1,2-BIS((2-AMINO-4-METHYLPYRIDIN-6-YL)-METHOXY)- PROPAN-3-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5j:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (S)-1,3-BIS((2-AMINO-4-METHYLPYRIDIN-6-YL)-METHOXY)- BUTAN-4-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5j:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (S)-1,3-BIS((2-AMINO-4-METHYLPYRIDIN-6-YL)-METHOXY)- BUTAN-4-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5k:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH ((2S, 3S)-1,3-BIS((6-(2,5-DIMETHYL-1H-PYRROL-1-YL)-4- METHYLPYRIDIN-2-YL)METHOXY)-2-AMINOBUTANE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4k5k:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH ((2S, 3S)-1,3-BIS((6-(2,5-DIMETHYL-1H-PYRROL-1-YL)-4- METHYLPYRIDIN-2-YL)METHOXY)-2-AMINOBUTANE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
1foj:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 7- NITROINDAZOLE-2-CARBOXAMIDINE (H4B PRESENT) | ALPHA-BETA FOLD, NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE
3hm6:X (ARG1747) to (ASP1819) CRYSTAL STRUCTURE OF THE CYTOPLASMIC DOMAIN OF HUMAN PLEXIN B1 | STRUCTURAL GENOMICS CONSORTIUM, SGC, MEMBRANE, TRANSMEMBRANE, RECEPTOR, CELL MEMBRANE, GLYCOPROTEIN, PHOSPHOPROTEIN, SECRETED, SIGNALING PROTEIN
4k7s:C (ILE3) to (ASP52) CRYSTAL STRUCTURE OF ZN2-HUB (HUMAN UBIQUITIN) ADDUCT FROM A SOLUTION 35 MM ZINC ACETATE/1.3 MM HUB | LIGASE, ZN ADDUCT
4k7w:C (ILE3) to (ASP52) CRYSTAL STRUCTURE OF ZN3-HUB(HUMAN UBIQUITIN) ADDUCT FROM A SOLUTION 100 MM ZINC ACETATE/1.3 MM HUB | LIGASE, ZN ADDUCT
4k81:A (LYS106) to (THR163) CRYSTAL STRUCTURE OF THE GRB14 RA AND PH DOMAINS IN COMPLEX WITH GTP- LOADED H-RAS | ADAPTOR PROTEIN, SIGNALING PROTEIN
4k81:C (LYS106) to (THR163) CRYSTAL STRUCTURE OF THE GRB14 RA AND PH DOMAINS IN COMPLEX WITH GTP- LOADED H-RAS | ADAPTOR PROTEIN, SIGNALING PROTEIN
4k81:E (LYS106) to (THR163) CRYSTAL STRUCTURE OF THE GRB14 RA AND PH DOMAINS IN COMPLEX WITH GTP- LOADED H-RAS | ADAPTOR PROTEIN, SIGNALING PROTEIN
4k81:G (LYS106) to (THR163) CRYSTAL STRUCTURE OF THE GRB14 RA AND PH DOMAINS IN COMPLEX WITH GTP- LOADED H-RAS | ADAPTOR PROTEIN, SIGNALING PROTEIN
1roe:A (ALA1) to (LEU76) NMR STUDY OF 2FE-2S FERREDOXIN OF SYNECHOCOCCUS ELONGATUS | ELECTRON TRANSPORT, IRON-SULFUR
1fxt:B (MET1) to (ASP52) STRUCTURE OF A CONJUGATING ENZYME-UBIQUITIN THIOLESTER COMPLEX | MODEL OF THE INTERACTION BETWEEN YEAST UBC1 AND UBIQUITIN AFTER THE FORMATION OF A COVALENT THIOLESTER, LIGASE
4kcp:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHEIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(4-(2-((3-(THIOPHENE-2-CARBOXIMIDAMIDO)BENZYL)AMINO) ETHYL)PHENYL)THIOPHENE-2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4kcs:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(3-((ETHYL(3-FLUOROPHENETHYL)AMINO)METHYL)PHENYL) THIOPHENE-2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4kcs:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(3-((ETHYL(3-FLUOROPHENETHYL)AMINO)METHYL)PHENYL) THIOPHENE-2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
1rs8:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NOS HEME DOMAIN WITH D-LYSINE-D-NITROARGININE AMIDE BOUND | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE, HEME-ENZYME
4z96:A (HIS683) to (ILE746) CRYSTAL STRUCTURE OF DNMT1 IN COMPLEX WITH USP7 | USP7, DNMT1, HYDROLASE
4z97:A (ASP684) to (ILE746) CRYSTAL STRUCTURE OF USP7 IN COMPLEX WITH DNMT1(K1115Q) | COMPLEX, TRANSFERASE, HYDROLASE
4z97:A (CYS896) to (GLU955) CRYSTAL STRUCTURE OF USP7 IN COMPLEX WITH DNMT1(K1115Q) | COMPLEX, TRANSFERASE, HYDROLASE
2fuh:B (MET1) to (ASP52) SOLUTION STRUCTURE OF THE UBCH5C/UB NON-COVALENT COMPLEX | PROTEIN-PROTEIN COMPLEX UBIQUITIN UBIQUITIN-CONJUGATING ENZYME, LIGASE
1glo:A (GLY62) to (LYS112) CRYSTAL STRUCTURE OF CYS25SER MUTANT OF HUMAN CATHEPSIN S | CATHEPSIN S, PROTEINASE, INHIBITOR, HYDROLASE, THIOL PROTEAS
2g3q:B (MET1) to (ASP52) SOLUTION STRUCTURE OF EDE1 UBA-UBIQUITIN COMPLEX | ENDOCYTOSIS, MONOUBIQUITIN SIGNALING, SOLUTION STRUCTURE, UBA DOMAIN, UBIQUITIN-BINDING MOTIF, ENDOCYTOSIS/SIGNALING PROTEIN COMPLEX
2g6o:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENOS HEME DOMAIN (BH4-FREE) COMPLEXED WITH CO | NITRIC OXIDE SYNTHASE, HEME PROTEIN, DIATOMIC LIGAND, OXIDOREDUCTASE
2gbm:A (MET1) to (ASP60) CRYSTAL STRUCTURE OF THE 35-36 8 GLYCINE INSERTION MUTANT OF UBIQUITIN | LOOP INSERTION, PROTEIN BINDING
4l1b:A (PRO18) to (PHE83) CRYSTAL STRUCTURE OF P110ALPHA COMPLEXED WITH NISH2 OF P85ALPHA | ATP BINDING, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
1t0q:C (THR3) to (PHE83) STRUCTURE OF THE TOLUENE/O-XYLENE MONOOXYGENASE HYDROXYLASE | DIIRON, CARBOXYLATE BRIDGE, 4-HELIX BUNDLE, CHANNEL, OXIDOREDUCTASE
4l23:A (PRO18) to (ASP84) CRYSTAL STRUCTURE OF P110ALPHA COMPLEXED WITH NISH2 OF P85ALPHA AND PI-103 | ATP BINDING, PI-103, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
4l2y:A (PRO18) to (PHE83) CRYSTAL STRUCTURE OF P110ALPHA COMPLEXED WITH NISH2 OF P85ALPHA AND COMPOUND 9D | ATP BINDING, SIGNALING PROTEIN-TRANSFERASE-INHIBITOR COMPLEX
3ibe:A (ILE220) to (VAL282) CRYSTAL STRUCTURE OF A PYRAZOLOPYRIMIDINE INHIBITOR BOUND TO PI3 KINASE GAMMA | PI3KINASE INHIBITOR, ATP-BINDING, KINASE, NUCLEOTIDE- BINDING, TRANSFERASE
1h4r:A (LYS20) to (LEU75) CRYSTAL STRUCTURE OF THE FERM DOMAIN OF MERLIN, THE NEUROFIBROMATOSIS 2 TUMOR SUPPRESSOR PROTEIN. | FERM, NEUROFIBROMATOSIS, NF2, STRUCTURAL PROTEIN, CYTOSKELETON, ANTI-ONCOGENE
4zop:A (GLY188) to (LEU262) CO-CRYSTAL STRUCTURE OF LIPID KINASE PI3K ALPHA WITH A SELECTIVE PHOSPHATIDYLINOSITOL-3 KINASE ALPHA INHIBITOR | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1t94:B (ARG454) to (ILE513) CRYSTAL STRUCTURE OF THE CATALYTIC CORE OF HUMAN DNA POLYMERASE KAPPA | REPLICATION; DNA REPAIR; Y-FAMILY DNA POLYMERASE; TRANSLESION DNA SYNTHESIS; LESION BYPASS
4zri:B (VAL24) to (LEU75) CRYSTAL STRUCTURE OF MERLIN-FERM AND LATS2 | MERLIN, FERM, LATS2
4zrj:A (VAL24) to (LEU75) STRUCTURE OF MERLIN-FERM AND CTD | MERLIN, FERM, CTD, SIGNALING PROTEIN
4zrk:B (PHE22) to (LEU75) MERLIN-FERM AND LATS1 COMPLEX | MERLIN, FERM, LATS1, SIGNALING PROTEIN-TRANSFERASE COMPLEX
4zrk:C (VAL24) to (LEU75) MERLIN-FERM AND LATS1 COMPLEX | MERLIN, FERM, LATS1, SIGNALING PROTEIN-TRANSFERASE COMPLEX
3in5:A (ARG454) to (SER514) STRUCTURE OF HUMAN DNA POLYMERASE KAPPA INSERTING DATP OPPOSITE AN 8-OXOG DNA LESION | ALTERNATIVE SPLICING, DNA DAMAGE, DNA REPAIR, DNA REPLICATION, DNA SYNTHESIS, DNA-BINDING, DNA-DIRECTED DNA POLYMERASE, MAGNESIUM, METAL-BINDING, MUTATOR PROTEIN, NUCLEOTIDYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SCHIFF BASE, TRANSFERASE, ZINC, ZINC-FINGER, TRANSFERASE/DNA COMPLEX
3in5:B (ARG454) to (SER514) STRUCTURE OF HUMAN DNA POLYMERASE KAPPA INSERTING DATP OPPOSITE AN 8-OXOG DNA LESION | ALTERNATIVE SPLICING, DNA DAMAGE, DNA REPAIR, DNA REPLICATION, DNA SYNTHESIS, DNA-BINDING, DNA-DIRECTED DNA POLYMERASE, MAGNESIUM, METAL-BINDING, MUTATOR PROTEIN, NUCLEOTIDYLTRANSFERASE, NUCLEUS, PHOSPHOPROTEIN, POLYMORPHISM, SCHIFF BASE, TRANSFERASE, ZINC, ZINC-FINGER, TRANSFERASE/DNA COMPLEX
1he8:A (ASN218) to (VAL282) RAS G12V - PI 3-KINASE GAMMA COMPLEX | KINASE/HYDROLASE, COMPLEX (PHOSPHOINOSITIDE KINASE/RAS), PHOSPHOINOSITIDE 3-KINASE GAMMA - H-RAS G12V COMPLEX, PHOSPHATIDYLINOSITOL 3-KINASE, PI3K, PI 3-K, PI 3-KINASE, SECOND MESSENGER GENERATION, RAS EFFECTOR, H-RAS G12V, ONCOGENE PROTEIN, GMPPNP, GTP, RAS-BINDING DOMAIN, HEAT DOMAIN
2w7o:A (ARG454) to (ASN518) STRUCTURE AND ACTIVITY OF BYPASS SYNTHESIS BY HUMAN DNA POLYMERASE KAPPA OPPOSITE THE 7,8-DIHYDRO-8- OXODEOXYGUANOSINE ADDUCT | 8-OXO-2P-DEOXY-GUANOSINE-5P-MONOPHOSPHATE, TRANSLESION DNA POLYMERASE, HUMAN DNA POLYMERASE KAPPA, DGTP, DNA REPAIR, DNA DAMAGE, DNA-BINDING PROTEIN
2w7o:B (ARG454) to (SER514) STRUCTURE AND ACTIVITY OF BYPASS SYNTHESIS BY HUMAN DNA POLYMERASE KAPPA OPPOSITE THE 7,8-DIHYDRO-8- OXODEOXYGUANOSINE ADDUCT | 8-OXO-2P-DEOXY-GUANOSINE-5P-MONOPHOSPHATE, TRANSLESION DNA POLYMERASE, HUMAN DNA POLYMERASE KAPPA, DGTP, DNA REPAIR, DNA DAMAGE, DNA-BINDING PROTEIN
3ivf:A (VAL2) to (ALA64) CRYSTAL STRUCTURE OF THE TALIN HEAD FERM DOMAIN | FERM DOMAIN, CELL MEMBRANE, CELL PROJECTION, CYTOSKELETON, MEMBRANE, PHOSPHOPROTEIN, CELL ADHESION, STRUCTURAL PROTEIN
1i35:A (LEU3) to (THR54) SOLUTION STRUCTURE OF THE RAS-BINDING DOMAIN OF THE PROTEIN KINASE BYR2 FROM SCHIZOSACCHAROMYCES POMBE | UBIQUITIN SUPERFOLD, TRANSFERASE
4luw:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-((((3R,5S)-5-(((6-AMINO-4-METHYLPYRIDIN-2-YL)METHOXY) METHYL)PYRROLIDIN-3-YL)OXY)METHYL)-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
2hx2:A (TYR253) to (VAL306) BOVINE ENOS HEME DOMAIN COMPLEXED WITH (4S)-N-{4-AMINO-5-[(2- AMINOETHYL)-HYDROXYAMINO]-PENTYL}-N'-NITROGUANIDINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, INHIBITOR, OXIDOREDUCTASE
1i83:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1,N14-BIS((S-METHYL)ISOTHIOUREIDO)TETRADECANE (H4B FREE) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1i83:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1,N14-BIS((S-METHYL)ISOTHIOUREIDO)TETRADECANE (H4B FREE) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1uf0:A (LYS12) to (SER73) SOLUTION STRUCTURE OF THE N-TERMINAL DCX DOMAIN OF HUMAN DOUBLECORTIN-LIKE KINASE | STRUCTURAL GENOMICS, UBIQUITIN-LIKE FOLD, MICROTUBULE- BINDING, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
1uh6:A (ILE29) to (ASP80) SOLUTION STRUCTURE OF THE MURINE UBIQUITIN-LIKE 5 PROTEIN FROM RIKEN CDNA 0610031K06 | BETA-GRASP FOLD, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, UNKNOWN FUNCTION
2wxf:A (ARG188) to (TYR251) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH PIK-39. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxi:A (ARG188) to (TYR251) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH SW30. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2wxl:A (ARG188) to (TYR251) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH ZSTK474. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
3wa0:C (VAL24) to (LEU75) CRYSTAL STRUCTURE OF MERLIN COMPLEXED WITH DCAF1/VPRBP | MERLIN FERM DOMAIN, CELL ADHESION
3wa0:F (VAL24) to (LEU75) CRYSTAL STRUCTURE OF MERLIN COMPLEXED WITH DCAF1/VPRBP | MERLIN FERM DOMAIN, CELL ADHESION
1isn:A (PHE22) to (MET77) CRYSTAL STRUCTURE OF MERLIN FERM DOMAIN | FERM DOMAIN, CELL ADHESION
5adk:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-(DIMETHYLAMINO)METHYL) PHENOXY)METHYL)QUINOLIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
5adl:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-(METHYLAMINO)METHYL)PHENOXY) METHYL)QUINOLIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
5adn:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-(((3-((DIMETHYLAMINO)METHYL) PHENYL)AMINO)METHYL)QUINOLIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
5ae9:A (ASN187) to (TYR251) CRYSTAL STRUCTURE OF MOUSE PI3 KINASE DELTA IN COMPLEX WITH GSK2292767 | TRANSFERASE
4mgk:E (ASP650) to (LYS706) SELECTIVE ACTIVATION OF EPAC1 AND EPAC2 | GUANINE NUCLEOTIDE EXCHANGE FACTOR, NUCLEOTIDE BINDING, SIGNALING PROTEIN-GTP-BINDING PROTEIN COMPLEX
4mgz:E (ASP650) to (LYS706) SELECTIVE ACTIVATION OF EPAC1 AND EPAC2 | GUANINE NUCLEOTIDE EXCHANGE FACTOR, NUCLEOTIDE BINDING, SIGNALING PROTEIN-GTP-BINDING PROTEIN COMPLEX
4mm3:A (MET1) to (GLY53) CRYSTAL STRUCTURE OF SARS-COV PAPAIN-LIKE PROTEASE PLPRO IN COMPLEX WITH UBIQUITIN ALDEHYDE | NSP3 PAPAIN-LIKE PROTEASE DOMAIN, SIGNALING PROTEIN-HYDROLASE COMPLEX
2j0j:A (ARG35) to (HIS99) CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS. | CELL MIGRATION, FERM, TRANSFERASE, INTEGRIN SIGNALING
2j0k:A (ARG35) to (HIS99) CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS. | CELL MIGRATION, TRANSFERASE, INTEGRIN SIGNALING
2j0k:B (ARG35) to (LEU98) CRYSTAL STRUCTURE OF A FRAGMENT OF FOCAL ADHESION KINASE CONTAINING THE FERM AND KINASE DOMAINS. | CELL MIGRATION, TRANSFERASE, INTEGRIN SIGNALING
2j0m:A (ARG35) to (LEU98) CRYSTAL STRUCTURE A TWO-CHAIN COMPLEX BETWEEN THE FERM AND KINASE DOMAINS OF FOCAL ADHESION KINASE. | FOCAL ADHESION, CELL MIGRATION, PHOSPHORYLATION, FERM, KINASE, TRANSFERASE, ATP-BINDING, INTEGRIN SIGNALING, NUCLEOTIDE-BINDING, TYROSINE-PROTEIN KINASE
4mzo:B (GLY185) to (SER234) MOUSE CATHEPSIN S WITH COVALENT LIGAND (3S,4S)-N-[(2E)-2-IMINOETHYL]- 4-(MORPHOLIN-4-YLCARBONYL)-1-(PHENYLSULFONYL)PYRROLIDINE-3- CARBOXAMIDE | HYDROLASE, CYSTEINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4mzo:H (GLY185) to (SER234) MOUSE CATHEPSIN S WITH COVALENT LIGAND (3S,4S)-N-[(2E)-2-IMINOETHYL]- 4-(MORPHOLIN-4-YLCARBONYL)-1-(PHENYLSULFONYL)PYRROLIDINE-3- CARBOXAMIDE | HYDROLASE, CYSTEINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3zdt:B (ARG35) to (LEU98) CRYSTAL STRUCTURE OF BASIC PATCH MUTANT FAK FERM DOMAIN FAK31-405 K216A, K218A, R221A, K222A | TRANSFERASE, CELL ADHESION
5b83:A (MET153) to (ASP204) CRYSTAL STRUCTURE OF OPTINEURIN UBAN IN COMPLEX WITH LINEAR UBIQUITIN | UBIQUITIN, COILED-COIL, CELLULAR, SIGNALING, NFKB PATHWAY, SIGNALING PROTEIN
2jrh:A (SER2) to (LEU52) SOLUTION STURCTURE OF HUMAN MEKK3 PB1 DOMAIN CIS ISOMER | KINASE SIGNALING DOMAIN, TRANSFERASE
2jt4:B (MET1) to (ASP52) SOLUTION STRUCTURE OF THE SLA1 SH3-3-UBIQUITIN COMPLEX | ENDOCYTOSIS, MONOUBIQUITIN SIGNALING, UBIQUITIN-BINDING MOTIF, SH3, UBIQUITIN, ACTIN-BINDING, CYTOPLASM, CYTOSKELETON, PHOSPHORYLATION, SH3 DOMAIN, DNA DAMAGE, DNA REPAIR, NUCLEUS, UBL CONJUGATION, SIGNALING PROTEIN
1wgr:A (PRO9) to (GLU67) SOLUTION STRUCTURE OF THE RA DOMAIN OF HUMAN GRB7 PROTEIN | RA DOMAIN, GRB7, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, PROTEIN BINDING
1wgy:A (GLY7) to (GLN65) RA DOMAIN OF GUANINE NUCLEOTIDE EXCHANGE FACTOR FOR RAP1 | UBIQUITIN FOLD, RA, GUANINE NUCLEOTIDE EXCHANGE, RAP1, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, STRUCTURAL GENOMICS, SIGNALING PROTEIN
1wi0:A (LEU17) to (SER74) SOLUTION STRUCTURE OF THE PB1 DOMAIN OF MOUSE MITOGEN ACTIVATED PROTEIN KINASE KINASE 5 (MAP2K5) | PB1 DOMAIN, PROTEIN-PROTEIN INTERACTION SITE, CYTOPLASMIC SIGNALLING, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
2kdb:A (THR3) to (ASP57) SOLUTION STRUCTURE OF HUMAN UBIQUITIN-LIKE DOMAIN OF HERPUD2_9_85, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM (NESG) TARGET HT53A | UBL DOMAIN, MEMBRANE, TRANSMEMBRANE, UNFOLDED PROTEIN RESPONSE, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, ONTARIO CENTRE FOR STRUCTURAL PROTEOMICS, OCSP, UNKNOWN FUNCTION, PROTEIN BINDING, SGC
2kfk:B (SER104) to (GLY161) SOLUTION STRUCTURE OF BEM1P PB1 DOMAIN COMPLEXED WITH CDC24P PB1 DOMAIN | PB1, BUDDING, YEAST, PHOX, SIGNALING PROTEIN
2y3a:A (GLY22) to (GLU87) CRYSTAL STRUCTURE OF P110BETA IN COMPLEX WITH ICSH2 OF P85BETA AND THE DRUG GDC-0941 | TRANSFERASE, PHOSPHOINOSITIDE 3-KINASE, RTK
2kk8:A (HIS10) to (ARG62) NMR SOLUTION STRUCTURE OF A PUTATIVE UNCHARACTERIZED PROTEIN OBTAINED FROM ARABIDOPSIS THALIANA: NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET AR3449A | SOLUTION NMR, ARABIDOPSIS THALIANA, AR3449A, UNCHARACTERIZED PUTATIVE PROTEIN, NESG, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, UNKNOWN FUNCTION
2kma:A (VAL2) to (ALA64) NMR STRUCTURE OF THE F0F1 DOUBLE DOMAIN (RESIDUES 1-202) OF THE TALIN FERM DOMAIN | TALIN, FERM, F0, N-TERMINAL, F1, ADHESION, CYTOPLASM, CYTOSKELETON, MEMBRANE, STRUCTURAL PROTEIN
2kma:A (PRO87) to (HIS176) NMR STRUCTURE OF THE F0F1 DOUBLE DOMAIN (RESIDUES 1-202) OF THE TALIN FERM DOMAIN | TALIN, FERM, F0, N-TERMINAL, F1, ADHESION, CYTOPLASM, CYTOSKELETON, MEMBRANE, STRUCTURAL PROTEIN
2kn5:A (MET1) to (ASP52) A CORRESPONDENCE BETWEEN SOLUTION-STATE DYNAMICS OF AN INDIVIDUAL PROTEIN AND THE SEQUENCE AND CONFORMATIONAL DIVERSITY OF ITS FAMILY | BACKRUB, RESIDUAL DIPOLAR COUPLING, BACKBONE FLEXIBILITY, PROTEIN DYNAMICS, CYTOPLASM, ISOPEPTIDE BOND, NUCLEUS, PHOSPHOPROTEIN, UBL CONJUGATION, GENE REGULATION
2knb:A (MET1) to (ASN52) SOLUTION NMR STRUCTURE OF THE PARKIN UBL DOMAIN IN COMPLEX WITH THE ENDOPHILIN-A1 SH3 DOMAIN | UBL, SH3, PARKIN, ENDOPHILIN, CELL JUNCTION, CELL MEMBRANE, CELL PROJECTION, ENDOPLASMIC RETICULUM, LIGASE, MEMBRANE, METAL-BINDING, NUCLEUS, POSTSYNAPTIC CELL MEMBRANE, S-NITROSYLATION, SYNAPSE, UBL CONJUGATION PATHWAY, ZINC-FINGER, ENDOCYTOSIS, LIPID-BINDING, PHOSPHOPROTEIN, SH3 DOMAIN, PROTEIN BINDING
2ktf:A (MET1) to (ASP52) SOLUTION NMR STRUCTURE OF HUMAN POLYMERASE IOTA UBM2 IN COMPLEX WITH UBIQUITIN | TRANSLESION SYNTHESIS DNA POLYMERASE, Y-FAMILY DNA POLYMERASE, UBIQUITIN BINDING MOTIF, UBIQUITIN, ISOPEPTIDE BOND, NUCLEUS, PHOSPHOPROTEIN, PROTEIN BINDING
2l76:A (LEU267) to (PRO315) SOLUTION NMR STRUCTURE OF HUMAN NFATC2IP UBIQUITIN-LIKE DOMAIN, NFATC2IP_244_338, NESG TARGET HT65A/OCSP TARGET HS00387_244_338/SGC- TORONTO | UBIQUITIN-LIKE DOMAIN, STRUCTURAL GENOMICS, PSI-BIOLOGY, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, ONTARIO CENTRE FOR STRUCTURAL PROTEOMICS, OCSP, TRANSCRIPTION
4nnj:B (MET1) to (ASP52) CRYSTAL STRUCTURE OF UBA1 IN COMPLEX WITH UBIQUITIN-AMP AND THIOESTERIFIED UBIQUITIN | UBIQUITIN ACTIVATING ENZYME (E1), UBA1, UBIQUITIN, ACYLADENYLATE, UBIQUITIN THIOESTER, UBIQUITIN ACTIVATION, AMP, THIOESTERIFIED UB, PROTEIN BINDING
4nnj:D (MET1) to (ASP52) CRYSTAL STRUCTURE OF UBA1 IN COMPLEX WITH UBIQUITIN-AMP AND THIOESTERIFIED UBIQUITIN | UBIQUITIN ACTIVATING ENZYME (E1), UBA1, UBIQUITIN, ACYLADENYLATE, UBIQUITIN THIOESTER, UBIQUITIN ACTIVATION, AMP, THIOESTERIFIED UB, PROTEIN BINDING
1wxa:A (GLY10) to (ILE80) SOLUTION STRUCTURE OF RAS-BINDING DOMAIN IN MOUSE AF-6 PROTEIN | RAS-BINDING DOMAIN, UBIQUITIN-LIKE FOLD, AF-6 PROTEIN, STRUCTURAL GENOMICS, AFADIN, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, CELL ADHESION
3zqj:D (SER176) to (GLU253) MYCOBACTERIUM TUBERCULOSIS UVRA | DNA BINDING PROTEIN, NUCLEOTIDE EXCISION REPAIR,
2lvp:B (MET1) to (ASP52) GP78CUE DOMAIN BOUND TO THE DISTAL UBIQUITIN OF K48-LINKED DIUBIQUITIN | CUE DOMAIN, SIGNALING PROTEIN-LIGASE COMPLEX
2lxa:A (VAL74) to (ASP128) SOLUTION STRUCTURE OF THE GET5 UBIQUITIN-LIKE DOMAIN | UBIQUITIN-LIKE DOMAIN, PROTEIN-PROTEIN INTERACTION, SGT2 BINDING DOMAIN, GET PATHWAY, PROTEIN BINDING
4nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, H4B-FREE, L-ARG COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, COMPLEX (OXIDOREDUCTASE-PEPTIDE), COMPLEX (OXIDOREDUCTASE-PEPTIDE) COMPLEX
2mh7:A (VAL3) to (ASP55) SOLUTION STRUCTURE OF OXIDIZED [2FE-2S] FERREDOXIN PETF FROM CHLAMYDOMONAS REINHARDTII | OXIDOREDUCTASE
2mlb:A (ILE4) to (PRO53) NMR SOLUTION STRUCTURE OF A COMPUTATIONAL DESIGNED PROTEIN BASED ON TEMPLATE OF HUMAN ERYTHROCYTIC UBIQUITIN | PROTEIN DESIGN, STATISTICAL ENERGY FUNCTION, UBIQUITIN, DE NOVO PROTEIN
3zvv:A (ASN218) to (VAL282) FRAGMENT BOUND TO PI3KINASE GAMMA | TRANSFERASE, PI3 KINASE GAMMA
5c56:A (ASP684) to (ILE746) CRYSTAL STRUCTURE OF USP7/HAUSP IN COMPLEX WITH ICP0 | VIRUS PROTEIN ICP0, USP7, DEUBIQUITINATION, HYDROLASE
5c56:A (ARG891) to (GLU955) CRYSTAL STRUCTURE OF USP7/HAUSP IN COMPLEX WITH ICP0 | VIRUS PROTEIN ICP0, USP7, DEUBIQUITINATION, HYDROLASE
2mre:A (ILE3) to (ASP52) NMR STRUCTURE OF THE RAD18-UBZ/UBIQUITIN COMPLEX | PROTEIN COMPLEX, LIGASE-TRANSLATION COMPLEX, REPLICATION-SIGNALING PROTEIN COMPLEX
2mur:B (ILE103) to (ASP152) SOLUTION STRUCTURE OF THE HUMAN FAAP20 UBZ-UBIQUITIN COMPLEX | UBZ, FAAP20, ZINC-FINGER, FANCONI ANEMIA, PROTEIN BINDING
2mw5:A (GLY22) to (ASP76) BACKBONE FOLD OF HUMAN SMALL UBIQUITIN LIKE MODIFIER PROTEIN-1 (SUMO- 1) BASED ON PROT3D-NMR APPROACH. | HUMAN SUMO, SMALL UBIQUITIN LIKE MODIFIER, SUMO-1, PROTEIN BINDING
2n13:B (ILE103) to (ASP152) COMPLEX STRUCTURE OF MYUB (1080-1122) OF HUMAN MYOSIN VI WITH K63-DIUB | MOTOR PROTEIN-PROTEIN BINDING COMPLEX
2n13:C (MET201) to (ASP252) COMPLEX STRUCTURE OF MYUB (1080-1122) OF HUMAN MYOSIN VI WITH K63-DIUB | MOTOR PROTEIN-PROTEIN BINDING COMPLEX
4ny0:A (ARG35) to (HIS99) CRYSTAL STRUCTURE OF FERM DOMAIN OF HUMAN FOCAL ADHESION KINASE | FERM DOMAIN, FOCAL ADHESION KINASE, FOCAL TARGETING DOMAIN, INTEGRIN SIGNALING, TRANSFERASE
4ny0:B (ARG35) to (LEU98) CRYSTAL STRUCTURE OF FERM DOMAIN OF HUMAN FOCAL ADHESION KINASE | FERM DOMAIN, FOCAL ADHESION KINASE, FOCAL TARGETING DOMAIN, INTEGRIN SIGNALING, TRANSFERASE
4ny0:C (ARG35) to (LEU98) CRYSTAL STRUCTURE OF FERM DOMAIN OF HUMAN FOCAL ADHESION KINASE | FERM DOMAIN, FOCAL ADHESION KINASE, FOCAL TARGETING DOMAIN, INTEGRIN SIGNALING, TRANSFERASE
2n3u:C (MET1) to (ASP52) SOLUTION STRUCTURE OF THE RPN1 T1 SITE ENGAGING TWO MONOUBIQUITIN MOLECULES | PROTEIN BINDING
2n7k:A (ILE3) to (ASP52) UNVEILING THE STRUCTURAL DETERMINANTS OF KIAA0323 BINDING PREFERENCE FOR NEDD8 | SIGNALING PROTEIN
2n9p:C (VAL19) to (ASP68) SOLUTION STRUCTURE OF RNF126 N-TERMINAL ZINC FINGER DOMAIN IN COMPLEX WITH BAG6 UBIQUITIN-LIKE DOMAIN | E3 LIGASE, ZINC FINGER, LIGASE
2nbv:B (LYS31) to (ASP83) SOLUTION STRUCTURE OF THE RPN13 PRU DOMAIN ENGAGING THE HPLIC2 UBL DOMAIN | PROTEIN BINDING
2ns5:A (GLU17) to (LEU78) THE CONSERVED N-TERMINAL DOMAIN OF PAR-3 ADOPTS A NOVEL PB1- LIKE STRUCTURE REQUIRED FOR PAR-3 OLIGOMERIZATION AND APICAL MEMBRANE LOCALIZATION | CELL POLARITY, PAR-3, N-TERMINAL DOMAIN, PB1 DOMAIN, ASYMMETRIC MEMBRANE LOCALIZATION, SIGNALING PROTEIN
2nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE SUBSTRATE COMPLEX | NITRIC OXIDE SYNTHASE, ARGININE, HEME PROTEIN, TETRAHYDROBIOPTERIN, COMPLEX (OXIDOREDUCTASE-PEPTIDE), COMPLEX (OXIDOREDUCTASE-PEPTIDE) COMPLEX
2nse:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE SUBSTRATE COMPLEX | NITRIC OXIDE SYNTHASE, ARGININE, HEME PROTEIN, TETRAHYDROBIOPTERIN, COMPLEX (OXIDOREDUCTASE-PEPTIDE), COMPLEX (OXIDOREDUCTASE-PEPTIDE) COMPLEX
2ylm:A (ASP684) to (ILE746) MECHANISM OF USP7 (HAUSP) ACTIVATION BY ITS C-TERMINAL UBIQUITIN-LIKE DOMAIN (HUBL) AND ALLOSTERIC REGULATION BY GMP-SYNTHETASE. | HYDROLASE, UBL
2ylm:A (ARG891) to (GLU955) MECHANISM OF USP7 (HAUSP) ACTIVATION BY ITS C-TERMINAL UBIQUITIN-LIKE DOMAIN (HUBL) AND ALLOSTERIC REGULATION BY GMP-SYNTHETASE. | HYDROLASE, UBL
1l7y:A (THR15) to (PRO69) SOLUTION NMR STRUCTURE OF C. ELEGANS PROTEIN ZK652.3. NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET WR41. | C.ELEGANS, UNKNOWN FUNCTION, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, ZK652.3, UBIQUITIN FOLD, BETA-GRASP FOLD, UFM1, UBIQUITIN-FOLD MODIFIER 1, NESG, STRUCTURAL GENOMICS, STRUCTURAL PROTEOMICS, HYPOTHETICAL, PSI, PROTEIN STRUCTURE INITIATIVE
3jwx:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-[(3'R,4'R)-4'-((6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL) PYRROLIDIN-3'-YL]-N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3jwx:B (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-[(3'R,4'R)-4'-((6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL) PYRROLIDIN-3'-YL]-N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3jwy:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-{(3'R,4'S)-4'-[(6"-AMINO-4"-METHYLPYRIDIN-2"-YL) METHYL]PYRROLIDIN-3'-YL}-N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3jwz:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-[(3' S,4' R)-4'-((6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL) PYRROLIDIN-3'-YL]-N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
5chw:H (GLU78) to (ASP131) STRUCTURE OF ISG15 IN SPACE GROUP P212121 | UBIQUITIN-LIKE PROTEIN, INTERFERON INDUCED, SIGNALING PROTEIN
1m9k:A (TYR251) to (LEU304) HUMAN ENDOTHELIAL NITRIC OXIDE SYNTHASE WITH 7- NITROINDAZOLE BOUND | OXIDOREDUCTASE
1m9r:B (TYR251) to (LEU304) HUMAN ENDOTHELIAL NITRIC OXIDE SYNTHASE WITH 3-BROMO-7- NITROINDAZOLE BOUND | OXIDOREDUCTASE
1xzq:B (THR3) to (GLU52) STRUCTURE OF THE GTP-BINDING PROTEIN TRME FROM THERMOTOGA MARITIMA COMPLEXED WITH 5-FORMYL-THF | GTP-BINDING, THF-BINDING, TRNA-MODIFICATION, HYDROLASE
5d68:B (LYS417) to (GLN473) CRYSTAL STRUCTURE OF KRIT1 ARD-FERM | ANKYRIN REPEAT DOMAIN, FERM DOMAIN, CEREBRAL CAVERNOUS MALFORMATIONS, SIGNALING PROTEIN
1yiw:B (LEU1) to (ASP52) X-RAY CRYSTAL STRUCTURE OF A CHEMICALLY SYNTHESIZED UBIQUITIN | UBIQUITIN, STRUCTURAL PROTEIN
3kuz:A (GLY1197) to (ASP1271) CRYSTAL STRUCTURE OF THE UBIQUITIN LIKE DOMAIN OF PLXNC1 | PLEXIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC
1yj1:A (ILE3) to (ASP52) X-RAY CRYSTAL STRUCTURE OF A CHEMICALLY SYNTHESIZED [D-GLN35]UBIQUITIN | UBIQUITIN, STRUCTURAL PROTEIN
1yj1:B (LEU1) to (ASP52) X-RAY CRYSTAL STRUCTURE OF A CHEMICALLY SYNTHESIZED [D-GLN35]UBIQUITIN | UBIQUITIN, STRUCTURAL PROTEIN
3l08:A (ASN218) to (LEU281) STRUCTURE OF PI3K GAMMA WITH A POTENT INHIBITOR: GSK2126458 | PI3K GAMMA, LIPID KINASE, PHOSPHOINOSITIDE, INHIBITOR, GSK2126458, SIGNALING, KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE
3l0w:B (ILE3) to (ASP52) STRUCTURE OF SPLIT MONOUBIQUITINATED PCNA WITH UBIQUITIN IN POSITION TWO | REPLICATION, DNA DAMAGE, DNA REPAIR, DNA REPLICATION, DNA- BINDING, ISOPEPTIDE BOND, NUCLEUS, UBL CONJUGATION
3l13:A (ASN218) to (VAL282) CRYSTAL STRUCTURES OF PAN-PI3-KINASE AND DUAL PAN-PI3-KINASE/MTOR INHIBITORS | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, PI3K-GAMMA P110 GAMMA
3l54:A (ASN218) to (LEU281) STRUCTURE OF PI3K GAMMA WITH INHIBITOR | PI3K, PI3K GAMMA, PHOSPHATIDYLINOSITOL, PI3, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, TRANSFERASE
1yx6:B (ILE3) to (ASP52) SOLUTION STRUCTURE OF S5A UIM-2/UBIQUITIN COMPLEX | NMR, POLYUBIQUITIN, PROTEASOME, S5A, UIM, HYDROLASE
4ps7:A (ASN218) to (VAL282) STRUCTURE OF PI3K GAMMA IN COMPLEX WITH N-[6-(PYRIDIN-3-YL)-1,3- BENZOTHIAZOL-2-YL]ACETAMIDE | SERINE/THREONINE PROTEIN KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4anv:A (ASN218) to (VAL282) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4anw:A (ASN218) to (LEU281) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4anx:A (ASN218) to (VAL282) COMPLEXES OF PI3KGAMMA WITH ISOFORM SELECTIVE INHIBITORS. | TRANSFERASE
4py5:A (ALA38) to (GLU98) THERMOVIBRIO AMMONIFICANS RNASE H3 IN COMPLEX WITH 19-MER RNA/DNA | RNASE H FOLD, RNA/DNA HYBRID, HYDROLASE-DNA-RNA COMPLEX
4pyu:A (ILE2) to (ASP53) THE CONSERVED UBIQUITIN-LIKE PROTEIN HUB1 PLAYS A CRITICAL ROLE IN SPLICING IN HUMAN CELLS | UBIQUITIN-LIKE, PRE-MRNA SPLICING, PROTEIN BINDING-ALLERGEN COMPLEX
4pyu:B (ILE2) to (ASP53) THE CONSERVED UBIQUITIN-LIKE PROTEIN HUB1 PLAYS A CRITICAL ROLE IN SPLICING IN HUMAN CELLS | UBIQUITIN-LIKE, PRE-MRNA SPLICING, PROTEIN BINDING-ALLERGEN COMPLEX
4pyu:K (HIS0) to (ASP53) THE CONSERVED UBIQUITIN-LIKE PROTEIN HUB1 PLAYS A CRITICAL ROLE IN SPLICING IN HUMAN CELLS | UBIQUITIN-LIKE, PRE-MRNA SPLICING, PROTEIN BINDING-ALLERGEN COMPLEX
4pyz:A (HIS683) to (ILE746) CRYSTAL STRUCTURE OF THE FIRST TWO UBL DOMAINS OF DEUBIQUITYLASE USP7 | DEUBIQUITYLASE, UBIQUITIN-LIKE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE
4pyz:B (ASP684) to (ILE746) CRYSTAL STRUCTURE OF THE FIRST TWO UBL DOMAINS OF DEUBIQUITYLASE USP7 | DEUBIQUITYLASE, UBIQUITIN-LIKE DOMAIN, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, HYDROLASE
5dxh:D (PRO18) to (ASP84) P110ALPHA/P85ALPHA WITH COMPOUND 5 | LIPID KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5dxu:A (ARG188) to (TYR251) P110DELTA/P85ALPHA WITH GDC-0326 | LIPID KINASE, INHIBITOR, TRANSFERASE-INHIBITOR COMPLEX
4q5h:B (MET1) to (ASP52) SHIGELLA EFFECTOR KINASE OSPG BOUND TO AMPPNP AND E2-UB UBCH7-UB CONJUGATE | PROTEIN-PROTEIN COMPLEX, STRUCTURAL GENOMICS, MONTREAL-KINGSTON BACTERIAL STRUCTURAL GENOMICS INITIATIVE, BSGI, KINASE FOLD, INHIBITION OF NF-KB PATHWAY, UNKNOWN FUNCTION, PROTEIN BINDING
2a5u:A (ASN218) to (VAL282) CRYSTAL STRUCTURE OF HUMAN PI3KGAMMA COMPLEXED WITH AS605240 | PROTEIN-INHIBITOR COMPLEX, PI3KG, TRANSFERASE
2aeh:A (MET33) to (LEU98) FOCAL ADHESION KINASE 1 | FERM DOMAIN, TRANSFERASE
3bc3:A (GLY61) to (THR110) EXPLORING INHIBITOR BINDING AT THE S SUBSITES OF CATHEPSIN L | CATHEPSIN L INHIBITOR BINDING AT THE S SUBSITES, GLYCOPROTEIN, HYDROLASE, LYSOSOME, PROTEASE, THIOL PROTEASE, ZYMOGEN
4bpv:B (GLY185) to (SER234) MOUSE CATHEPSIN S WITH COVALENT LIGAND | HYDROLASE, CYSTEINE PROTEASE, COVALENT LIGAND
3n11:A (GLY230) to (ARG273) CRYSTAL STRICTURE OF WILD-TYPE CHITINASE FROM BACILLUS CEREUS NCTU2 | CHITINASE, CHINCTU2, WILD-TYPE, HYDROLASE
3n12:A (GLY230) to (ARG273) CRYSTAL STRICTURE OF CHITINASE IN COMPLEX WITH ZINC ATOMS FROM BACILLUS CEREUS NCTU2 | CHITINASE, CHINCTU2, ZINC ATOMS, COMPLEX, HYDROLASE
3n1a:A (GLY230) to (ARG273) CRYSTAL STRICTURE OF E145G/Y227F CHITINASE IN COMPLEX WITH CYCLO-(L- HIS-L-PRO) FROM BACILLUS CEREUS NCTU2 | CHITINASE, CHINCTU2, COMPLEX, CYCLO-(L-HIS-L-PRO), MUTATION, HYDROLASE
3n5q:B (ALA254) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6,6'-(2,2'-(5-AMINO-1,3-PHENYLENE)BIS(ETHANE-2,1-DIYL))BIS(4- METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n5r:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 4-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2-YL)ETHYL)PHENETHYL)-6- METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n5s:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 4-(2-(5-(2-(6-AMINO-4-METHYLPYRIDIN-2-YL)ETHYL)PYRIDIN-3-YL) ETHYL)-6-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n5t:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6,6'-(2,2'-(PYRIDINE-3,5-DIYL)BIS(ETHANE-2,1-DIYL))BIS(4- METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n6b:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE H373S SINGLE MUTANT HEME DOMAIN COMPLEXED WITH 6,6'-(2,2'-(PYRIDINE-3,5-DIYL)BIS(ETHANE- 2,1-DIYL))BIS(4-METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
5fj3:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((4-CHLORO-3-((METHYLAMINO)METHYL) PHENOXY)METHYL)QUINOLIN-2-AMINE IN THE ABSENCE OF ACETATE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4c3a:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-((((3S, 5R)-5-(((6-AMINO-4- METHYLPYRIDIN-2-YL)METHOXY)METHYL)PYRROLIDIN-3-YL)OXY) METHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4c3a:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-((((3S, 5R)-5-(((6-AMINO-4- METHYLPYRIDIN-2-YL)METHOXY)METHYL)PYRROLIDIN-3-YL)OXY) METHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
3cf6:E (ASP650) to (LYS706) STRUCTURE OF EPAC2 IN COMPLEX WITH CYCLIC-AMP AND RAP | EPAC, RAPGEF4, RAP, RAP1B, CAMP, SP-CAMPS, GEF, GUNANINE NUCLEOTIDE EXCHANGE FACTOR, G-PROTEIN, GTP-BINDING, NUCLEOTIDE-BINDING, SIGNALING PROTEIN REGULATOR-GTP-BINDING PROTEIN COMPLEX, SIGNALING PROTEIN-GTP-BINDING PROTEIN COMPLEX
4rf0:B (MET1) to (ASP52) CRYSTAL STRUCTURE OF THE MIDDLE-EAST RESPIRATORY SYNDROME CORONAVIRUS PAPAIN-LIKE PROTEASE IN COMPLEX WITH UBIQUITIN (SPACE GROUP P6522) | ZINC RIBBON, DEUBIQUITINASE, PAPAIN-LIKE PROTEASE, PROTEIN BINDING
3nlg:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'S,4'R)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nlf:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'S)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nlf:B (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'S)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nlh:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN N368D MUTANT COMPLEXED WITH 6-{{(3'S,4'S)-3'-[2"-(3'''- FLUOROPHENETHYLAMINO)ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN- 2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nli:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE N368D MUTANT HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'R)-3'-[2"-(3'''- FLUOROPHENETHYLAMINO)ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN- 2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nli:B (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE N368D MUTANT HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'R)-3'-[2"-(3'''- FLUOROPHENETHYLAMINO)ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN- 2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3cmm:B (MET1) to (ASP52) CRYSTAL STRUCTURE OF THE UBA1-UBIQUITIN COMPLEX | UBIQUITIN, E1, UBA1, PROTEIN TURNOVER, LIGASE, CONFORMATIONAL CHANGE, THIOESTER, ADENYLATION, TRANSTHIOESTERIFICATION, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, UBL CONJUGATION PATHWAY, DNA DAMAGE, DNA REPAIR, LIGASE-PROTEIN BINDING COMPLEX
3nlu:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-{(3'R,4'R)-4'-[(6"-AMINO-4"-METHYLPYRIDIN-2"-YL) METHYL]PYRROLIDIN-3'-YL}-N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nob:H (MET1) to (ASP52) STRUCTURE OF K11-LINKED DI-UBIQUITIN | UBIQUITIN LYSINE-11, PROTEIN BINDING
4car:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-FLUOROPHENETHYLAMINO)METHYL) QUINOLIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4car:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-FLUOROPHENETHYLAMINO)METHYL) QUINOLIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4rm8:B (VAL7) to (LEU61) CRYSTAL STRUCTURE OF HUMAN EZRIN IN SPACE GROUP P21 | FERM DOMAIN, C-ERMAD DOMAIN, MEMBRANE CYTOSKELETON LINKERS, ACTIN BINDING, PEPTIDE BINDING PROTEIN
4rm9:A (VAL7) to (LEU61) CRYSTAL STRUCTURE OF HUMAN EZRIN IN SPACE GROUP C2221 | FERM DOMAIN, C-ERMAD DOMAIN, MEMBRANE CYTOSKELETON LINKERS, ACTIN BINDING, PEPTIDE BINDING PROTEIN
3nse:A (TYR253) to (VAL306) BOVINE ENOS, H4B-FREE, SEITU COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, COMPLEX (OXIDOREDUCTASE-PEPTIDE), COMPLEX (OXIDOREDUCTASE-PEPTIDE) COMPLEX
4cft:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-FLUOROPHENETHYLAMINO)ETHYL) QUINOLIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cft:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 7-((3-FLUOROPHENETHYLAMINO)ETHYL) QUINOLIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
5fvz:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(2-(5-(3-(DIMETHYLAMINO)PROPYL) PYRIDIN-3-YL)ETHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
5fvz:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(2-(5-(3-(DIMETHYLAMINO)PROPYL) PYRIDIN-3-YL)ETHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
5fvy:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(2-(5-(4-METHYLPIPERAZIN- 1-YL)PYRIDIN-3-YL)ETHYL)PYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
3nzs:A (ASN218) to (VAL282) STRUCTURE-BASED OPTIMIZATION OF PYRAZOLO -PYRIMIDINE AND -PYRIDINE INHIBITORS OF PI3-KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3nzu:A (ASN218) to (VAL282) STRUCTURE-BASED OPTIMIZATION OF PYRAZOLO -PYRIMIDINE AND -PYRIDINE INHIBITORS OF PI3-KINASE | KINASE P110, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5g2n:A (ASN218) to (VAL282) X-RAY STRUCTURE OF PI3KINASE GAMMA IN COMPLEX WITH COPANLISIB | TRANSFERASE
5g55:A (ASN218) to (VAL282) 3-QUINOLINE CARBOXAMIDES INHIBITORS OF PI3K | TRANSFERASE, ATM
4ctz:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (S)-6-(2-AMINO-2-(3-(2-(4-METHYLPYRIDIN-2-YL) ETHYL)PHENYL)ETHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cty:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (R)-6-(2-AMINO-2-(3-(2-(6-AMINO-4-METHYLPYRIDIN- 2-YL)ETHYL)PHENYL)ETHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cu0:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (R)-6-(3-AMINO-2-(5-(2-(6-AMINO-4- METHYLPYRIDIN-2-YL)ETHYL)PYRIDIN-3-YL)PROPYL)-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cu1:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-[(2S)-3-AMINO-2-{5-[2-(6-AMINO- 4-METHYLPYRIDIN-2-YL)ETHYL]PYRIDIN-3-YL}PROPYL]-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cul:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-ACETYL-2-AMINO-7,7-DIMETHYL-7,8- DIHYDROPTERIDIN-4(3H)-ONE | OXIDOREDUCTASE, COFACTOR ANALOG COMPLEX
4cum:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (9AS)-2-AMINO-9A-METHYL-6,7,8,9,9A, 10-HEXAHYDROBENZO[G]PTERIDIN-4(3H)-ONE | OXIDOREDUCTASE, COFACTOR ANALOG COMPLEX
4cum:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (9AS)-2-AMINO-9A-METHYL-6,7,8,9,9A, 10-HEXAHYDROBENZO[G]PTERIDIN-4(3H)-ONE | OXIDOREDUCTASE, COFACTOR ANALOG COMPLEX
4cun:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (9AS)-2-AMINO-9A-METHYL-8,9,9A,10- TETRAHYDROBENZO[G]PTERIDINE-4,6(3H,7H)-DIONE | OXIDOREDUCTASE, COFACTOR ANALOG COMPLEX
4cvg:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN (H4B-FREE) SUPPLEMENTED WITH 50UM ZN ACETATE AND WITH POOR BINDING OF 6-ACETYL-2-AMINO-7,7-DIMETHYL-7,8-DIHYDROPTERIDIN-4(3H)-ONE. | OXIDOREDUCTASE, COFACTOR ANALOG COMPLEX
3dbs:A (ASN218) to (VAL282) STRUCTURE OF PI3K GAMMA IN COMPLEX WITH GDC0941 | PI3K GAMMA, INHIBITOR, KINASE, TRANSFERASE
4cww:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-((5-(4- METHYLPYRIDIN-2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL) PYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cwx:A (TYR253) to (VAL306) ALPHA-KETOGLUTARATE-DEPENDENT DIOXYGENASE COMPLEX1 | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cwy:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(5-(((3R,4R)-4-((6-AMINO-4- METHYLPYRIDIN-2-YL)METHYL)PYRROLIDIN-3-YL)OXY)PENTYL)-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cwy:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(5-(((3R,4R)-4-((6-AMINO-4- METHYLPYRIDIN-2-YL)METHYL)PYRROLIDIN-3-YL)OXY)PENTYL)-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cx0:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE Y477A MUTANT HEME DOMAIN IN COMPLEX WITH 6-((((3S, 5R)-5-(((6- AMINO-4-METHYLPYRIDIN-2-YL)METHOXY)METHYL)PYRROLIDIN-3-YL) OXY)METHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cx1:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE L111A MUTANT HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-( (5-(4-METHYLPYRIDIN-2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL) PYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cx2:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(5-(((3R,4R)-4-((6-AMINO-4- METHYLPYRIDIN-2-YL)METHYL)PYRROLIDIN-3-YL)OXY)PENTYL)-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cx2:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(5-(((3R,4R)-4-((6-AMINO-4- METHYLPYRIDIN-2-YL)METHYL)PYRROLIDIN-3-YL)OXY)PENTYL)-4- METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
3ddc:B (GLY229) to (SER331) CRYSTAL STRUCTURE OF NORE1A IN COMPLEX WITH RAS | ONCOGENE, TUMORSUPPRESSOR, UBIQUITIN FOLD, RAS EFFECTOR, RAP1, H-RAS, RASSF1, RASSF5, RAPL, NORE1, GMPPNP, ADAPTOR, APOPTOSIS, MICROTUBULES, HYDROLASE-APOPTOSIS COMPLEX, DISEASE MUTATION, GOLGI APPARATUS, GTP-BINDING, LIPOPROTEIN, MEMBRANE, METHYLATION, NUCLEOTIDE-BINDING, PALMITATE, PRENYLATION, PROTO-ONCOGENE, ANTI- ONCOGENE, CELL CYCLE, METAL-BINDING, MICROTUBULE, PHORBOL-ESTER BINDING, ZINC-FINGER
4d1p:A (TYR251) to (LEU304) STRUCTURE OF HUMAN ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-((((3S, 5R)-5-(((6-AMINO-4- METHYLPYRIDIN-2-YL)METHOXY)METHYL)PYRROLIDIN-3-YL)OXY) METHYL)-4-METHYLPYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE,
4d33:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (N1-(2-(1H-IMIDAZOL-1-YL)PYRIMIDIN- 4-YL)-N2-(3-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d34:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 2-(2-(1H-IMIDAZOL-1-YL)PYRIMIDIN-4- YL)-N-(3-FLUOROPHENETHYL)ETHAN-1-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d34:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 2-(2-(1H-IMIDAZOL-1-YL)PYRIMIDIN-4- YL)-N-(3-FLUOROPHENETHYL)ETHAN-1-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d35:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-2-(2-(1H-IMIDAZOL-1-YL)PYRIMIDIN- 4-YL)ETHYL-3-(3-FLUOROPHENYL)PROPAN-1-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d35:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-2-(2-(1H-IMIDAZOL-1-YL)PYRIMIDIN- 4-YL)ETHYL-3-(3-FLUOROPHENYL)PROPAN-1-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d37:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-{[(1R,2R)-2-(3-FLUOROPHENYL)CYCLOPROPYL] ETHYL}-2-[2-(1H-IMIDAZOL-1-YL)PYRIMIDIN-4-YL]ETHANAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
3dqt:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NOS HEME DOMAIN IN COMPLEX WITH A INHIBITOR (+-)-N1-{TRANS-4'-[(6"-AMINO-4"-METHYLPYRIDIN-2"-YL) METHYL]PYRROLIDIN-3'-YL}-N2-(3'-CHLOROBENZYL)ETHANE-1,2-DIAMINE | NITRIC OXIDE SYNTHASE HEME ENZYME INHIBITOR, BLOOD COAGULATION, CALMODULIN-BINDING, CYTOSKELETON, FAD, FMN, GOLGI APPARATUS, HEME, IRON, LIPOPROTEIN, MEMBRANE, METAL-BINDING, MYRISTATE, NADP, OXIDOREDUCTASE, PALMITATE, PHOSPHOPROTEIN
4u6p:B (ARG454) to (SER514) STRUCTURAL MECHANISM OF ERROR-FREE BYPASS OF MAJOR BENZO[A]PYRENE ADDUCT BY HUMAN POLYMERASE KAPPA | BENZO[A]PYRENE-N2-GUANINE, DNA REPLICATION, DNA DAMAGE TOLERANCE, POLYMERASE KAPPA, ENVIRONMENT POLLUTION, TRANSFERASE-DNA COMPLEX
4dk5:A (ILE222) to (VAL282) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH A PYRIDYL- TRIAZINE INHIBITOR | PHOSPHOTRANSFERASE, CANCER, P85-ALPHA, P85-BETA, RAS, TRANSFERASE- INHIBITOR COMPLEX
4u7c:A (ARG454) to (SER514) STRUCTURE OF DNA POLYMERASE KAPPA IN COMPLEX WITH BENZOPYRENE ADDUCTED DNA | BENZO[A]PYRENE-N2-GUANINE, DNA REPLICATION, DNA DAMAGE TOLERANCE, POLYMERASE KAPPA, ENVIRONMENT POLLUTION, TRANSFERASE-DNA COMPLEX
4u7c:B (ARG454) to (SER514) STRUCTURE OF DNA POLYMERASE KAPPA IN COMPLEX WITH BENZOPYRENE ADDUCTED DNA | BENZO[A]PYRENE-N2-GUANINE, DNA REPLICATION, DNA DAMAGE TOLERANCE, POLYMERASE KAPPA, ENVIRONMENT POLLUTION, TRANSFERASE-DNA COMPLEX
4uh7:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)PHENYL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4uh7:B (LEU250) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)PHENYL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4uh8:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(5-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)PYRIDIN-3-YL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4uh8:B (LEU250) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(5-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)PYRIDIN-3-YL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4uh9:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)-5-FLUOROPHENYL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4uh9:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N1-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2- YL)ETHYL)-5-FLUOROPHENYL)-N1,N2-DIMETHYLETHANE-1,2-DIAMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4uha:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 3-(2-(6-AMINO-4-METHYLPYRIDIN-2-YL) ETHYL)-5-(METHYL(2-(METHYLAMINO)ETHYL)AMINO)BENZONITRILE | OXIDOREDUCTASE, INHIBITOR COMPLEX
3phx:B (GLU80) to (ASP133) OTU DOMAIN OF CRIMEAN CONGO HEMORRHAGIC FEVER VIRUS IN COMPLEX WITH ISG15 | OTU DOMAIN, DE-UBIQUITINASE, DE-ISGYLASE, HYDROLASE-PROTEIN BINDING COMPLEX
3pnh:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(((3R,4R)-4-(2-((2-FLUORO-2-(3-FLUOROPHENYL) ETHYL) AMINO)ETHOXY)PYRROLIDIN-3-YL)METHYL)-4-METHYLPYRIDIN-2-AMINE | HEME ENZYME, INHIBITOR, OXIDOREDUCTASE-INHIBITOR COMPLEX
3pnh:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 6-(((3R,4R)-4-(2-((2-FLUORO-2-(3-FLUOROPHENYL) ETHYL) AMINO)ETHOXY)PYRROLIDIN-3-YL)METHYL)-4-METHYLPYRIDIN-2-AMINE | HEME ENZYME, INHIBITOR, OXIDOREDUCTASE-INHIBITOR COMPLEX
4upq:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N',N'-{[(2R)-3-AMINOPROPANE-1,2-DIYL] BIS(OXYMETHANEDIYLBENZENE-3,1-DIYL)}DITHIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4upr:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N,N''-{[(2S)-3-AMINOPROPANE-1,2-DIYL] BIS(OXYMETHANEDIYLBENZENE-3,1-DIYL)}DITHIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4upr:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N,N''-{[(2S)-3-AMINOPROPANE-1,2-DIYL] BIS(OXYMETHANEDIYLBENZENE-3,1-DIYL)}DITHIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4upt:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N'-[4-[[(2S,4R)-4-[3-[(C-THIOPHEN-2- YLCARBONIMIDOYL)AMINO]PHENOXY]PYRROLIDIN-2- YL]METHOXY]PHENYL]THIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4upt:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N'-[4-[[(2S,4R)-4-[3-[(C-THIOPHEN-2- YLCARBONIMIDOYL)AMINO]PHENOXY]PYRROLIDIN-2- YL]METHOXY]PHENYL]THIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4ups:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-[3-({[(3S,5S)-5-{[(3-{[(Z)-IMINO (THIOPHEN-2-YL)METHYL]AMINO}BENZYL)OXY]METHYL}PYRROLIDIN-3 -YL]OXY}METHYL)PHENYL]THIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4ups:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-[3-({[(3S,5S)-5-{[(3-{[(Z)-IMINO (THIOPHEN-2-YL)METHYL]AMINO}BENZYL)OXY]METHYL}PYRROLIDIN-3 -YL]OXY}METHYL)PHENYL]THIOPHENE-2-CARBOXIMIDAMIDE | OXIDOREDUCTASE, INHIBITOR COMPLEX
3pre:A (ASN218) to (LEU281) QUINAZOLINES WITH INTRA-MOLECULAR HYDROGEN BONDING SCAFFOLD (IMHBS) AS PI3K/MTOR DUAL INHIBITORS. | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
5io9:A (MET132) to (SER210) X-RAY STRUCURE OF THE N-TERMINAL DOMAIN OF HUMAN DOUBLECORTIN | DCX DOMAIN, UBIQUITIN-LIKE FOLD, MICROTUBULE ASSOCIATED, SIGNALING PROTEIN, TRANSFERASE
3pzd:A (GLN1698) to (ALA1754) STRUCTURE OF THE MYOSIN X MYTH4-FERM/DCC COMPLEX | PROTEIN-PROTEIN COMPLEX, MYTH4 DOMAIN, FERM DOMAIN, CARGO BINDING, MOTOR PROTEIN-APOPTOSIS COMPLEX
3q3j:A (LYS1498) to (ASP1567) CRYSTAL STRUCTURE OF PLEXIN A2 RBD IN COMPLEX WITH RND1 | RAS-BINDING DOMAIN, PLEXIN, SMALL GTPASE, STRUCTURAL GENOMICS CONSORTIUM, SGC, MEMBRANE PROTEIN-PROTEIN BINDING COMPLEX
3q7x:A (GLU11) to (SER58) CRYSTAL STRUCTURE OF SYMFOIL-4P/PV1: DE NOVO DESIGNED BETA-TREFOIL ARCHITECTURE WITH SYMMETRIC PRIMARY STRUCTURE, PRIMITIVE VERSION 1 | BETA-TREFOIL, BETA-TERFOIL, DE NOVO PROTEIN
4ezj:A (ASN218) to (VAL282) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4ezk:A (ASN218) to (VAL282) POTENT AND SELECTIVE INHIBITORS OF PI3K-DELTA: OBTAINING ISOFORM SELECTIVITY FROM THE AFFINITY POCKET AND TRYPTOPHAN SHELF | KINASE P110, P110-GAMMA, LIPID KINASE, CYTOPLASMIC, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4f1s:A (ILE220) to (VAL282) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH A PYRIDYL- TRIAZINE-SULFONAMIDE INHIBITOR | PHOSPHOTRANSFERASE, LIPID KINASE, P85, TRANSFERASE-INHIBITOR COMPLEX
5j18:A (PRO155) to (GLY209) SOLUTION STRUCTURE OF RAS BINDING DOMAIN (RBD) OF B-RAF COMPLEXED WITH RIGOSERTIB (COMPLEX I) | MAPK, PI3K, PROTEIN BINDING
3qij:A (HIS211) to (ASP266) PRIMITIVE-MONOCLINIC CRYSTAL STRUCTURE OF THE FERM DOMAIN OF PROTEIN 4.1R | CYTOSKELETON, STRUCTURAL GENOMICS, STRUCTURAL GENOMICS CONSORTIUM, SGC, STRUCTURAL PROTEIN
5j7t:A (HIS683) to (ILE746) MOLECULAR UNDERSTANDING OF USP7 SUBSTRATE RECOGNITION AND C-TERMINAL ACTIVATION | USP7, HAUSP, DUB, ACTIVATION, HYDROLASE
4fa6:A (ASN218) to (VAL282) DESIGN AND SYNTHESIS OF A NOVEL PYRROLIDINYL PYRIDO PYRIMIDINONE DERIVATIVE AS A POTENT INHIBITOR OF PI3KA AND MTOR | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4fad:A (ILE222) to (VAL282) DESIGN AND SYNTHESIS OF A NOVEL PYRROLIDINYL PYRIDO PYRIMIDINONE DERIVATIVE AS A POTENT INHIBITOR OF PI3KA AND MTOR | PHOSPHOINOSITIDE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4v0i:A (ASN187) to (TYR251) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
4v0i:B (SER186) to (TYR251) WATER NETWORK DETERMINES SELECTIVITY FOR A SERIES OF PYRIMIDONE INDOLINE AMIDE PI3KBETA INHIBITORS OVER PI3K-DELTA | TRANSFERASE, PI3K, KINASE SELECTIVITY
3qx1:A (GLU571) to (THR625) CRYSTAL STRUCTURE OF FAF1 UBX DOMAIN | UBX, PROTEIN BINDING, P97 BINDING
4flh:A (ILE220) to (VAL282) CRYSTAL STRUCTURE OF HUMAN PI3K-GAMMA IN COMPLEX WITH AMG511 | P110, PHOSPHOTRANSFERASE, CANCER, P85, PHOSPHORYLATION, TRANSFERASE- INHIBITOR COMPLEX
3r66:D (GLU80) to (ASP133) CRYSTAL STRUCTURE OF HUMAN ISG15 IN COMPLEX WITH NS1 N-TERMINAL REGION FROM INFLUENZA VIRUS B, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET IDS HX6481, HR2873, AND OR2 | STRUCTURAL GENOMICS, PSI-BIOLOGY, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, INNATE IMMUNITY, ISG15 CONJUGATION, VIRAL PROTEIN- ANTIVIRAL PROTEIN COMPLEX
4gb9:A (ASN218) to (VAL282) POTENT AND HIGHLY SELECTIVE BENZIMIDAZOLE INHIBITORS OF PI3K-DELTA | KINASE P110 GAMMA-ISOFORM, KINASE, LIPID KINASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
5kho:B (GLY146) to (VAL228) RASIP1 RA DOMAIN IN COMPLEX WITH RAP1B | RASIP1, RAS-ASSOCIATION DOMAIN, RAP1B, COMPLEX, SIGNALING PROTEIN
5khq:B (GLY146) to (GLY230) RASIP1 RA DOMAIN | RASIP1, RAS-ASSOCIATION DOMAIN, RAP EFFECTOR, SIGNALING PROTEIN
5kz6:B (GLY230) to (ARG273) 1.25 ANGSTROM CRYSTAL STRUCTURE OF CHITINASE FROM BACILLUS ANTHRACIS. | CHITINASE, TIM BARREL, HYDROLASE, STRUCTURAL GENOMICS, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, CSGID
5lrv:B (MET1) to (ASP52) STRUCTURE OF CEZANNE/OTUD7B OTU DOMAIN BOUND TO LYS11-LINKED DIUBIQUITIN | HYDROLASE, PROTEASE, DEUBIQUITINASE, OTU DOMAIN
6nse:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, H4B-FREE, CANAVANINE COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
8nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, NNA COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
9nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, ETHYL-ISOSELENOUREA COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
3ene:A (ASN218) to (VAL282) COMPLEX OF PI3K GAMMA WITH AN INHIBITOR | LIPID KINASE, PHOSPHOINOSITIDE, INHIBITOR, 3-KINASE, SIGNALING, PYRAZOLOPYRIMIDINE, PIK-208, S2, KINASE, TRANSFERASE
2bhj:A (TYR261) to (GLU314) MURINE INO SYNTHASE WITH COUMARIN INHIBITOR | INOS, CALMODULIN-BINDING, FAD, FMN, HEME, METAL-BINDING, NADP, OXIDOREDUCTASE, POLYMORPHISM, ZINC
1d1y:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 1, 3-PBITU (H4B FREE) | ALPHA-BETA FOLD, OXIDOREDUCTASE
1p6l:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NOS HEME DOMAIN WITH L-N(OMEGA)-NITROARGININE-2,4- L-DIAMINOBUTYRIC AMIDE BOUND | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE, HEME-ENZYME
1q1o:A (GLY760) to (GLY829) SOLUTION STRUCTURE OF THE PB1 DOMAIN OF CDC24P (LONG FORM) | PB1 DOMAIN, PCCR, PC MOTIF, OPCA MOTIF, YEAST, CELL POLARITY, PROTEIN-PROTEIN INTERACTION, SIGNALING PROTEIN
1e8z:A (ASN218) to (VAL282) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | TRANSFERASE, PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, STAUROSPORINE
1e90:A (ASN218) to (VAL282) STRUCTURE DETERMINANTS OF PHOSPHOINOSITIDE 3-KINASE INHIBITION BY WORTMANNIN, LY294002, QUERCETIN, MYRICETIN AND STAUROSPORINE | PHOSPHOINOSITIDE 3-KINASE GAMMA, SECONDARY MESSENGER GENERATION, PI3K, PI 3K, MYRICETIN
2dhz:A (SER6) to (GLN71) SOLUTION STRUCTURE OF THE RA DOMAIN IN THE HUMAN LINK GUANINE NUCLEOTIDE EXCHANGE FACTOR II (LINK-GEFII) | LINK GUANINE NUCLEOTIDE EXCHANGE FACTOR II, LINK-GEFII, RA DOMAIN, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, SIGNALING PROTEIN
3tl5:A (ASN218) to (VAL282) DISCOVERY OF GDC-0980: A POTENT, SELECTIVE, AND ORALLY AVAILABLE CLASS I PHOSPHATIDYLINOSITOL 3-KINASE (PI3K)/MAMMALIAN TARGET OF RAPAMYCIN (MTOR) KINASE INHIBITOR FOR THE TREATMENT OF CANCER | TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2uwq:A (MET2) to (ASP58) SOLUTION STRUCTURE OF ASPP2 N-TERMINUS | ASPP2, UBIQUITIN-LIKE, SH3-DOMAIN, APOPTOSIS, CELL CYCLE, ANK REPEAT, SH3-BINDING
4kcq:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(4-(2-(ETHYL(3-(THIOPHENE-2-CARBOXIMIDAMIDO)BENZYL) AMINO)ETHYL)PHENYL)THIOPHENE-2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4kcq:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(4-(2-(ETHYL(3-(THIOPHENE-2-CARBOXIMIDAMIDO)BENZYL) AMINO)ETHYL)PHENYL)THIOPHENE-2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
4kcr:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH N-(3-(((3-FLUOROPHENETHYL)AMINO)METHYL)PHENYL)THIOPHENE- 2-CARBOXIMIDAMIDE | NITRIC OXIDE SYNTHASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
2wxo:A (ASN187) to (TYR251) THE CRYSTAL STRUCTURE OF THE MURINE CLASS IA PI 3-KINASE P110DELTA IN COMPLEX WITH AS5. | TRANSFERASE, PHOSPHOPROTEIN, ISOFORM-SPECIFIC INHIBITORS, CANCER
2jy6:A (ILE3) to (ASP52) SOLUTION STRUCTURE OF THE COMPLEX OF UBIQUITIN AND UBIQUILIN 1 UBA DOMAIN | UBIQUILIN, UBA, UBIQUITIN, COMPLEX, ALTERNATIVE SPLICING, CYTOPLASM, NUCLEUS, PHOSPHOPROTEIN, PROTEASOME, SIGNALING PROTEIN
2kde:C (ILE79) to (ASP128) NMR STRUCTURE OF MAJOR S5A (196-306):K48 LINKED DIUBIQUITIN SPECIES | PROTEIN COMPLEX, UBIQUITIN INTERACTING MOTIFS, CYTOPLASM, NUCLEUS, UBL CONJUGATION, ALTERNATIVE SPLICING, PHOSPHOPROTEIN, PROTEASOME, PROTEIN BINDING
4nkx:D (VAL37) to (HIS78) HUMAN STEROIDOGENIC CYTOCHROME P450 17A1 MUTANT A105L WITH SUBSTRATE PROGESTERONE | HEME PROTEIN, MONOOXYGENASE, STEROID 17ALPHA-HYDROXYLASE, STEROID C17,20 LYASE, NADPH-CYTOCHROME P450 REDUCTASE, CYTOCHROME B5, ENDOPLASMIC RETICULUM MEMBRANE, OXIDOREDUCTASE, LYASE
2mbh:A (ILE3) to (ASP52) NMR STRUCTURE OF EKLF(22-40)/UBIQUITIN COMPLEX | PROTEIN-PROTEIN COMPLEX, EKLF, UBIQUITIN, UIM/MIU, TRANSCRIPTION FACTOR TAD, TRANSCRIPTION
3zw3:A (ASN218) to (VAL282) FRAGMENT BASED DISCOVERY OF A NOVEL AND SELECTIVE PI3 KINASE INHIBITOR | TRANSFERASE
3jww:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-[(3'S,4'S)-4'-((6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL) PYRROLIDIN-3'-YL]-N2- (3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3jww:B (ALA254) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-[(3'S,4'S)-4'-((6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL) PYRROLIDIN-3'-YL]-N2- (3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3jx4:B (TYR482) to (GLN535) STRUCTURE OF RAT NEURONAL NITRIC OXIDE SYNTHASE D597N/M336V MUTANT HEME DOMAIN IN COMPLEX WITH N1-{(3'R,4'S)-4'-[(6"-AMINO-4"- METHYLPYRIDIN-2"-YL)METHYL]PYRROLIDIN-3'-YL}-N2-(3'-FLUOROPHENETHYL) ETHANE-1,2-DIAMINE | HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
2zcb:A (MET1) to (ASP52) CRYSTAL STRUCTURE OF UBIQUITIN P37A/P38A | UB-FOLD, CYTOPLASM, NUCLEUS, PHOSPHORYLATION, UBL CONJUGATION, SIGNALING PROTEIN
2zcb:B (MET1) to (ASP52) CRYSTAL STRUCTURE OF UBIQUITIN P37A/P38A | UB-FOLD, CYTOPLASM, NUCLEUS, PHOSPHORYLATION, UBL CONJUGATION, SIGNALING PROTEIN
4ovv:A (ILE20) to (ASP84) CRYSTAL STRUCTURE OF PI3KALPHA IN COMPLEX WITH DIC4-PIP2 | P110, P85, PI3KCA, PI3K, PIK3R1, PHOSPHATIDILYNOSITOL 3, 4, 5 TRIPHOSPHATE, PIP2, PHOSPHATIDYLINOSITOL 4, 5 BISPHOSPHATE, LIPID KINASE, PHOSPHOINOSITIDE, 3-KINASE, SIGNALING, PHOSPHATIDYLINOSITOL 3-KINASE, TRANSFERASE-TRANSFERASE REGULATOR COMPLEX
4aj3:A (ARG96) to (GLU154) 3D STRUCTURE OF E. COLI ISOCITRATE DEHYDROGENASE IN COMPLEX WITH ISOCITRATE, CALCIUM(II) AND NADP - THE PSEUDO-MICHAELIS COMPLEX | OXIDOREDUCTASE, OXIDATIVE BETA-DECARBOXYLATION
3l16:A (ASN218) to (LEU281) DISCOVERY OF (THIENOPYRIMIDIN-2-YL)AMINOPYRIMIDINES AS POTENT, SELECTIVE, AND ORALLY AVAILABLE PAN-PI3-KINASE AND DUAL PAN-PI3- KINASE/MTOR INHIBITORS FOR THE TREATMENT OF CANCER | KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, PI3K-GAMMA P110 GAMMA
5e6p:A (PRO1466) to (ASP1532) PLEXINB2 CYTOPLASMIC REGION/PDZ-RHOGEF PDZ DOMAIN COMPLEX | PLEXIN, PDZ, PDZ-RHOGEF, COMPLEX, SIGNALING PROTEIN
3n13:A (GLY230) to (ARG273) CRYSTAL STRICTURE OF D143A CHITINASE IN COMPLEX WITH NAG FROM BACILLUS CEREUS NCTU2 | CHITINASE, CHINCTU2, COMPLEX, NAG, MUTATION, HYDROLASE
3n5p:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 4-(2-(6-(2-(6-AMINO-4-METHYLPYRIDIN-2-YL)ETHYL)PYRIDIN-2-YL) ETHYL)-6-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n67:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE N368D/V106M DOUBLE MUTANT HEME DOMAIN COMPLEXED WITH 6,6'-(2,2'-(5-AMINO-1,3-PHENYLENE) BIS(ETHANE-2,1-DIYL))BIS(4-METHYLPYRIDIN-2-AMINE) | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3n68:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN N368D/V106M DOUBLE MUTANT COMPLEXED WITH 4-(3-(2-(6-AMINO-4-METHYLPYRIDIN-2-YL) ETHYL)PHENETHYL)-6-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR COMPLEX
3nld:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'S,4'S)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nle:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'R)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nle:B (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH 6-{{(3'R,4'R)-3'-[2"-(3'''-FLUOROPHENETHYLAMINO) ETHOXY]PYRROLIDIN-4'-YL}METHYL}-4-METHYLPYRIDIN-2-AMINE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
3nlt:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN COMPLEXED WITH N1-{(3'S,4'S)-4'-[(6"-AMINO-4"-METHYLPYRIDIN-2"-YL) METHYL]PYRROLIDIN-3'-YL}- N2-(3'-FLUOROPHENETHYL)ETHANE-1,2-DIAMINE TETRAHYDROCHLORIDE | NITRIC OXIDE SYNTHASE, HEME ENZYME, SUBSTRATE INHIBITOR, OXIDOREDUCTASE
4cwv:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-((5-(PYRIDIN- 2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL)PYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cwv:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-((5-(PYRIDIN- 2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL)PYRIDIN-2-AMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4cwz:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE Y477A MUTANT HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-( (5-(4-METHYLPYRIDIN-2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL) PYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4cwz:B (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE Y477A MUTANT HEME DOMAIN IN COMPLEX WITH 4-METHYL-6-(((3R,4R)-4-( (5-(4-METHYLPYRIDIN-2-YL)PENTYL)OXY)PYRROLIDIN-3-YL)METHYL) PYRIDIN-2-AMINE | OXIDOREDUCTASE, INHIBITOR COMPLEX
4tv3:A (GLY188) to (GLU263) ISOLATED P110A SUBUNIT OF PI3KA PROVIDES A PLATFORM FOR STRUCTURE- BASED DRUG DESIGN | LIPID KINASE ACTIVITY, ATPASE ACTIVITY, SURFACE PLASMON RESONANCE (SPR), ISOTHERMAL TITRATION CALORIMETRY (ITC)., TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4d38:A (TYR253) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (1R,2R)-2-(3-FLUOROBENZYL)-N-{2-[2- (1H-IMIDAZOL-1-YL)PYRIMIDIN-4-YL]ETHYL}CYCLOPROPANAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
4d38:B (ALA254) to (VAL306) STRUCTURE OF BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE HEME DOMAIN IN COMPLEX WITH (1R,2R)-2-(3-FLUOROBENZYL)-N-{2-[2- (1H-IMIDAZOL-1-YL)PYRIMIDIN-4-YL]ETHYL}CYCLOPROPANAMINE | OXIDOREDUCTASE, NITRIC OXIDE SYNTHASE, INHIBITOR COMPLEX
3dqs:A (TYR253) to (VAL306) STRUCTURE OF ENDOTHELIAL NOS HEME DOMAIN IN COMPLEX WITH A INHIBITOR (+-)-N1-{CIS-4'-[(6"-AMINO-4"-METHYLPYRIDIN-2"-YL)METHYL]PYRROLIDIN- 3'-YL}-N2-(4'-CHLOROBENZYL)ETHANE-1,2-DIAMINE | NITRIC OXIDE SYNTHASE HEME ENZYME INHIBITOR, BLOOD COAGULATION, CALMODULIN-BINDING, CYTOSKELETON, FAD, FMN, GOLGI APPARATUS, HEME, IRON, LIPOPROTEIN, MEMBRANE, METAL-BINDING, MYRISTATE, NADP, OXIDOREDUCTASE, PALMITATE, PHOSPHOPROTEIN
5j17:A (PRO155) to (GLY209) SOLUTION STRUCTURE OF RAS BINDING DOMAIN (RBD) OF B-RAF | MAPK, PI3K, PROTEIN BINDING
4fhj:A (ASN218) to (VAL282) CRYSTAL STRUCTURE OF PI3K-GAMMA IN COMPLEX WITH IMIDAZOPYRIDINE 2 | INHIBITOR, P110, KINASE, TRANSFERASE, ATP-BINDING, P84, P101, TRANSFERASE-INHIBITOR COMPLEX
5jtv:E (ARG892) to (GLU955) USP7CD-UBL45 IN COMPLEX WITH UBIQUITIN | USP7, HAUSP, C-TERMINAL ACTIVATION, HYDROLASE
5jtv:G (ARG892) to (GLU955) USP7CD-UBL45 IN COMPLEX WITH UBIQUITIN | USP7, HAUSP, C-TERMINAL ACTIVATION, HYDROLASE
5l72:A (ARG188) to (TYR251) PI3 KINASE DELTA IN COMPLEX WITH N-[6-(5-METHANESULFONAMIDO-6- METHOXYPYRIDIN-3-YL)-1,3-DIHYDRO-2-BENZOFURAN-4-YL]-2-(MORPHOLIN-4- YL)ACETAMIDE | PI3 KINASE DELTA, TRANSFERASE
5nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, H4B-FREE, HYDROXY-ARG COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
7nse:A (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, H4B-FREE, ADMA COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE
7nse:B (TYR253) to (VAL306) BOVINE ENDOTHELIAL NITRIC OXIDE SYNTHASE, H4B-FREE, ADMA COMPLEX | NITRIC OXIDE SYNTHASE, HEME PROTEIN, TETRAHYDROBIOPTERIN, OXIDOREDUCTASE