2o8t:A (PHE30) to (GLU84) CRYSTAL STRUCTURE AND BINDING EPITOPES OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR (C122A/N145Q) IN COMPLEX WITH INHIBITORS | UROKINASE-TYPE PLASMINOGEN ACTIVATOR, BENZAMIDINE, PHENYLGUANIDINE, CONTACT AREA, HYDROLASE
1n8s:A (HIS354) to (ALA417) STRUCTURE OF THE PANCREATIC LIPASE-COLIPASE COMPLEX | HYDROLASE, PANCREAS, SIGNAL
1a3b:H (GLN30) to (MET84) COMPLEX OF HUMAN ALPHA-THROMBIN WITH THE BIFUNCTIONAL BORONATE INHIBITOR BOROLOG1 | COMPLEX (SERINE PROTEASE-INHIBITOR), HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a3e:H (GLN30) to (MET84) COMPLEX OF HUMAN ALPHA-THROMBIN WITH THE BIFUNCTIONAL BORONATE INHIBITOR BOROLOG2 | COMPLEX (SERINE PROTEASE-INHIBITOR), HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a46:H (GLN30) to (MET84) THROMBIN COMPLEXED WITH HIRUGEN AND A BETA-STRAND MIMETIC INHIBITOR | COMPLEX (SERINE PROTEASE-INHIBITOR), HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a5g:H (GLN30) to (MET84) HUMAN THROMBIN COMPLEXED WITH NOVEL SYNTHETIC PEPTIDE MIMETIC INHIBITOR AND HIRUGEN | COMPLEX (SERINE PROTEASE-INHIBITOR),HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a5h:B (TRP29) to (GLU84) CATALYTIC DOMAIN OF HUMAN TWO-CHAIN TISSUE PLASMINOGEN ACTIVATOR COMPLEX OF A BIS-BENZAMIDINE | TRYPSIN LIKE SERINE PROTEASE, FIBRINOLYTIC ENZYME, HYDROLASE
1nc6:A (GLN30) to (SER84) POTENT, SMALL MOLECULE INHIBITORS OF HUMAN MAST CELL TRYPTASE. ANTI-ASTHMATIC ACTION OF A DIPEPTIDE-BASED TRANSITION STATE ANALOGUE CONTAINING BENZOTHIAZOLE KETONE | PROTEIN-INHIBITOR COMPLEX, HYDROLASE
3eaj:A (VAL18) to (ILE78) CRYSTAL STRUCTURE OF SARS-COV MAIN PROTEASE QUADRUPLE MUTANT STIF/A WITH TWO MOLECULES IN ONE ASYMMETRIC UNIT | SARS CORONAVIRUS MAIN PROTEASE MUTANT EXTRA HELICAL DOMAIN, CYTOPLASM, HYDROLASE, MEMBRANE, METAL-BINDING, PROTEASE, RIBOSOMAL FRAMESHIFTING, RNA-BINDING, THIOL PROTEASE, TRANSMEMBRANE, ZINC, ZINC-FINGER
1a7s:A (LEU15) to (SER72) ATOMIC RESOLUTION STRUCTURE OF HBP | SERINE PROTEASE HOMOLOG, ENDOTOXIN BINDING, HEPARIN
1a8i:A (LEU198) to (THR240) SPIROHYDANTOIN INHIBITOR OF GLYCOGEN PHOSPHORYLASE | GLYCOGEN PHOSPHORYLASE, GLUCOPYRANOSE SPIROHYDANTOIN, WATER STRUCTURE, INHIBITOR BINDING, ANTI-HYPERGLYCEMIC AGENT
2ank:H (GLN30) to (MET84) ORALLY ACTIVE THROMBIN INHIBITORS IN COMPLEX WITH THROMBIN AND AN EXOSITE DECAPEPTIDE | BLOOD CLOTTING, HYDROLASE, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3rp2:B (MET30) to (LYS84) THE STRUCTURE OF RAT MAST CELL PROTEASE II AT 1.9-ANGSTROMS RESOLUTION | SERINE PROTEINASE
1ab9:B (GLN30) to (LYS84) CRYSTAL STRUCTURE OF BOVINE GAMMA-CHYMOTRYPSIN | HYDROLASE, SERINE PROTEASE, DIGESTION, PANCREAS, ZYMOGEN, COMPLEX (SERINE PROTEASE/PEPTIDE)
2ok5:A (TRP470) to (HIS531) HUMAN COMPLEMENT FACTOR B | PRO-ENZYME, SERINE PROTEASE DOMAIN,VON WILLEBRAND FACTOR-A DOMAIN, CCP DOMAIN, HYDROLASE
1acb:E (GLN30) to (LYS84) CRYSTAL AND MOLECULAR STRUCTURE OF THE BOVINE ALPHA-CHYMOTRYPSIN-EGLIN C COMPLEX AT 2.0 ANGSTROMS RESOLUTION | SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2auk:E (SER18) to (LYS57) STRUCTURE OF E. COLI RNA POLYMERASE BETA' G/G' INSERT | SANDWICH-BARREL HYBRID MOTIF, TRANSFERASE
3ee7:A (CYS14) to (GLU68) CRYSTAL STRUCTURE OF SARS-COV NSP9 G104E | GXXXG, DIMERIZATION, SARS-COV, HELIX-HELIX, HYDROLASE, MEMBRANE, METAL-BINDING, PROTEASE, RNA-BINDING, THIOL PROTEASE, TRANSMEMBRANE, ZINC-FINGER, VIRAL PROTEIN
3ee7:D (CYS14) to (GLU68) CRYSTAL STRUCTURE OF SARS-COV NSP9 G104E | GXXXG, DIMERIZATION, SARS-COV, HELIX-HELIX, HYDROLASE, MEMBRANE, METAL-BINDING, PROTEASE, RNA-BINDING, THIOL PROTEASE, TRANSMEMBRANE, ZINC-FINGER, VIRAL PROTEIN
1afe:H (GLN30) to (MET84) HUMAN ALPHA-THROMBIN INHIBITION BY CBZ-PRO-AZALYS-ONP | COMPLEX (SERINE PROTEASE-INHIBITOR), BLOOD COAGULATION, N- CARBOBENZOXY-PRO-ALFA-AZALYS-P-NITROPHENYLESTER, SERINE PROTEINASE INHIBITION, GLYCOSYLATED PROTEIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1afq:B (GLN30) to (LYS84) CRYSTAL STRUCTURE OF BOVINE GAMMA-CHYMOTRYPSIN COMPLEXED WITH A SYNTHETIC INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1aht:H (GLN30) to (MET84) CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN COMPLEXED WITH HIRUGEN AND P-AMIDINOPHENYLPYRUVATE AT 1.6 ANGSTROMS RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1nm6:A (GLN30) to (MET84) THROMBIN IN COMPLEX WITH SELECTIVE MACROCYCLIC INHIBITOR AT 1.8A | THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
1aks:A (GLN30) to (ASN84) CRYSTAL STRUCTURE OF THE FIRST ACTIVE AUTOLYSATE FORM OF THE PORCINE ALPHA TRYPSIN | HYDROLASE, SERINE PROTEASE
1amh:B (GLN30) to (ASN84) UNCOMPLEXED RAT TRYPSIN MUTANT WITH ASP 189 REPLACED WITH SER (D189S) | SERINE PROTEASE, ACTIVATION DOMAIN, SUBSTRATE SPECIFICITY HYDROLASE
1ao5:A (GLN30) to (LYS87) MOUSE GLANDULAR KALLIKREIN-13 (PRORENIN CONVERTING ENZYME) | GLANDULAR KALLIKREIN, SERINE PROTEASE, PROTEIN MATURATION
1ao5:B (GLN30) to (LEU84) MOUSE GLANDULAR KALLIKREIN-13 (PRORENIN CONVERTING ENZYME) | GLANDULAR KALLIKREIN, SERINE PROTEASE, PROTEIN MATURATION
2oqu:A (GLN15) to (GLY73) HIGH PRESSURE CRYOCOOLING OF CAPILLARY SAMPLE CRYOPROTECTION AND DIFFRACTION PHASING AT LONG WAVELENGTHS | HIGH PRESSURE CRYOCOOLING, XENON, SAD PHASING, HYDROLASE
4h4f:A (GLN30) to (VAL85) CRYSTAL STRUCTURE OF HUMAN CHYMOTRYPSIN C (CTRC) BOUND TO INHIBITOR EGLIN C FROM HIRUDO MEDICINALIS | SERINE PROTEASE, PROTEASE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1nrn:H (GLN30) to (MET84) CRYSTALLOGRAPHIC STRUCTURES OF THROMBIN COMPLEXED WITH THROMBIN RECEPTOR PEPTIDES: EXISTENCE OF EXPECTED AND NOVEL BINDING MODES | SERINE PROTEINASE/RECEPTOR
1nrq:H (GLN30) to (MET84) CRYSTALLOGRAPHIC STRUCTURES OF THROMBIN COMPLEXED WITH THROMBIN RECEPTOR PEPTIDES: EXISTENCE OF EXPECTED AND NOVEL BINDING MODES | SERINE PROTEINASE, RECEPTOR, HYDROLASE/HYDROLASE RECEPTOR COMPLEX
1nrr:H (GLN30) to (MET84) CRYSTALLOGRAPHIC STRUCTURES OF THROMBIN COMPLEXED WITH THROMBIN RECEPTOR PEPTIDES: EXISTENCE OF EXPECTED AND NOVEL BINDING MODES | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, BLOOD CLOTTING
3s0n:A (TYR14) to (GLU71) CRYSTAL STRUCTURE OF HUMAN CHYMASE WITH BENZIMIDAZOLONE INHIBITOR | SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1nt1:A (GLN30) to (MET84) THROMBIN IN COMPLEX WITH SELECTIVE MACROCYCLIC INHIBITOR | THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
3ela:H (GLN167) to (ARG224) CRYSTAL STRUCTURE OF ACTIVE SITE INHIBITED COAGULATION FACTOR VIIA MUTANT IN COMPLEX WITH SOLUBLE TISSUE FACTOR | SERINE PROTEASE, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2b5t:B (GLN30) to (MET84) 2.1 ANGSTROM STRUCTURE OF A NONPRODUCTIVE COMPLEX BETWEEN ANTITHROMBIN, SYNTHETIC HEPARIN MIMETIC SR123781 AND TWO S195A THROMBIN MOLECULES | BLOOD COAGULATION, BLOOD CLOTTING
3ens:D (GLN30) to (GLU84) CRYSTAL STRUCTURE OF HUMAN FXA IN COMPLEX WITH METHYL (2Z)-3-[(3- CHLORO-1H-INDOL-7-YL)AMINO]-2-CYANO-3-{[(3S)-2-OXO-1-(2-OXO-2- PYRROLIDIN-1-YLETHYL)AZEPAN-3-YL]AMINO}ACRYLATE | SERINE PROTEASE, HYDROLASE, EPIDERMAL GROWTH FACTOR LIKE DOMAIN, BLOOD COAGULATION FACTOR, CLEAVAGE ON PAIR OF BASIC RESIDUES, EGF- LIKE DOMAIN, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROXYLATION, ZYMOGEN, BLOOD CLOTTING
1awf:H (GLN30) to (MET84) NOVEL COVALENT THROMBIN INHIBITOR FROM PLANT EXTRACT | PROTEINASE, BLOOD COAGULATION, TRYPSIN LIKE PROTEINASE, COMPLEX (PROTEASE-INHIBITOR), HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ay6:H (GLN30) to (MET84) THROMBIN INHIBITOR FROM THEONALLA, CYCLOTHEANAMIDE-BASED MACROCYCLIC TRIPEPTIDE MOTIF | COMPLEX OF SERINE PROTEASE-INHIBITOR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1azz:A (HIS29) to (THR86) FIDDLER CRAB COLLAGENASE COMPLEXED TO ECOTIN | COMPLEX (SERINE PROTEASE/INHIBITOR), SERINE PROTEASE, INHIBITOR, COMPLEX, PROTEASE-SUBSTRATE INTERACTIONS, COLLAGEN
1b0f:A (MET30) to (ALA84) CRYSTAL STRUCTURE OF HUMAN NEUTROPHIL ELASTASE WITH MDL 101, 146 | SERINE PROTEASE, FLUOROETHYL KETONES, HYDROLASE
1nzq:H (GLN30) to (MET84) D-PHE-PRO-ARG-TYPE THROMBIN INHIBITOR | THROMBIN, THROMBIN INHIBITOR, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2p3f:H (GLN30) to (GLU84) CRYSTAL STRUCTURE OF THE FACTOR XA/NAP5 COMPLEX | FACTOR XA, NEMATODE ANTICOAGULANT PROTEIN, HYDROLASE
4wwy:B (GLN30) to (ASN84) HUMAN CATIONIC TRYPSIN G193R MUTANT IN COMPLEX WITH BOVINE PANCREATIC TRYPSIN INHIBITOR | TRYPSIN INHIBITORS, COMPLEX, BPTI, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4wxk:A (LEU79) to (GLY125) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE | PEPTIDE DEFORMYLASE, HYDROLASE
4wxk:B (ASN75) to (ALA123) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE | PEPTIDE DEFORMYLASE, HYDROLASE
4wxk:C (LEU79) to (GLY125) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE | PEPTIDE DEFORMYLASE, HYDROLASE
4wxl:A (LEU79) to (GLY125) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE COMPLEX WITH ACTINONIN | PEPTIDE DEFORMYLASE, HYDROLASE
4wxl:B (ASN75) to (GLY125) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE COMPLEX WITH ACTINONIN | PEPTIDE DEFORMYLASE, HYDROLASE
4wxl:D (LEU79) to (GLY125) CRYSTAL STRUCTURE OF A PEPTIDE DEFORMYLASE FROM HAEMOPHILUS INFLUENZAE COMPLEX WITH ACTINONIN | PEPTIDE DEFORMYLASE, HYDROLASE
1b5g:H (GLN30) to (MET84) HUMAN THROMBIN COMPLEXED WITH NOVEL SYNTHETIC PEPTIDE MIMETIC INHIBITOR AND HIRUGEN | SERINE PROTEASE-INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2p8o:B (GLN30) to (LYS84) CRYSTAL STRUCTURE OF A BENZOHYDROXAMIC ACID/VANADATE COMPLEX BOUND TO CHYMOTRYPSIN A | PROTEIN-INHIBITOR COMPLEX, HYDROLASE
1ba8:B (GLN30) to (MET84) THROMBIN INHIBITOR WITH A RIGID TRIPEPTIDYL ALDEHYDES | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1bb0:B (GLN30) to (MET84) THROMBIN INHIBITORS WITH RIGID TRIPEPTIDYL ALDEHYDES | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3f1s:B (GLN151) to (LYS203) CRYSTAL STRUCTURE OF PROTEIN Z COMPLEXED WITH PROTEIN Z-DEPENDENT INHIBITOR | PZ, ZPI, COMPLEX, SERPIN, PROTEASE INHIBITOR, PROTEASE, GLYCOPROTEIN, SECRETED, SERINE PROTEASE INHIBITOR, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, EGF-LIKE DOMAIN, GAMMA-CARBOXYGLUTAMIC ACID, HYDROXYLATION, SERINE PROTEASE HOMOLOG, HYDROLASE INHIBITOR- HYDROLASE COMPLEX
1o2g:H (GLN30) to (MET84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, BLOOD CLOTTING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, BLOOD CLOTTING, HYDROLASE-INHIBITOR COMPLEX
1o2i:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2j:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2k:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2l:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2m:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2n:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2q:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2s:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2u:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2v:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2w:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2y:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o30:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o31:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o33:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o34:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o35:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o37:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3a:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3c:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3d:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3f:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3e:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3g:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3i:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3j:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3k:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3l:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3m:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3n:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o59:A (GLN275) to (GLY342) CRYSTAL STRUCTURE OF ALLANTOICASE (YIR029W) FROM SACCHAROMYCES CEREVISIAE AT 2.40 A RESOLUTION | YIR029W, ALLANTOICASE, STRUCTURAL GENOMICS, JCSG, PSI, PROTEIN STRUCTURE INITIATIVE, JOINT CENTER FOR STRUCTURAL GENOMICS, HYDROLASE
1bma:A (GLN30) to (GLY88) BENZYL METHYL AMINIMIDE INHIBITOR COMPLEXED TO PORCINE PANCREATIC ELASTASE | SERINE PROTEASE,METAL-BINDING, PROTEASE, SECRETED, ZYMOGEN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3s69:A (LEU30) to (ASN82) CRYSTAL STRUCTURE OF SAXTHROMBIN | BETA-BARREL, SERINE ENZYMES, FIBRINOGEN BINDING, GLYCOSYLATION, HYDROLASE
4x6n:A (GLN30) to (HIS91) FACTOR XIA IN COMPLEX WITH THE INHIBITOR 1-{(1S)-1-[4-(3-AMINO-1H- INDAZOL-6-YL)-5-CHLORO-1H-IMIDAZOL-2-YL]-2-PHENYLETHYL}-3-[5-CHLORO- 2-(1H-TETRAZOL-1-YL)BENZYL]UREA | SERINE PROTEASE, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2brw:A (SER704) to (PHE746) CRYSTAL STRUCTURE OF STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE FROM 30PERCENT PEGMME. | (ALFA5/ALFA5) BARREL, CELL WALL, LYASE, PEPTIDOGLYCAN-ANCHOR
2brw:B (SER704) to (PHE746) CRYSTAL STRUCTURE OF STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE FROM 30PERCENT PEGMME. | (ALFA5/ALFA5) BARREL, CELL WALL, LYASE, PEPTIDOGLYCAN-ANCHOR
1bsz:B (GLU579) to (GLY624) PEPTIDE DEFORMYLASE AS FE2+ CONTAINING FORM (NATIVE) IN COMPLEX WITH INHIBITOR POLYETHYLENE GLYCOL | COMPLEX(ENZYME-INHIBITOR), HYDROLASE, IRON METALLOPROTEASE, PROTEIN SYNTHESIS
1bth:H (GLN30) to (MET84) STRUCTURE OF THROMBIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR | THROMBIN INHIBITOR, SERINE PROTEINASE KUNITZ-LIKE INHIBITOR, (SERINE PROTEASE/INHIBITOR), COMPLEX (SERINE PROTEASE/INHIBITOR) COMPLEX
1bth:K (GLN30) to (MET84) STRUCTURE OF THROMBIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR | THROMBIN INHIBITOR, SERINE PROTEINASE KUNITZ-LIKE INHIBITOR, (SERINE PROTEASE/INHIBITOR), COMPLEX (SERINE PROTEASE/INHIBITOR) COMPLEX
1btx:A (GLN30) to (SER84) EPISELECTION: NOVEL KI ~NANOMOLAR INHIBITORS OF SERINE PROTEASES SELECTED BY BINDING OR CHEMISTRY ON AN ENZYME SURFACE | TRIPEPTIDEBORONATE ETHYL ESTER INHIBITED, SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1bty:A (GLN30) to (SER84) CRYSTAL STRUCTURE OF BETA-TRYPSIN IN COMPLEX WITH BENZAMIDINE | BENZAMIDINE INHIBITED, HYDROLASE (SERINE PROTEINASE), HYDROLASE
1bu8:A (TYR354) to (ALA417) RAT PANCREATIC LIPASE RELATED PROTEIN 2 | HYDROLASE, LIPID DEGRADATION, PANCREATIC LIPASE
1bwu:Q (GLY52) to (SER100) MANNOSE-SPECIFIC AGGLUTININ (LECTIN) FROM GARLIC (ALLIUM SATIVUM) BULBS COMPLEXED WITH ALPHA-D-MANNOSE | BULB LECTIN, MANNOSE, PLANT PROTEIN
1bx3:A (LEU198) to (THR240) EFFECTS OF COMMONLY USED CRYOPROTECTANTS ON GLYCOGEN PHOSPHORYLASE ACTIVITY AND STRUCTURE | PHOSPHORYLASE, INHIBITOR, CRYOPROTECTANT, MPD, DMSO, CRYOCRYSTALLOGRAPHY, TRANSFERASE
4hsi:D (GLY205) to (HIS248) GLYCOPROTEIN B FROM HERPES SIMPLEX VIRUS TYPE 1, A504P/R505G/Q507G/N511G MUTANT, LOW-PH | VIRAL FUSION PROTEIN, VIRAL ENVELOPE, VIRAL PROTEIN
1c1n:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1o:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1q:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1r:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1s:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1u:H (GLN30) to (MET84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
1c1v:H (GLN30) to (MET84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1w:H (GLN30) to (MET84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, BLOOD CLOTTING,HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1c2e:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2f:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2g:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1c2h:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2i:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2j:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2k:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2l:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c2m:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4xcr:B (GLY41) to (GLN110) MONOMERIC HUMAN CU,ZN SUPEROXIDE DISMUTASE, LOOPS IV AND VII DELETED, APO FORM, MUTANT I35A | OXIDOREDUCTASE
2pks:B (GLN51) to (MET116) THROMBIN IN COMPLEX WITH INHIBITOR | INHIBITOR COMPLEX, THROMBIN INHIBITOR, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2bxu:H (GLN30) to (MET84) DESIGN AND DISCOVERY OF NOVEL, POTENT THROMBIN INHIBITORS WITH A SOLUBILIZING CATIONIC P1-P2-LINKER | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4xde:A (TYR367) to (ALA424) COAGULATION FACTOR XII PROTEASE DOMAIN CRYSTAL STRUCTURE | FACTOR XII, CATALYTIC DOMAIN, ZYMOGENS, HYDROLASE, BLOOD CLOTTING
3se4:A (SER35) to (VAL90) HUMAN IFNW-IFNAR TERNARY COMPLEX | TYPE I INTERFERON SIGNALING COMPLEX, EXTRACELLULAR SPACE, IMMUNE SYSTEM RECEPTOR
4hzh:B (GLN335) to (MET400) STRUCTURE OF RECOMBINANT GLA-DOMAINLESS PROTHROMBIN MUTANT S525A | PROTHROMBIN, KRINGLE, SERINE PROTEASE, COAGULATION, HYDROLASE
1c4v:2 (GLN30) to (MET84) SELECTIVE NON ELECTROPHILIC THROMBIN INHIBITORS WITH CYCLOHEXYL MOIETIES. | COMPLEX (SERINE PROTEASE-INHIBITOR), HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3sep:C (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (S796A) | DYNAMIC LOOP CONFORMATION, SER-796, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN, BETA SUPERSANDWICH, BETA- GALACTOSIDASE, GLYCOSIDASE, HYDROLASE
1c5l:H (GLN30) to (MET84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB- MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
1c5o:H (GLN30) to (MET84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB- MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
1c5q:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c5s:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c5t:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c5v:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c9t:B (GLN30) to (ILE83) COMPLEX OF BDELLASTASIN WITH BOVINE TRYPSIN | COMPLEX (HYDROLASE/INHIBITOR), HYDROLASE, INHIBITOR, ANTISTASIN, PLASMIN, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1c9t:C (GLN30) to (ILE83) COMPLEX OF BDELLASTASIN WITH BOVINE TRYPSIN | COMPLEX (HYDROLASE/INHIBITOR), HYDROLASE, INHIBITOR, ANTISTASIN, PLASMIN, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1c9t:E (GLN30) to (ILE83) COMPLEX OF BDELLASTASIN WITH BOVINE TRYPSIN | COMPLEX (HYDROLASE/INHIBITOR), HYDROLASE, INHIBITOR, ANTISTASIN, PLASMIN, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1ca8:B (GLN30) to (MET84) THROMBIN INHIBITORS WITH RIGID TRIPEPTIDYL ALDEHYDES | SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2ppl:A (GLN372) to (ALA434) HUMAN PANCREATIC LIPASE-RELATED PROTEIN 1 | HYDROLASE, LIPID DEGRADATION, PANCREATIC LIPASE, STRUCTURAL GENOMICS CONSORTIUM, SGC
2pv9:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF MURINE THROMBIN IN COMPLEX WITH THE EXTRACELLULAR FRAGMENT OF MURINE PAR4 | SERINE PROTEASE, HYDROLASE
2pvs:A (TYR355) to (ALA417) STRUCTURE OF HUMAN PANCREATIC LIPASE RELATED PROTEIN 2 MUTANT N336Q | LIPASE, GALACTO LIPIDS HYDROLYSIS, HYDROLASE
1op2:A (LEU30) to (ASN84) CRYSTAL STRUCTURE OF AAV-SP-II, A GLYCOSYLATED SNAKE VENOM SERINE PROTEINASE FROM AGKISTRODON ACUTUS | SNAKE VENOM, SERINE PROTEINASE, GLYCOPROTEIN, AGKISTRODON ACUTUS, HYDROLASE
1cho:F (GLN30) to (LYS84) CRYSTAL AND MOLECULAR STRUCTURES OF THE COMPLEX OF ALPHA- *CHYMOTRYPSIN WITH ITS INHIBITOR TURKEY OVOMUCOID THIRD DOMAIN AT 1.8 ANGSTROMS RESOLUTION | COMPLEX(SERINE PROTEINASE-INHIBITOR)
1op8:B (TYR29) to (MET83) CRYSTAL STRUCTURE OF HUMAN GRANZYME A | GRANZYME A, SERINE PROTEINASE, APOPTOSIS, HYDROLASE
2pyd:A (LEU198) to (THR240) THE CRYSTAL STRUCTURE OF GLYCOGEN PHOSPHORYLASE IN COMPLEX WITH GLUCOSE AT 100 K | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, TRANSFERASE
2pyi:A (LEU198) to (THR240) CRYSTAL STRUCTURE OF GLYCOGEN PHOSPHORYLASE IN COMPLEX WITH GLUCOSYL TRIAZOLEACETAMIDE | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, TRANSFERASE
3fp9:F (PRO98) to (THR154) CRYSTAL STRUCTURE OF INTERN DOMAIN OF PROTEASOME-ASSOCIATED ATPASE, MYCOBACTERIUM TUBERCULOSIS | FIVE STRAND BETA BARREL, HEXAMER, ATP-BINDING, NUCLEOTIDE- BINDING, HYDROLASE, AAA ATPASE, PROTEASOMAL ATPASE
3fp9:I (PRO98) to (THR154) CRYSTAL STRUCTURE OF INTERN DOMAIN OF PROTEASOME-ASSOCIATED ATPASE, MYCOBACTERIUM TUBERCULOSIS | FIVE STRAND BETA BARREL, HEXAMER, ATP-BINDING, NUCLEOTIDE- BINDING, HYDROLASE, AAA ATPASE, PROTEASOMAL ATPASE
3so3:A (GLN30) to (ARG84) STRUCTURES OF FAB-PROTEASE COMPLEXES REVEAL A HIGHLY SPECIFIC NON- CANONICAL MECHANISM OF INHIBITION. | ANTIBODY-PROTEIN, PROTEIN-PROTEIN, PROTEASE INHIBITOR, DISEASE MUTATION, GLYCOPROTEIN, HYDROLASE, MEMBRANE, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
1oss:A (PHE29) to (ARG84) T190P STREPTOMYCES GRISEUS TRYPSIN IN COMPLEX WITH BENZAMIDINE | TRYPSIN, SERINE PROTEASE, MUTANT, HYDROLASE
4ic5:C (VAL103) to (VAL181) CRYSTAL STRUCTURE OF DEG5 | BETS-BARREL, ENDOPEPTIDASE, CALCIUM BINDING, CHLOROPLAST, HYDROLASE
3sti:B (VAL27) to (GLY106) CRYSTAL STRUCTURE OF THE PROTEASE DOMAIN OF DEGQ FROM ESCHERICHIA COLI | SERINE PROTEASE, PDZ DOMAIN, PROTEASE, CHAPERONE, HYDROLASE
1p2n:C (GLN30) to (LYS84) STRUCTURAL CONSEQUENCES OF ACCOMMODATION OF FOUR NON- COGNATE AMINO-ACID RESIDUES IN THE S1 POCKET OF BOVINE TRYPSIN AND CHYMOTRYPSIN | TRYPSIN; CHYMOTRYPSIN; SERINE PROTEINASE; BOVINE PANCREATIC TRYPSIN INHIBITOR; PROTEIN-PROTEIN INTERACTION; NON-COGNATE BINDING; S1 POCKET; PRIMARY SPECIFICITY; CRYSTAL STRUCTURE, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1d4p:B (GLN51) to (MET116) CRYSTAL STRUCTURE OF HUMAN ALPHA THROMBIN IN COMPLEX WITH 5- AMIDINOINDOLE-4-BENZYLPIPERIDINE INHIBITOR | THROMBIN; NONPEPTIDYL INHIBITOR; STRUCTURE-BASED DRUG DESIGN, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1d6w:A (GLN30) to (MET84) STRUCTURE OF THROMBIN COMPLEXED WITH SELECTIVE NON-ELECTROPHILIC INHIBITORS HAVING CYCLOHEXYL MOIETIES AT P1 | HYDROLASE, THROMBIN, THROMBIN INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2cga:A (GLN30) to (LYS84) BOVINE CHYMOTRYPSINOGEN A. X-RAY CRYSTAL STRUCTURE ANALYSIS AND REFINEMENT OF A NEW CRYSTAL FORM AT 1.8 ANGSTROMS RESOLUTION | HYDROLASE(ZYMOGEN)
2cha:B (GLN30) to (LYS84) THE STRUCTURE OF CRYSTALLINE ALPHA-CHYMOTRYPSIN, $V.THE ATOMIC STRUCTURE OF TOSYL-ALPHA-CHYMOTRYPSIN AT 2 ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
2cha:F (GLN30) to (LYS84) THE STRUCTURE OF CRYSTALLINE ALPHA-CHYMOTRYPSIN, $V.THE ATOMIC STRUCTURE OF TOSYL-ALPHA-CHYMOTRYPSIN AT 2 ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
1d9i:A (GLN30) to (MET84) STRUCTURE OF THROMBIN COMPLEXED WITH SELECTIVE NON-ELECTOPHILIC INHIBITORS HAVING CYCLOHEXYL MOIETIES AT P1 | GLOBULAR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1p8v:C (GLN15) to (MET80) CRYSTAL STRUCTURE OF THE COMPLEX OF PLATELET RECEPTOR GPIB-ALPHA AND ALPHA-THROMBIN AT 2.6A | PLATELET GLYCOPROTEIN RECEPTOR, LEUCINE RICH REPEAT DOMAIN, MEMBRANE PROTEIN-HYDROLASE COMPLEX
1p9m:A (GLU133) to (PHE192) CRYSTAL STRUCTURE OF THE HEXAMERIC HUMAN IL-6/IL-6 ALPHA RECEPTOR/GP130 COMPLEX | IG DOMAIN, FOUR HELIX BUNDLE, CYTOKINE, INTERLEUKIN-6, GP130, SIGNALING PROTEIN-CYTOKINE COMPLEX
1ddj:A (GLN576) to (GLU634) CRYSTAL STRUCTURE OF HUMAN PLASMINOGEN CATALYTIC DOMAIN | PLASMINOGEN, CATALYTIC DOMAIN, BLOOD CLOTTING
1ddj:B (GLN576) to (GLU634) CRYSTAL STRUCTURE OF HUMAN PLASMINOGEN CATALYTIC DOMAIN | PLASMINOGEN, CATALYTIC DOMAIN, BLOOD CLOTTING
1ddj:C (GLN576) to (GLU634) CRYSTAL STRUCTURE OF HUMAN PLASMINOGEN CATALYTIC DOMAIN | PLASMINOGEN, CATALYTIC DOMAIN, BLOOD CLOTTING
1ddj:D (GLN576) to (GLU634) CRYSTAL STRUCTURE OF HUMAN PLASMINOGEN CATALYTIC DOMAIN | PLASMINOGEN, CATALYTIC DOMAIN, BLOOD CLOTTING
1de7:H (GLN30) to (MET84) INTERACTION OF FACTOR XIII ACTIVATION PEPTIDE WITH ALPHA-THROMBIN: CRYSTAL STRUCTURE OF THE ENZYME-SUBSTRATE COMPLEX | ENZYME-SUBSTRATE COMPLEX, ALPHA-THROMBIN, FACTOR XIII ACTIVATION PEPTIDE, HYDROLASE/PEPTIDE, BLOOD CLOTTING, HYDROLASE-HYDROLASE SUBSTRATE COMPLEX
3t0a:C (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (S796T) | DYNAMPIC LOOP CONFORMATION, SER-796, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
3t0b:B (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (S796T) IPTG COMPLEX | DYNAMPIC LOOP CONFORMATION, SER-796, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
3t0d:B (LEU651) to (ALA716) E.COLI (LACZ) BETA-GALACTOSIDASE (S796T) IN COMPLEX WITH GALACTONOLACTONE | DYNAMPIC LOOP CONFORMATION, SER-796, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
2qlv:E (SER175) to (ARG246) CRYSTAL STRUCTURE OF THE HETEROTRIMER CORE OF THE S. CEREVISIAE AMPK HOMOLOG SNF1 | HETEROTRIMER, ATP-BINDING, CARBOHYDRATE METABOLISM, KINASE, MEMBRANE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, LIPOPROTEIN, MYRISTATE, CBS DOMAIN, TRANSCRIPTION, TRANSCRIPTION REGULATION, TRANSFERASE/PROTEIN BINDING COMPLEX
1dlp:A (THR56) to (PRO105) STRUCTURAL CHARACTERIZATION OF THE NATIVE FETUIN-BINDING PROTEIN SCILLA CAMPANULATA AGGLUTININ (SCAFET): A NOVEL TWO-DOMAIN LECTIN | TWO-DOMAIN LECTIN, BETA PRISM II FOLD, NATIVE, SUGAR BINDING PROTEIN
2qn5:T (GLN33) to (SER84) CRYSTAL STRUCTURE AND FUNCTIONAL STUDY OF THE BOWMAN-BIRK INHIBITOR FROM RICE BRAN IN COMPLEX WITH BOVINE TRYPSIN | RBTI, BOWMAN-BIRK INHIBITOR, MONOCOTYLEDONOUS PLANT, REACTIVE-SITE LOOP, PROTEASE-INHIBITOR, PLANT-PEST SYSTEMS, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, CALCIUM, DIGESTION, HYDROLASE, METAL-BINDING, SECRETED, ZYMOGEN, HYDROLASE INHIBITOR/HYDROLASE COMPLEX, HETERO-DIMER
3gch:B (GLN30) to (LYS84) CHEMISTRY OF CAGED ENZYMES. BINDING OF PHOTOREVERSIBLE CINNAMATES TO CHYMOTRYPSIN | HYDROLASE (SERINE PROTEINASE)
3gct:F (GLN30) to (LYS84) STRUCTURE OF GAMMA-*CHYMOTRYPSIN IN THE RANGE $P*H 2.0 TO $P*H 10.5 SUGGESTS THAT GAMMA-CHYMOTRYPSIN IS A COVALENT ACYL-ENZYME ADDUCT AT LOW $P*H | HYDROLASE, SERINE PROTEINASE, HYDROLASE-PEPTIDE COMPLEX
3t3g:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH GLCBRU | A+B PROTEIN, TRANSFERASE, MUSCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3t3h:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH GLCIU | A+B PROTEIN, TRANSFERASE, MUSCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3t3i:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH GLCCF3U | A+B PROTEIN, TRANSFERASE, MUSCLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2cv3:A (GLN30) to (GLY88) CRYSTAL STRUCTURE OF PORCINE PANCREATIC ELASTASE COMPLEXED WITH A MACROCLYCLIC PEPTIDE INHIBITOR | PROTEIN-INHIBITOR INTERACTION, MACROCYCLIC PEPTIDE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
2qrp:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH (1R)-3'-(2- NAPHTHYL)-SPIRO[1,5-ANHYDRO-D-GLUCITOL-1,5'-ISOXAZOLINE] | GLYCOGENOLYSIS, TYPE 2 DIABETES, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PYRIDOXAL PHOSPHATE, TRANSFERASE
2qrq:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH (1R)-3'-(4- METHYLPHENYL)-SPIRO[1,5-ANHYDRO-D-GLUCITOL-1,5'- ISOXAZOLINE] | GLYCOGENOLYSIS, TYPE 2 DIABETES, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PYRIDOXAL PHOSPHATE, TRANSFERASE
3t62:C (GLN30) to (LYS84) CRYSTAL STRUCTURE OF RECOMBINANT KUNITZ TYPE SERINE PROTEASE INHIBITOR-1 FROM THE CARIBBEAN SEA ANEMONE STICHODACTYLA HELIANTHUS IN COMPLEX WITH BOVINE CHYMOTRYPSIN | CHYMOTRYPSIN-INHIBITOR COMPLEX, KUNITZ-TYPE SERINE PROTEASE INHIBITOR, SECRETED, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3gir:A (ALA304) to (SER358) CRYSTAL STRUCTURE OF GLYCINE CLEAVAGE SYSTEM AMINOMETHYLTRANSFERASE T FROM BARTONELLA HENSELAE | BARTONELLA HENSELAE, GLYCINE CLEAVAGE SYSTEM, AMINOMETHYLTRANSFERASE, AMINOTRANSFERASE, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE, SSGCID
3gis:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF NA-FREE THROMBIN IN COMPLEX WITH THROMBOMODULIN | PROTEIN-PROTEIN COMPLEX, COAGULATION, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, EGF-LIKE DOMAIN, HYDROXYLATION, MEMBRANE, RECEPTOR, THROMBOPHILIA, TRANSMEMBRANE, BLOOD CLOTTING
3gis:F (GLN30) to (MET84) CRYSTAL STRUCTURE OF NA-FREE THROMBIN IN COMPLEX WITH THROMBOMODULIN | PROTEIN-PROTEIN COMPLEX, COAGULATION, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, EGF-LIKE DOMAIN, HYDROXYLATION, MEMBRANE, RECEPTOR, THROMBOPHILIA, TRANSMEMBRANE, BLOOD CLOTTING
1ppf:E (MET30) to (ALA84) X-RAY CRYSTAL STRUCTURE OF THE COMPLEX OF HUMAN LEUKOCYTE ELASTASE (PMN ELASTASE) AND THE THIRD DOMAIN OF THE TURKEY OVOMUCOID INHIBITOR | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ppg:E (MET30) to (ALA84) THE REFINED 2.3 ANGSTROMS CRYSTAL STRUCTURE OF HUMAN LEUKOCYTE ELASTASE IN A COMPLEX WITH A VALINE CHLOROMETHYL KETONE INHIBITOR | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ppz:A (ILE30) to (SER83) TRYPSIN COMPLEXES AT ATOMIC AND ULTRA-HIGH RESOLUTION | TRYPSIN, SERINE PROTEASE, ATOMIC AND ULTRA-HIGH RESOLUTION, COMPLEX, DFP, HYDROLASE
1dwb:H (GLN30) to (MET84) CRYSTALLOGRAPHIC ANALYSIS AT 3.0-ANGSTROMS RESOLUTION OF THE BINDING TO HUMAN THROMBIN OF FOUR ACTIVE SITE-DIRECTED INHIBITORS | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1dwc:H (GLN30) to (MET84) CRYSTALLOGRAPHIC ANALYSIS AT 3.0-ANGSTROMS RESOLUTION OF THE BINDING TO HUMAN THROMBIN OF FOUR ACTIVE SITE-DIRECTED INHIBITORS | SERINE PROTEINASE, HYDROLASE-HYROLASE INHIBITOR COMPLEX
1dwd:H (GLN30) to (MET84) CRYSTALLOGRAPHIC ANALYSIS AT 3.0-ANGSTROMS RESOLUTION OF THE BINDING TO HUMAN THROMBIN OF FOUR ACTIVE SITE-DIRECTED INHIBITORS | SERINE PROTEINASE, HYDROLASE-HYROLASE INHIBITOR COMPLEX
1pq5:A (ILE30) to (SER83) TRYPSIN AT PH 5, 0.85 A | TRYPSIN, ULTRA-HIGH RESOLUTION, SERINE PROTEASE, CATALYSIS, HYDROLASE
1pq7:A (ILE30) to (SER83) TRYPSIN AT 0.8 A, PH5 / BORAX | TRYPSIN, ULTRA-HIGH RESOLUTION, CATALYSIS, HYDROLASE
1pqa:A (ILE30) to (SER83) TRYPSIN WITH PMSF AT ATOMIC RESOLUTION | TRYPSIN, ATOMIC RESOLUTION, PMSF, CATALYSIS, HYDROLASE
1e0f:E (GLN30) to (MET84) CRYSTAL STRUCTURE OF THE HUMAN ALPHA-THROMBIN-HAEMADIN COMPLEX: AN EXOSITE II-BINDING INHIBITOR | COAGULATION/CRYSTAL STRUCTURE/HEPARIN-B, COAGULATION/CRYSTAL STRUCTURE/HEPARIN-BINDING SITE/ HIRUDIN/THROMBIN INHIBITOR, HYDROLASE
2qxg:A (GLN30) to (SER86) CRYSTAL STRUCTURE OF HUMAN KALLIKREIN 7 IN COMPLEX WITH ALA- ALA-PHE-CHLOROMETHYLKETONE | DIMER, 37 LOOP, ACTIVE SITE INHIBITOR, CHLOROMETHYL KETONE, ALTERNATIVE SPLICING, GLYCOPROTEIN, HYDROLASE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN
2qxg:B (GLN30) to (SER86) CRYSTAL STRUCTURE OF HUMAN KALLIKREIN 7 IN COMPLEX WITH ALA- ALA-PHE-CHLOROMETHYLKETONE | DIMER, 37 LOOP, ACTIVE SITE INHIBITOR, CHLOROMETHYL KETONE, ALTERNATIVE SPLICING, GLYCOPROTEIN, HYDROLASE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN
2r0k:A (ALA31) to (GLY84) PROTEASE DOMAIN OF HGFA WITH INHIBITOR FAB58 | SERINE PROTEASE, ANTIBODY, INHIBITOR, EGF-LIKE DOMAIN, GLYCOPROTEIN, HYDROLASE, KRINGLE, SECRETED, ZYMOGEN, IMMUNE SYSTEM
2r0l:A (ALA31) to (GLY84) SHORT FORM HGFA WITH INHIBITORY FAB75 | SERINE PROTEASE, ANTIBODY, ALLOSTERIC INHIBITOR, EGF-LIKE DOMAIN, GLYCOPROTEIN, HYDROLASE, KRINGLE, SECRETED, ZYMOGEN, IMMUNE SYSTEM
1px3:A (ASN649) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (G794A) | LOOP CONFORMATION, HYDROLASE
1px3:D (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (G794A) | LOOP CONFORMATION, HYDROLASE
2de9:A (GLN15) to (GLY73) CRYSTAL STRUCTURE OF PORCINE PANCREATIC ELASTASE COMPLEXED WITH TRIS AFTER SOAKING A TRIS-FREE SOLUTION | SERINE PROTEASE, HYDROLASE
4y76:A (GLN30) to (GLU84) FACTOR XA COMPLEX WITH GTC000401 | HYDROLASE, INHIBITOR
3th2:H (GLN30) to (ARG84) MG2+ IS REQUIRED FOR OPTIMAL FOLDING OF THE GAMMA-CARBOXYGLUTAMIC ACID (GLA) DOMAINS OF VITAMIN K-DEPENDENT CLOTTING FACTORS AT PHYSIOLOGICAL CA2+ | HYDROLASE, BLOOD CLOTTING, SERINE PROTEASE, BLOOD COAGULATION, SOLUBLE TISSUE FACTOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3th4:H (GLN30) to (ARG84) MG2+ IS REQUIRED FOR OPTIMAL FOLDING OF THE GAMMA-CARBOXYGLUTAMIC ACID (GLA) DOMAINS OF VITAMIN K-DEPENDENT CLOTTING FACTORS AT PHYSIOLOGICAL CA2+ | HYDROLASE, SERINE PROTEASE, BLOOD CLOTTING, SOLUBLE TISSUE FACTOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4y9w:A (SER2) to (LYS49) ASPARTIC PROTEINASE SAPP2 SECRETED FROM CANDIDA PARAPSILOSIS AT 0.82 A RESOLUTION. | CANDIDAPEPSIN, ASPARTIC ACID ENDOPEPTIDASE, HYDROLASE
4jf7:D (VAL400) to (GLY486) STRUCTURE OF THE PARAINFLUENZA VIRUS 5 (PIV5) HEMAGGLUTININ- NEURAMINIDASE (HN) ECTODOMAIN | PARAMYXOVIRUS, PIV5, ATTACHMENT PROTEIN, HN, RECEPTOR BINDING PROTEIN, ECTODOMAIN, VIRAL PROTEIN
4jf7:A (SER399) to (GLY486) STRUCTURE OF THE PARAINFLUENZA VIRUS 5 (PIV5) HEMAGGLUTININ- NEURAMINIDASE (HN) ECTODOMAIN | PARAMYXOVIRUS, PIV5, ATTACHMENT PROTEIN, HN, RECEPTOR BINDING PROTEIN, ECTODOMAIN, VIRAL PROTEIN
2rab:A (ALA232) to (THR266) STRUCTURE OF GLUTATHIONE AMIDE REDUCTASE FROM CHROMATIUM GRACILE IN COMPLEX WITH NAD | GLUTATHIONE, SUBSTRATE ANALOG, NAD, FAD, REDOX, OXIDOREDUCTASE
1qbv:H (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN COMPLEXED WITH AN GUANIDINE-MIMETIC INHIBITOR | THROMBIN, INHIBITOR, 3DP, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4jjo:A (ARG136) to (PRO182) CRYSTAL STRUCTURE OF APO-CLAVIBACTER MICHIGANENSIS EXPANSIN | CELLULOSE BINDING PROTEIN, CELL WALL LOOSENING, SUGAR BINDING PROTEIN
3h0c:B (THR221) to (PRO290) CRYSTAL STRUCTURE OF HUMAN DIPEPTIDYL PEPTIDASE IV (CD26) IN COMPLEX WITH A REVERSED AMIDE INHIBITOR | COMPLEX (HYDROLASE-INHIBITOR), DPP-IV, DIABETES MELLITUS, DRUG DESIGN, HYDROLASE, SERINE PROTEASE, AMINOPEPTIDASE, GLYCOPROTEIN, PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, CELL MEMBRANE, DISULFIDE BOND, MEMBRANE, SECRETED
1ela:A (GLN30) to (GLY88) ANALOGOUS INHIBITORS OF ELASTASE DO NOT ALWAYS BIND ANALOGOUSLY | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEINASE
1elf:A (GLN30) to (GLY88) NATURE OF THE INACTIVATION OF ELASTASE BY N-PEPTIDYL-O- AROYL HYDROXYLAMINE AS A FUNCTION OF PH | COMPLEX (HYDROLASE/INHIBITOR)
1eoj:A (GLN30) to (MET84) DESIGN OF P1' AND P3' RESIDUES OF TRIVALENT THROMBIN INHIBITORS AND THEIR CRYSTAL STRUCTURES | THROMBIN INHIBITORS, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1esa:A (GLN30) to (GLY88) DIRECT STRUCTURE OBSERVATION OF AN ACYL-ENZYME INTERMEDIATE IN THE HYDROLYSIS OF AN ESTER SUBSTRATE BY ELASTASE | HYDROLASE(SERINE PROTEINASE)
1eth:A (HIS355) to (GLY415) TRIACYLGLYCEROL LIPASE/COLIPASE COMPLEX | COMPLEX (HYDROLASE-COFACTOR), LIPID DEGRADATION, COMPLEX (HYDROLASE- COFACTOR) COMPLEX
1eth:C (HIS355) to (GLY415) TRIACYLGLYCEROL LIPASE/COLIPASE COMPLEX | COMPLEX (HYDROLASE-COFACTOR), LIPID DEGRADATION, COMPLEX (HYDROLASE- COFACTOR) COMPLEX
1ets:H (GLN30) to (MET84) REFINED 2.3 ANGSTROMS X-RAY CRYSTAL STRUCTURE OF BOVINE THROMBIN COMPLEXES FORMED WITH THE BENZAMIDINE AND ARGININE-BASED THROMBIN INHIBITORS NAPAP, 4-TAPAP AND MQPA: A STARTING POINT FOR IMPROVING ANTITHROMBOTICS | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ett:H (GLN30) to (MET84) REFINED 2.3 ANGSTROMS X-RAY CRYSTAL STRUCTURE OF BOVINE THROMBIN COMPLEXES FORMED WITH THE BENZAMIDINE AND ARGININE-BASED THROMBIN INHIBITORS NAPAP, 4-TAPAP AND MQPA: A STARTING POINT FOR IMPROVING ANTITHROMBOTICS | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ex3:A (GLN30) to (LYS84) CRYSTAL STRUCTURE OF BOVINE CHYMOTRYPSINOGEN A (TETRAGONAL) | HYDROLASE
2snv:A (GLY187) to (GLY232) THE REFINED STRUCTURE OF SINDBIS VIRUS CORE PROTEIN IN COMPARISON WITH OTHER CHYMOTRYPSIN-LIKE SERINE PROTEINASE STRUCTURES | VIRAL PROTEIN
3h43:I (PRO91) to (LEU151) N-TERMINAL DOMAIN OF THE PROTEASOME-ACTIVATING NUCLEOTIDASE OF METHANOCALDOCOCCUS JANNASCHII | PROTEASOME, REGULATORY PARTICLE, NUCLEOSIDASE, ATP-BINDING, CYTOPLASM, NUCLEOTIDE-BINDING, HYDROLASE
1ezu:C (GLN430) to (ASN484) ECOTIN Y69F, D70P BOUND TO D102N TRYPSIN | MACROMOLECULAR COMPLEX, PROTEASE INHIBITOR, PROTEIN-PROTEIN INTERACTIONS, HYDROLASE/INHIBITOR COMPLEX
2e5y:B (GLU21) to (ALA62) EPSILON SUBUNIT AND ATP COMPLEX OF F1F0-ATP SYNTHASE FROM THE THERMOPHILIC BACILLUS PS3 | ATP SYNTHASE, F1FO ATP SYNTHASE, F1-ATPASE, EPSILON SUBUNIT, ATP, HYDROLASE
1qrz:A (GLN576) to (GLU634) CATALYTIC DOMAIN OF PLASMINOGEN | MICROPLASMINOGEN, SERINE PROTEASE, ZYMOGEN, CHYMOTRYPSIN FAMILY, HYDROLASE
1qrz:B (GLN576) to (GLU634) CATALYTIC DOMAIN OF PLASMINOGEN | MICROPLASMINOGEN, SERINE PROTEASE, ZYMOGEN, CHYMOTRYPSIN FAMILY, HYDROLASE
1qrz:D (GLN576) to (GLU634) CATALYTIC DOMAIN OF PLASMINOGEN | MICROPLASMINOGEN, SERINE PROTEASE, ZYMOGEN, CHYMOTRYPSIN FAMILY, HYDROLASE
3h7l:A (THR31) to (SER86) CRYSTAL STRUCTURE OF ENDOGLUCANASE-RELATED PROTEIN FROM VIBRIO PARAHAEMOLYTICUS | ENDOGLUCANASE, DEHYDROGENASE, PSI-2, NYSGXRC, STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE, NEW YORK SGX RESEARCH CENTER FOR STRUCTURAL GENOMICS, HYDROLASE
3h7o:A (VAL16) to (TYR73) CRYSTAL STRUCTURE OF SCABIES MITE INACTIVATED PROTEASE PARALOGUE S-I1 (SMIPP-S-I1) | HYDROLASE
3h7t:A (VAL16) to (MET68) CRYSTAL STRUCTURE OF SCABIES MITE INACTIVATED PROTEASE PARALOGUE S-D1 (SMIPP-S-D1) | HYDROLASE
3u34:B (ARG39) to (GLY105) CRYSTAL STRUCTURE OF THE GENERAL STRESS FMN/FAD BINDING PROTEIN FROM THE PHYTOPATHOGEN XANTHOMONAS CITRI | XANTHOMONAS CITRI GENERAL STRESS PROTEIN FMN BINDING PROTEIN FAD BINDING PROTEIN, PNP-OXIDASE LIKE FOLD, FMN FAD, PROTEIN BINDING
3u34:C (ARG39) to (GLY105) CRYSTAL STRUCTURE OF THE GENERAL STRESS FMN/FAD BINDING PROTEIN FROM THE PHYTOPATHOGEN XANTHOMONAS CITRI | XANTHOMONAS CITRI GENERAL STRESS PROTEIN FMN BINDING PROTEIN FAD BINDING PROTEIN, PNP-OXIDASE LIKE FOLD, FMN FAD, PROTEIN BINDING
3u35:A (ARG39) to (GLY105) CRYSTAL STRUCTURE OF THE GENERAL STRESS FMN/FAD BINDING PROTEIN FROM THE PHYTOPATHOGEN XANTHOMONAS CITRI | XANTHOMONAS CITRI GENERAL STRESS PROTEIN FMN BINDING PROTEIN FAD BINDING PROTEIN, PNP-OXIDASE LIKE FOLD, FMN/FAD, PROTEIN BINDING
3hat:H (GLN30) to (MET84) ACTIVE SITE MIMETIC INHIBITION OF THROMBIN | COMPLEX (SERINE PROTEASE-INHIBITOR), COMPLEX (SERINE PROTEASE- INHIBITOR) COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1qz8:A (CYS14) to (GLU68) CRYSTAL STRUCTURE OF SARS CORONAVIRUS NSP9 | SARS, REPLICATION, NSP9, CORONAVIRUS, UNKNOWN FUNCTION
1qz8:B (CYS14) to (GLU68) CRYSTAL STRUCTURE OF SARS CORONAVIRUS NSP9 | SARS, REPLICATION, NSP9, CORONAVIRUS, UNKNOWN FUNCTION
4jz1:A (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MATRIPTASE IN COMPLEX WITH INHIBITOR | MATRIPTASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2est:E (GLN30) to (GLY84) CRYSTALLOGRAPHIC STUDY OF THE BINDING OF A TRIFLUOROACETYL DIPEPTIDE ANILIDE INHIBITOR WITH ELASTASE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEINASE
4k3j:A (MET508) to (ASN566) CRYSTAL STRUCTURE OF ONARTUZUMAB FAB IN COMPLEX WITH MET AND HGF-BETA | ANTIBODY, GLYCOSYLATION, TRANSFERASE-IMMUNE SYSTEM-GROWTH FACTOR COMPLEX
1fn8:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA BARREL, HYDROLASE, HYDROLASE-HYDROLASE SUBSTRATE COMPLEX
3hk6:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF MURINE THROMBIN MUTANT W215A/E217A (TWO MOLECULES IN THE ASYMMETRIC UNIT) | SERINE PROTEASE, ACUTE PHASE, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISULFIDE BOND, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, ZYMOGEN
3hk6:D (GLN30) to (MET84) CRYSTAL STRUCTURE OF MURINE THROMBIN MUTANT W215A/E217A (TWO MOLECULES IN THE ASYMMETRIC UNIT) | SERINE PROTEASE, ACUTE PHASE, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISULFIDE BOND, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, ZYMOGEN
3ufi:A (ASP65) to (GLY167) CRYSTAL STRUCTURE OF A PUTATIVE CELL ADHESION PROTEIN (BACOVA_04980) FROM BACTEROIDES OVATUS ATCC 8483 AT 2.18 A RESOLUTION | FIMBRIAL PROTEIN, CELL ADHESION, MAJOR FIMBRIAL SUBUNIT PROTEIN (FIMA),, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY
3hkj:E (GLN30) to (MET84) CRYSTAL STRUCTURE OF HUMAN THROMBIN MUTANT W215A/E217A IN COMPLEX WITH THE EXTRACELLULAR FRAGMENT OF HUMAN PAR1 | SERINE PROTEASE, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, SECRETED, ZYMOGEN, CELL MEMBRANE, G-PROTEIN COUPLED RECEPTOR, MEMBRANE, PHOSPHOPROTEIN, RECEPTOR, TRANSDUCER, TRANSMEMBRANE
4yt7:H (GLN30) to (ARG84) FACTOR VIIA IN COMPLEX WITH THE INHIBITOR 2-(2-{(R)-[(4- CARBAMIMIDOYLPHENYL)AMINO][5-ETHOXY-2-FLUORO-3-(PROPAN-2-YLOXY) PHENYL]METHYL}-1H-IMIDAZOL-4-YL)BENZAMIDE | GLYCOPROTEIN, HYDROLASE, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM-BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4yta:A (GLN30) to (SER84) BOND LENGTH ANALYSIS OF ASP, GLU AND HIS RESIDUES IN TRYPSIN AT 1.2A RESOLUTION | SERINE PROTEASE, HYDROLASE
4k5z:A (TYR29) to (GLU84) CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH FRAGMENT INHIBITOR 6-CHLORO-2,3-DIHYDRO-1H-ISOINDOL-1-ONE | SERINE PROTEASE, GLYCOSYLATED, MAST CELLS, SECRETED, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4k60:A (TYR29) to (GLU84) CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH FRAGMENT 6-BROMO-1, 3-DIHYDRO-2H-INDOL-2-ONE | SERINE PROTEASE, GLYCOSYLATED, MAST CELLS, SECRETED, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1rd3:D (GLN30) to (MET84) 2.5A STRUCTURE OF ANTICOAGULANT THROMBIN VARIANT E217K | HYDROLASE
4k69:A (TYR29) to (GLU84) CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH FRAGMENT LINKED BENZIMIDAZOLONE INHIBITOR: (3S)-3-{3-[(6-BROMO-2-OXO-2,3-DIHYDRO-1H- INDOL-4-YL)METHYL]-2-OXO-2,3-DIHYDRO-1H-BENZIMIDAZOL-1-YL}HEXANOIC ACID | SERINE PROTEASE, GLYCOSYLATED, MAST CELLS, SECRETED, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1fq3:A (TYR29) to (PRO84) CRYSTAL STRUCTURE OF HUMAN GRANZYME B | CHYMOTRYPSIN-LIKE SERINE PROTEINASE, HYDROLASE
1fq3:B (TYR29) to (PRO84) CRYSTAL STRUCTURE OF HUMAN GRANZYME B | CHYMOTRYPSIN-LIKE SERINE PROTEINASE, HYDROLASE
1rfn:A (GLN30) to (ASN84) HUMAN COAGULATION FACTOR IXA IN COMPLEX WITH P-AMINO BENZAMIDINE | SERINE PROTEINASE, BLOOD COAGULATION, COAGULATION FACTOR
1riw:B (GLN51) to (MET116) THROMBIN IN COMPLEX WITH NATURAL PRODUCT INHIBITOR OSCILLARIN | PROTEASE, THROMBIN, INHIBITOR COMPLEX, OSCILLARIN, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1fuj:A (MET30) to (SER84) PR3 (MYELOBLASTIN) | HYDROLASE, SERINE PROTEASE, GLYCOPROTEIN, ZYMOGEN, HYDROLASE (SERINE PROTEASE)
1rp1:A (GLN354) to (ALA417) DOG PANCREATIC LIPASE RELATED PROTEIN 1 | HYDROLASE, LIPID DEGRADATION, PANCREATIC LIPASE
1fy3:A (LEU15) to (SER72) [G175Q]HBP, A MUTANT OF HUMAN HEPARIN BINDING PROTEIN (CAP37) | SERINE PROTEASE HOMOLOG, BPTI BINDING SITE, ANTIMICROBIAL PROTEIN
1fy4:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA BARREL, HYDROLASE
1fy5:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA BARREL, HYDROLASE
1rqc:A (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:B (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:C (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:D (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:F (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:H (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rqc:J (VAL143) to (GLY190) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | HYDROLASE
1rrh:A (SER57) to (VAL128) SOYBEAN LIPOXYGENASE (LOX-3) AT AMBIENT TEMPERATURES AT 2.0 A RESOLUTION | OXIDOREDUCTASE, IRON METALLOPROTEIN, LIPOXYGENASE
2f91:A (GLN30) to (THR84) 1.2A RESOLUTION STRUCTURE OF A CRAYFISH TRYPSIN COMPLEXED WITH A PEPTIDE INHIBITOR, SGTI | SERINE PROTEASE, TRYPSIN, CANONICAL INHIBITOR, ATOMIC RESOLUTION, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1g27:A (LEU78) to (GLY124) CRYSTAL STRUCTURE OF E.COLI POLYPEPTIDE DEFORMYLASE COMPLEXED WITH THE INHIBITOR BB-3497 | BB-3497, INHIBITION, POLYPEPTIDE DEFORMYLASE, HYDROLASE
1g37:A (GLN30) to (MET84) CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN COMPLEXED WITH BCH-10556 AND EXOSITE-DIRECTED PEPTIDE | PROTEASE, THROMBIN, INHIBITOR, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3unr:A (GLN30) to (SER84) BOND LENGTH ANALYSIS OF ASP, GLU AND HIS RESIDUES IN TRYPSIN AT 1.2A RESOLUTION | SERINE PROTEASE, HYDROLASE
4kga:A (GLN30) to (HIS91) CRYSTAL STRUCTURE OF KALLIKREIN-RELATED PEPTIDASE 4 | KLK4, KALLIKREIN-4, SERINE PROTEASE, PROTEASE, HYDROLASE
4kga:B (GLN30) to (SER86) CRYSTAL STRUCTURE OF KALLIKREIN-RELATED PEPTIDASE 4 | KLK4, KALLIKREIN-4, SERINE PROTEASE, PROTEASE, HYDROLASE
2fes:H (GLN30) to (MET84) ORALLY ACTIVE THROMBIN INHIBITORS | THROMBIN INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2vgc:B (GLN30) to (LYS84) GAMMA-CHYMOTRYPSIN D-PARA-CHLORO-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX | HYDROLASE, SERINE PROTEASE
1gct:B (GLN30) to (LYS84) IS GAMMA-CHYMOTRYPSIN A TETRAPEPTIDE ACYL-ENZYME ADDUCT OF GAMMA- CHYMOTRYPSIN? | HYDROLASE, SERINE PROTEINASE, HYDROLASE-PEPTIDE COMPLEX
1gdn:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA BARREL, HYDROLASE, HYDROLASE-HYDROLASE SUBSTRATE COMPLEX
1gdq:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA-BARREL, HYDROLASE
1gdu:A (ILE30) to (SER84) FUSARIUM OXYSPORUM TRYPSIN AT ATOMIC RESOLUTION | BETA-BARREL, HYDROLASE
2vkx:C (LYS534) to (LYS594) HUMAN NCAM, FN3 DOMAINS 1 AND 2, M610R MUTANT | ADHESION RECEPTOR, CELL ADHESION
2fmj:A (PHE29) to (ARG84) 220-LOOP MUTANT OF STREPTOMYCES GRISEUS TRYPSIN | TRYPSIN, SERINE PROTEASE, HYDROLASE
3uwi:A (GLN30) to (SER84) BOVINE TRYPSIN VARIANT X(TRIPLEGLU217PHE227) IN COMPLEX WITH SMALL MOLECULE INHIBITOR | TRYPSIN-LIKE SERINE PROTEASE, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2fo9:A (GLN30) to (GLY88) STRUCTURE OF PORCINE PANCREATIC ELASTASE IN 95% ACETONE | ELASTASE; SOLVENT MAPPING; ORGANIC SOLVENTS; PROTEIN BINDING SITES; MULTIPLE SOLVENT CRYSTAL STRUCTURES, HYDROLASE
2foa:A (GLN30) to (GLY88) STRUCTURE OF PORCINE PANCREATIC ELASTASE IN 40/50/10 % BENZENE | ELASTASE; SOLVENT MAPPING; ORGANIC SOLVENTS; PROTEIN BINDING SITES; MULTIPLE SOLVENT CRYSTAL STRUCTURES, HYDROLASE
2fob:A (GLN30) to (GLY88) STRUCTURE OF PORCINE PANCREATIC ELASTASE IN 40/50/10 CYCLOHEXANE | ELASTASE; SOLVENT MAPPING; ORGANIC SOLVENTS; PROTEIN BINDING SITES; MULTIPLE SOLVENT CRYSTAL STRUCTURES, HYDROLASE
1ggd:B (GLN30) to (LYS84) CRYSTAL STUCTURE OF GAMMA CHYMOTRYPSIN WITH N-ACETYL-LEUCIL- PHENYLALANINE ALDEHYDE BOUND AT THE ACTIVE SITE | CHYMOTRYPSIN, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1gha:F (GLN30) to (LYS84) A SECOND ACTIVE SITE IN CHYMOTRYPSIN? THE X-RAY CRYSTAL STRUCTURE OF N-ACETYL-D-TRYPTOPHAN BOUND TO GAMMA-CHYMOTRYPSIN | HYDROLASE, SERINE PROTEINASE
1ghb:F (GLN30) to (LYS84) A SECOND ACTIVE SITE IN CHYMOTRYPSIN? THE X-RAY CRYSTAL STRUCTURE OF N-ACETYL-D-TRYPTOPHAN BOUND TO GAMMA-CHYMOTRYPSIN | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ghx:H (GLN30) to (MET84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI-CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1gi2:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI- CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gi4:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI- CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gi5:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI- CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gi6:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI- CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gj4:H (GLN30) to (MET84) SELECTIVITY AT S1, H2O DISPLACEMENT, UPA, TPA, SER190/ALA190 PROTEASE, STRUCTURE-BASED DRUG DESIGN | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, BLOOD CLOTTING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1gj5:H (GLN30) to (MET84) SELECTIVITY AT S1, H2O DISPLACEMENT, UPA, TPA, SER190/ALA190 PROTEASE, STRUCTURE-BASED DRUG DESIGN | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, BLOOD CLOTTING, HYDROLASE,HYDROLASE-HYDROLASE INHIBITOR COMPLEX, BLOOD CLOTTING,HYDROLASE-INHIBITOR COMPLEX
1gj6:A (GLN30) to (SER84) ENGINEERING INHIBITORS HIGHLY SELECTIVE FOR THE S1 SITES OF SER190 TRYPSIN-LIKE SERINE PROTEASE DRUG TARGETS | SELECTIVITY AT S1, H2O DISPLACEMENT, UPA, TPA, SER190/ALA190 PROTEASE, STRUCTURE-BASED DRUG DESIGN, HYDROLASE
1gl1:A (GLN30) to (LYS84) STRUCTURE OF THE COMPLEX BETWEEN BOVINE ALPHA-CHYMOTRYPSIN AND PMP-C, AN INHIBITOR FROM THE INSECT LOCUSTA MIGRATORIA | HYDROLASE/INHIBITOR, COMPLEX (PROTEASE/INHIBITOR), HYDROLASE, SERINE PROTEASE, SERINE PROTEASE INHIBITOR
1gl1:B (GLN30) to (LYS84) STRUCTURE OF THE COMPLEX BETWEEN BOVINE ALPHA-CHYMOTRYPSIN AND PMP-C, AN INHIBITOR FROM THE INSECT LOCUSTA MIGRATORIA | HYDROLASE/INHIBITOR, COMPLEX (PROTEASE/INHIBITOR), HYDROLASE, SERINE PROTEASE, SERINE PROTEASE INHIBITOR
1gmd:F (GLN30) to (LYS84) X-RAY CRYSTAL STRUCTURE OF GAMMA-CHYMOTRYPSIN IN HEXANE | HYDROLASE, SERINE PROTEASE
1gmh:F (GLN30) to (LYS84) REFINED CRYSTAL STRUCTURE OF "AGED" AND "NON-AGED" ORGANOPHOSPHORYL CONJUGATES OF GAMMA-CHYMOTRYPSIN | HYDROLASE(SERINE PROTEINASE)
1sgf:A (TRP29) to (LEU84) CRYSTAL STRUCTURE OF 7S NGF: A COMPLEX OF NERVE GROWTH FACTOR WITH FOUR BINDING PROTEINS (SERINE PROTEINASES) | GROWTH FACTOR (BETA-NGF), HYDROLASE - SERINE PROTEINASE (GAMMA-NGF), INACTIVE SERINE PROTEINASE (ALPHA-NGF), GROWTH FACTOR
1sgf:G (HIS30) to (PHE84) CRYSTAL STRUCTURE OF 7S NGF: A COMPLEX OF NERVE GROWTH FACTOR WITH FOUR BINDING PROTEINS (SERINE PROTEINASES) | GROWTH FACTOR (BETA-NGF), HYDROLASE - SERINE PROTEINASE (GAMMA-NGF), INACTIVE SERINE PROTEINASE (ALPHA-NGF), GROWTH FACTOR
1sgf:X (VAL31) to (LEU84) CRYSTAL STRUCTURE OF 7S NGF: A COMPLEX OF NERVE GROWTH FACTOR WITH FOUR BINDING PROTEINS (SERINE PROTEINASES) | GROWTH FACTOR (BETA-NGF), HYDROLASE - SERINE PROTEINASE (GAMMA-NGF), INACTIVE SERINE PROTEINASE (ALPHA-NGF), GROWTH FACTOR
1shh:B (GLN30) to (MET84) SLOW FORM OF THROMBIN BOUND WITH PPACK | SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2g00:A (GLN30) to (GLU84) FACTOR XA IN COMPLEX WITH THE INHIBITOR 3-(6-(2'- ((DIMETHYLAMINO)METHYL)-4-BIPHENYLYL)-7-OXO-3- (TRIFLUOROMETHYL)-4,5,6,7-TETRAHYDRO-1H-PYRAZOLO[3,4- C]PYRIDIN-1-YL)BENZAMIDE | GLYCOPROTEIN, HYDROLASE, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM- BINDING
1shy:A (TRP507) to (ASN566) THE CRYSTAL STRUCTURE OF HGF BETA-CHAIN IN COMPLEX WITH THE SEMA DOMAIN OF THE MET RECEPTOR. | PROTEASE, SEMA DOMAIN, PSI DOMAIN, RECEPTOR ECTODOMAIN GROWTH FACTOR, GROWTH FACTOR-GROWTH FACTOR RECEPTOR COMPLEX
1gpl:A (GLY353) to (ALA417) RP2 LIPASE | SERINE ESTERASE, HYDROLASE, LIPID DEGRADATION, PANCREAS, GLYCOPROTEIN, CHIMERIC
2g3x:B (VAL28) to (VAL93) CRYSTAL STRUCTURE OF TRANSTHYRETIN MUTANT I84S AT ACIDIC PH | TTR, AMYLOID FIBRILS, POINT MUTATION, TRANSPORT PROTEIN
3i3b:B (LEU651) to (ALA716) E.COLI (LACZ) BETA-GALACTOSIDASE (M542A) IN COMPLEX WITH D- GALACTOPYRANOSYL-1-ON | BETA-GALACTOSIDASE, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
1sl3:A (GLN30) to (MET84) CRYSTAL STRUCTUE OF THROMBIN IN COMPLEX WITH A POTENT P1 HETEROCYCLE- ARYL BASED INHIBITOR | THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING, HYDROLASE-INHIBITOR COMPLEX, BLOOD CLOTTING,HYDROLASE-INHIBITOR COMPLEX
3i3d:B (LEU651) to (ARG721) E. COLI (LACZ) BETA-GALACTOSIDASE (M542A) IN COMPLEX WITH IPTG | BETA-GALACTOSIDASE, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3i3d:D (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (M542A) IN COMPLEX WITH IPTG | BETA-GALACTOSIDASE, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3i3e:B (ASN649) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (M542A) | BETA-GALACTOSIDASE, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3i3e:C (ASN649) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (M542A) | BETA-GALACTOSIDASE, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
2g51:A (ILE30) to (SER83) ANOMALOUS SUBSTRUCTURE OF TRYPSIN (P1) | ANOMALOUS SUBSTRUCTURE OF TRYPSIN (P1), HYDROLASE
2g52:A (ILE30) to (SER83) ANOMALOUS SUBSTRUCTURE OF TRYPSIN (P21) | ANOMALOUS SUBSTRUCTURE OF TRYPSIN (P21), HYDROLASE
1spj:A (TRP29) to (VAL83) STRUCTURE OF MATURE HUMAN TISSUE KALLIKREIN (HUMAN KALLIKREIN 1 OR KLK1) AT 1.70 ANGSTROM RESOLUTION WITH VACANT ACTIVE SITE | SERINE PROTEASE, KLK1, HK1, HUMAN KALLIKREIN 1, HUMAN TISSUE KALLIKREIN 1, TISSUE KALLIKREIN, HYDROLASE
2vu8:E (VAL31) to (SER84) CRYSTAL STRUCTURE OF AN INSECT INHIBITOR WITH A FUNGAL TRYPSIN | HYDROLASE/INHIBITOR, CANONICAL INHIBITOR, INHIBITOR, SERINE PROTEASE, SPECIES SELECTIVITY, INSECT, ZYMOGEN, PROTEASE, SECRETED, HYDROLASE
3vd4:B (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (N460D) IN COMPLEX WITH IPTG | TRANSITION STATE STABILIZATION, SUBSTRATE BINDING, 2-STAGE BINDING, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
1gvl:A (GLN30) to (VAL86) HUMAN PROKALLIKREIN 6 (HK6)/ PROZYME/ PROPROTEASE M/ PRONEUROSIN | HYDROLASE, ZYMOGEN, HUMAN KALLIKREIN
2gch:F (GLN30) to (LYS84) REFINED CRYSTAL STRUCTURE OF GAMMA-CHYMOTRYPSIN AT 1.9 ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
2gd4:H (GLN30) to (GLU84) CRYSTAL STRUCTURE OF THE ANTITHROMBIN-S195A FACTOR XA-PENTASACCHARIDE COMPLEX | SERPIN, MICHAELIS COMPLEX, HYDROLASE
2gd4:B (GLN30) to (GLU84) CRYSTAL STRUCTURE OF THE ANTITHROMBIN-S195A FACTOR XA-PENTASACCHARIDE COMPLEX | SERPIN, MICHAELIS COMPLEX, HYDROLASE
3veq:B (GLN30) to (SER81) A BINARY COMPLEX BETWWEN BOVINE PANCREATIC TRYPSIN AND A ENGINEERED MUTANT TRYPSIN INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3vfe:A (GLN30) to (SER84) VIRTUAL SCREENING AND X-RAY CRYSTALLOGRAPHY FOR HUMAN KALLIKREIN 6 INHIBITORS WITH AN AMIDINOTHIOPHENE P1 GROUP | HUMAN KALLIKREIN 6, HK6, SERINE PROTEASE, PROTEIN-LIGAND COMPLEX, AMIDINOTHIOPHENE, HYDROLASE
3vgc:B (GLN30) to (LYS84) GAMMA-CHYMOTRYPSIN L-NAPHTHYL-1-ACETAMIDO BORONIC ACID ACID INHIBITOR COMPLEX | HYDROLASE, SERINE PROTEASE
4l0z:A (LEU102) to (THR161) CRYSTAL STRUCTURE OF RUNX1 AND ETS1 BOUND TO TCR ALPHA PROMOTER (CRYSTAL FORM 2) | RUNT DOMAIN, ETS DOMAIN, TRANSCRIPTION-DNA COMPLEX
3iaq:B (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (E416V) | GLU-416-VAL BETA-GALACTOSIDASE HYDROLASE TIM BARREL(ALPHA/BETA BARREL) JELLY-ROLL BARREL IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3iaq:C (ASN649) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (E416V) | GLU-416-VAL BETA-GALACTOSIDASE HYDROLASE TIM BARREL(ALPHA/BETA BARREL) JELLY-ROLL BARREL IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3idb:B (PHE169) to (ASN215) CRYSTAL STRUCTURE OF (108-268)RIIB:C HOLOENZYME OF CAMP- DEPENDENT PROTEIN KINASE | PKA, CAMP, SPR, AFFINITY, KINASE, LINKER, CRYSTAL STRUCTURE, RII HOLOENZYME, ALTERNATIVE SPLICING, ATP-BINDING, CYTOPLASM, LIPOPROTEIN, MYRISTATE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, SERINE/THREONINE-PROTEIN KINASE, TRANSFERASE, ACETYLATION, CAMP-BINDING
2gmt:B (GLN30) to (LYS84) THREE-DIMENSIONAL STRUCTURE OF CHYMOTRYPSIN INACTIVATED WITH (2S) N- ACETYL-L-ALANYL-L-PHENYLALANYL-CHLOROETHYL KETONE: IMPLICATIONS FOR THE MECHANISM OF INACTIVATION OF SERINE PROTEASES BY CHLOROKETONES | HYDROLASE(SERINE PROTEINASE)
2w1u:B (ASN880) to (SER945) A FAMILY 32 CARBOHYDRATE-BINDING MODULE, FROM THE MU TOXIN PRODUCED BY CLOSTRIDIUM PERFRINGENS, IN COMPLEX WITH BETA- D-GLCNAC-BETA(1,3)GALNAC | FAMILY 32 CARBOHYDRATE BINDING MODULE, FAMILY 84 GLYCOSIDE HYDROLASE, GLYCOSIDASE, HEXOSAMINIDASE, CLOSTRIDIUM PERFRINGENS, CBM, TOXIN, SECRETED, VIRULENCE, HYDROLASE
1t7c:C (GLN30) to (LYS84) CRYSTAL STRUCTURE OF THE P1 GLU BPTI MUTANT- BOVINE CHYMOTRYPSIN COMPLEX | CHYMOTRYPSIN; SERINE PROTEINASE; BOVINE PANCREATIC TRYPSIN INHIBITOR; BPTI; PROTEIN-PROTEIN INTERACTION; NON-COGNATE BINDING; S1 POCKET; PRIMARY SPECIFICITY; CRYSTAL STRUCTURE, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1h6y:B (GLN21) to (GLU81) THE ROLE OF CONSERVED AMINO ACIDS IN THE CLEFT OF THE C-TERMINAL FAMILY 22 CARBOHYDRATE BINDING MODULE OF CLOSTRIDIUM THERMOCELLUM XYN10B IN LIGAND BINDING | XYLAN DEGRADATION, HYDROLASE, GLYCOSIDASE
1t8o:C (GLN30) to (LYS84) CRYSTAL STRUCTURE OF THE P1 TRP BPTI MUTANT- BOVINE CHYMOTRYPSIN COMPLEX | CHYMOTRYPSIN, SERINE PROTEINASE, BOVINE PANCREATIC TRYPSIN INHIBITOR, BPTI, PROTEIN-PROTEIN INTERACTION, NON-COGNATE BINDING, S1 POCKET, PRIMARY SPECIFICITY, CRYSTAL STRUCTURE, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
2w47:A (ALA66) to (SER130) CLOSTRIDIUM THERMOCELLUM CBM35 IN COMPLEX WITH DELTA-4,5- ANHYDROGALACTURONIC ACID | HYDROLASE
1ta2:A (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH COMPOUND 1 | THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1ta6:A (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH COMPOUND 14B | THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1h9i:E (GLN30) to (ASN84) COMPLEX OF EETI-II MUTANT WITH PORCINE TRYPSIN | HYDROLASE/INHIBITOR, COMPLEX (SERINE PROTEASE/INHIBITOR), TRYPSIN, SQUASH INHIBITOR, CYSTINE KNOT
1hah:H (GLN30) to (MET84) THE ISOMORPHOUS STRUCTURES OF PRETHROMBIN2, HIRUGEN-AND PPACK- THROMBIN: CHANGES ACCOMPANYING ACTIVATION AND EXOSITE BINDING TO THROMBIN | COMPLEX(SERINE PROTEINASE-INHIBITOR), COMPLEX(SERINE PROTEINASE- INHIBITOR) COMPLEX
2w5e:B (CYS438) to (GLU479) STRUCTURAL AND BIOCHEMICAL ANALYSIS OF HUMAN PATHOGENIC ASTROVIRUS SERINE PROTEASE AT 2.0 ANGSTROM RESOLUTION | COILED COIL, TRANSMEMBRANE, THIOL PROTEASE, RNA REPLICATION, RIBOSOMAL FRAMESHIFTING, SERINE PROTEASE, CATALYTIC TRIAD, PROTEASE, MEMBRANE, HYDROLASE, ANTIVIRAL, ASTROVIRUS
2w5e:C (CYS438) to (GLU479) STRUCTURAL AND BIOCHEMICAL ANALYSIS OF HUMAN PATHOGENIC ASTROVIRUS SERINE PROTEASE AT 2.0 ANGSTROM RESOLUTION | COILED COIL, TRANSMEMBRANE, THIOL PROTEASE, RNA REPLICATION, RIBOSOMAL FRAMESHIFTING, SERINE PROTEASE, CATALYTIC TRIAD, PROTEASE, MEMBRANE, HYDROLASE, ANTIVIRAL, ASTROVIRUS
2w5e:D (CYS438) to (GLU479) STRUCTURAL AND BIOCHEMICAL ANALYSIS OF HUMAN PATHOGENIC ASTROVIRUS SERINE PROTEASE AT 2.0 ANGSTROM RESOLUTION | COILED COIL, TRANSMEMBRANE, THIOL PROTEASE, RNA REPLICATION, RIBOSOMAL FRAMESHIFTING, SERINE PROTEASE, CATALYTIC TRIAD, PROTEASE, MEMBRANE, HYDROLASE, ANTIVIRAL, ASTROVIRUS
2w5e:E (CYS438) to (GLU479) STRUCTURAL AND BIOCHEMICAL ANALYSIS OF HUMAN PATHOGENIC ASTROVIRUS SERINE PROTEASE AT 2.0 ANGSTROM RESOLUTION | COILED COIL, TRANSMEMBRANE, THIOL PROTEASE, RNA REPLICATION, RIBOSOMAL FRAMESHIFTING, SERINE PROTEASE, CATALYTIC TRIAD, PROTEASE, MEMBRANE, HYDROLASE, ANTIVIRAL, ASTROVIRUS
1hb0:B (GLN30) to (GLY84) SNAPSHOTS OF SERINE PROTEASE CATALYSIS: (D) ACYL-ENZYME INTERMEDIATE BETWEEN PORCINE PANCREATIC ELASTASE AND HUMAN BETA-CASOMORPHIN-7 JUMPED TO PH 10 FOR 2 MINUTES | HYDROLASE, SERINE PROTEINASE, HYDROLASE (SERINE PROTEINASE)
1tbr:H (GLN30) to (MET84) CRYSTAL STRUCTURE OF INSECT DERIVED DOUBLE DOMAIN KAZAL INHIBITOR RHODNIIN IN COMPLEX WITH THROMBIN | COMPLEX (SERINE PROTEASE-INHIBITOR), KAZAL-TYPE INHIBITOR, THROMBIN, COMPLEX (SERINE PROTEASE-INHIBITOR) COMPLEX
1tfx:B (GLN30) to (ASN84) COMPLEX OF THE SECOND KUNITZ DOMAIN OF TISSUE FACTOR PATHWAY INHIBITOR WITH PORCINE TRYPSIN | COMPLEX (SERINE PROTEASE/INHIBITOR), HYDROLASE, INHIBITOR, BLOOD COAGULATION
1hdt:H (GLN30) to (MET84) STRUCTURE OF A RETRO-BINDING PEPTIDE INHIBITOR COMPLEXED WITH HUMAN ALPHA-THROMBIN | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1tgs:Z (GLN30) to (SER84) THREE-DIMENSIONAL STRUCTURE OF THE COMPLEX BETWEEN PANCREATIC SECRETORY INHIBITOR (KAZAL TYPE) AND TRYPSINOGEN AT 1.8 ANGSTROMS RESOLUTION. STRUCTURE SOLUTION, CRYSTALLOGRAPHIC REFINEMENT AND PRELIMINARY STRUCTURAL INTERPRETATION | COMPLEX (PROTEINASE/INHIBITOR)
1thr:H (GLN30) to (MET84) STRUCTURES OF THROMBIN COMPLEXES WITH A DESIGNED AND A NATURAL EXOSITE INHIBITOR | HYDROLASE(SERINE PROTEINASE)
1ths:H (GLN30) to (MET84) STRUCTURES OF THROMBIN COMPLEXES WITH A DESIGNED AND A NATURAL EXOSITE INHIBITOR | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1hgt:H (GLN30) to (MET84) STRUCTURE OF THE HIRUGEN AND HIRULOG 1 COMPLEXES OF ALPHA- THROMBIN | HYDROLASE(SERINE PROTEASE)
1hlt:H (GLN30) to (MET84) THE STRUCTURE OF A NONADECAPEPTIDE OF THE FIFTH EGF DOMAIN OF THROMBOMODULIN COMPLEXED WITH THROMBIN | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ton:A (GLN30) to (LEU84) RAT SUBMAXILLARY GLAND SERINE PROTEASE, TONIN. STRUCTURE SOLUTION AND REFINEMENT AT 1.8 ANGSTROMS RESOLUTION | HYDROLASE(SERINE PROTEINASE)
1tq0:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF THE POTENT ANTICOAGULANT THROMBIN MUTANT W215A/E217A IN FREE FORM | THROMBIN, ANTICOAGULANT, BLOOD CLOTTING
1hne:E (MET30) to (ALA84) STRUCTURE OF HUMAN NEUTROPHIL ELASTASE IN COMPLEX WITH A PEPTIDE CHLOROMETHYL KETONE INHIBITOR AT 1.84-ANGSTROMS RESOLUTION | HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4zxx:H (GLN30) to (ARG84) FACTOR VIIA IN COMPLEX WITH THE INHIBITOR N-{3-[(2R)-1-{(2R)-2-[(1- AMINOISOQUINOLIN-6-YL)AMINO]-2-PHENYLACETYL}PYRROLIDIN-2-YL]-4- (PROPAN-2-YLSULFONYL)PHENYL}ACETAMIDE | GLYCOPROTEIN, HYDROLASE, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM-BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4zxy:H (GLN30) to (ARG84) FACTOR VIIA IN COMPLEX WITH THE INHIBITOR (2R)-2-[(1-AMINOISOQUINOLIN- 6-YL)AMINO]-4,11-DIAZATRICYCLO[14.2.2.1~6,10~]HENICOSA-1(18),6(21),7, 9,16,19-HEXAENE-3,12-DIONE | GLYCOPROTEIN, HYDROLASE, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM-BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1hpl:B (HIS354) to (ALA417) HORSE PANCREATIC LIPASE. THE CRYSTAL STRUCTURE AT 2.3 ANGSTROMS RESOLUTION | HYDROLASE(CARBOXYLIC ESTERASE)
4lk4:A (ILE47) to (ALA107) STRUCTURE OF VIBRIO CHOLERAE VESB PROTEASE | TRYPSIN, PEPTIDASE S1 FAMILY, ENDOPEPTIDASE, DUF3466, SECRETED PROTEIN, EXTRACELLULAR, HYDROLASE
1trn:B (GLN30) to (ASN84) CRYSTAL STRUCTURE OF HUMAN TRYPSIN 1: UNEXPECTED PHOSPHORYLATION OF TYROSINE 151 | HUMAN TRYPSIN, DFP INHIBITED, HYDROLASE (SERINE PROTEINASE)
1try:A (PHE29) to (SER84) STRUCTURE OF INHIBITED TRYPSIN FROM FUSARIUM OXYSPORUM AT 1.55 ANGSTROMS | HYDROLASE (SERINE PROTEINASE)
2wfw:C (PRO80) to (THR136) STRUCTURE AND ACTIVITY OF THE N-TERMINAL SUBSTRATE RECOGNITION DOMAINS IN PROTEASOMAL ATPASES - THE ARC DOMAIN STRUCTURE | ATP-BINDING PROTEIN, PROTEASOMAL ATPASES, PAN, ARC, AAA, ATP-BINDING, NUCLEOTIDE-BINDING
2hlc:A (TYR29) to (ASN84) HL COLLAGENASE STRUCTURE AT 1.7A RESOLUTION | SERINE PROTEASE, HYDROLASE, COLLAGEN DEGRADATION
2hlc:B (TYR29) to (ASN84) HL COLLAGENASE STRUCTURE AT 1.7A RESOLUTION | SERINE PROTEASE, HYDROLASE, COLLAGEN DEGRADATION
2wiq:B (ASP141) to (ALA222) FLUORESCENT PROTEIN KILLERRED IN THE NATIVE STATE | FLUORESCENT PROTEIN, CALI, ROS, REACTIVE OXYGEN SPECIES
1txk:A (PRO77) to (LEU152) CRYSTAL STRUCTURE OF ESCHERICHIA COLI OPGG | BETA-SANDWICH, BIOSYNTHETIC PROTEIN
1hxe:H (GLN30) to (MET84) SERINE PROTEASE | SERINE PROTEASE IN BLOOD COAGULATION, HYDROLASE, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASEE-HYDROLASE INHIBITOR COMPLEX
1hxf:H (GLN30) to (MET84) HUMAN THROMBIN COMPLEX WITH HIRUDIN VARIANT | COMPLEX (SERINE PROTEASE INHIBITOR), SULFATATION, MULTIGENE FAMILY, BLOOD COAGULATION, PLASMA, CALCIUM-BINDING, GLYCOPROTEIN, DUPLICATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2hpp:H (GLN30) to (MET84) STRUCTURES OF THE NONCOVALENT COMPLEXES OF HUMAN AND BOVINE PROTHROMBIN FRAGMENT 2 WITH HUMAN PPACK-THROMBIN | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEINASE
3vxf:H (GLN30) to (MET84) X/N JOINT REFINEMENT OF HUMAN ALPHA-THROMBIN-BIVALIRUDIN COMPLEX PD5 | SERINE PROTEASE, HYDROLYSIS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lxb:H (GLN30) to (MET84) CRYSTAL STRUCTURE ANALYSIS OF THROMBIN IN COMPLEX WITH COMPOUND D58 | SERINE PROTEASES, ANTITHROMBOTIC AGENTS, DUAL THROMBIN/FACTOR XA INHI, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4lz1:H (GLN30) to (MET84) X-RAY STRUCTURE OF THE COMPLEX BETWEEN HUMAN THROMBIN AND THE TBA DELETION MUTANT LACKING THYMINE 12 NUCLEOBASE | PROTEIN-DNA COMPLEX, BLOOD COAGULATION, APTAMER, INHIBITOR-DNA COMPLEX, DNA APTAMER, G-QUADRUPLEX, SERINE PROTEASE, HYDROLASE, ABASIC FURAN, DNA THYMINE NUCLEOBASE DELETION, BLOOD, HYDROLASE-DNA COMPLEX, HYDROLASE-HYDROLASE INHIBITOR-DNA COMPLEX
1icj:B (GLU579) to (GLY624) PDF PROTEIN IS CRYSTALLIZED AS NI2+ CONTAINING FORM, COCRYSTALLIZED WITH INHIBITOR POLYETHYLENE GLYCOL (PEG) | HYDROLASE, IRON METALLOPROTEASE, PROTEIN SYNTHESIS
1uhb:A (GLN30) to (ASN84) CRYSTAL STRUCTURE OF PORCINE ALPHA TRYPSIN BOUND WITH AUTO CATALYTICALY PRODUCED NATIVE PEPTIDE AT 2.15 A RESOLUTION | SERINE PROTEASE, HYDROLASE, PEPTIDE TRYPSIN COMPLEX
2wvx:A (THR209) to (PHE253) STRUCTURE OF THE FAMILY GH92 INVERTING MANNOSIDASE BT3990 FROM BACTEROIDES THETAIOTAOMICRON VPI-5482 | GLYCOSIDE HYDROLASE FAMILY 92, GH92, HYDROLASE, BT3990
2wvx:D (THR209) to (PHE253) STRUCTURE OF THE FAMILY GH92 INVERTING MANNOSIDASE BT3990 FROM BACTEROIDES THETAIOTAOMICRON VPI-5482 | GLYCOSIDE HYDROLASE FAMILY 92, GH92, HYDROLASE, BT3990
4m37:A (ASN258) to (SER314) CRYSTAL STRUCTURE OF TRYPANOSOMA BRUCEI PROTEIN ARGININE METHYLTRANSFERASE 7 COMPLEX WITH ADOHCY | METHYLTRANSFERASE, TRANSFERASE
4m38:B (ASN258) to (SER314) CRYSTAL STRUCTURE OF TRYPANOSOMA BRUCEI PROTEIN ARGININE METHYLTRANSFERASE 7 COMPLEX WITH ADOHCY AND HISTONE H4 PEPTIDE | METHYLTRANSFERASE, TRANSFERASE-TRANSFERASE SUBSTRATE COMPLEX
5a8x:A (MET30) to (ALA84) CRYSTAL STRUCTURE OF HUMAN NEUTROPHIL ELASTASE IN COMPLEX WITH A DIHYDROPYRIMIDONE INHIBITOR | TRYPSIN FAMILY FOLD, PROTEASE, HYDROLASE, HYDROLASE- INHIBITOR COMPLEX
1uma:H (GLN30) to (MET84) ALPHA-THROMBIN (HIRUGEN) COMPLEXED WITH NA-(N,N-DIMETHYLCARBAMOYL)- ALPHA-AZALYSINE | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEASE, KRINGLE, ALPHA-THROMBIN- HIRUGEN COMPLEX
1iqn:A (GLN30) to (GLU84) HUMAN COAGULATION FACTOR XA IN COMPLEX WITH M55192 | HYDROLASE, SERINE PROTEASE, BLOOD COAGULATION FACTOR, COMPLEX
4m7g:A (THR15) to (ASN73) STREPTOMYCES ERYTHRAEUS TRYPSIN | SERINE PROTEASE, HYDROLASE
3j26:F (THR196) to (GLN266) THE 3.5 A RESOLUTION STRUCTURE OF THE SPUTNIK VIROPHAGE BY CRYO-EM | DOUBLE JELLY-ROLL, SINGLE JELLY-ROLL, VIRUS
5abe:A (LEU659) to (GLU714) STRUCTURE OF GH84 WITH LIGAND | HYDROLASE, TIM-BARREL, INHIBITOR
5abf:A (LEU659) to (GLU714) STRUCTURE OF GH84 WITH LIGAND | HYDROLASE, TIM-BARREL, INHIBITOR
2wzs:G (THR209) to (PHE253) STRUCTURE OF THE FAMILY GH92 INVERTING MANNOSIDASE BT3990 FROM BACTEROIDES THETAIOTAOMICRON VPI-5482 IN COMPLEX WITH MANNOIMIDAZOLE | GLYCOSIDE HYDROLASE FAMILY 92, ALPHA-1\,2 LINKAGE, BT3990, HYDROLASE
1uto:A (GLN30) to (SER84) TRYPSIN SPECIFICITY AS ELUCIDATED BY LIE CALCULATIONS, X-RAY STRUCTURES AND ASSOCIATION CONSTANT MEASUREMENTS | HYDROLASE, TRYPSIN, INHIBITOR SPECIFICITY, ELECTROSTATIC INTERACTIONS, COLD-ADAPTATION, MOLECULAR DYNAMICS, BINDING FREE ENERGY
1utq:A (GLN30) to (SER84) TRYPSIN SPECIFICITY AS ELUCIDATED BY LIE CALCULATIONS, X-RAY STRUCTURES AND ASSOCIATION CONSTANT MEASUREMENTS | HYDROLASE, TRYPSIN, INHIBITOR SPECIFICITY, ELECTROSTATIC INTERACTIONS, COLD-ADAPTATION, MOLECULAR DYNAMICS, BINDING FREE ENERGY HYDROLASE
1j15:A (GLN30) to (ASN84) BENZAMIDINE IN COMPLEX WITH RAT TRYPSIN MUTANT X99/175/190RT | SERINE PROTEASE, HYDROLASE, SERINE PROTEINASE
4mho:A (LEU198) to (THR240) CRYSTAL STRUCTURE OF GPB IN COMPLEX WITH S3, SUGAR (N-[(BIPHENYL-4- YLOXY)ACETYL]-BETA-D-GLUCOPYRANOSYLAMINE) | ALPHA AND BETA PROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4mi3:A (LEU198) to (THR240) CRYSTAL STRUCTURE OF GPB IN COMPLEX WITH SUGAR (N-{(2R)-2-METHYL-3-[4- (PROPAN-2-YL)PHENYL]PROPANOYL}-BETA-D-GLUCOPYRANOSYLAMINE) (S21) | ALPHA AND BETA PROTEIN, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1v2l:T (GLN30) to (SER84) BENZAMIDINE IN COMPLEX WITH BOVINE TRYPSIN VARIANT X(TRIPLE.GLU)BT.D1 | SERINE PROTEASE, HYDROLASE, SERINE PROTEINASE
1v2m:T (GLN30) to (SER84) BENZAMIDINE IN COMPLEX WITH BOVINE TRYPSIN VARIANT X(TRIPLE.GLU)BT.A1 | SERINE PROTEASE, HYDROLASE, SERINE PROTEINASE
1vgc:B (GLN30) to (LYS84) GAMMA-CHYMOTRYPSIN L-PARA-CHLORO-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX | HYDROLASE, SERINE PROTEASE
1jnq:A (SER57) to (VAL128) LIPOXYGENASE-3 (SOYBEAN) COMPLEX WITH EPIGALLOCATHECHIN (EGC) | METALLOPROTEIN, FE(II) COMPLEX, PURPLE LIPOXYGENASE, CATECHIN INHIBITOR, GREEN TEA, OXIDOREDUCTASE
2j97:A (THR14) to (GLU64) HUMAN CORONAVIRUS 229E NON STRUCTURAL PROTEIN 9 (NSP9) | SSB, ZINC, HCOV, MEMBRANE, HELICASE, SARS COV, VIRAL REPLICASE, RNA REPLICATION, ATP-BINDING, NUCLEOTIDE-BINDING, RIBOSOMAL FRAMESHIFT, RNA-BINDING PROTEIN
1jwt:A (GLN51) to (MET116) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH A NOVEL BICYCLIC LACTAM INHIBITOR | HYDROLASE
1jym:C (VAL142) to (GLY188) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | PDF, MALARIA, PLASMODIUM, DEFORMYLATION, METALLOENZYME, HYDROLASE
1jym:E (VAL142) to (GLY188) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | PDF, MALARIA, PLASMODIUM, DEFORMYLATION, METALLOENZYME, HYDROLASE
1jym:F (VAL142) to (GLY188) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | PDF, MALARIA, PLASMODIUM, DEFORMYLATION, METALLOENZYME, HYDROLASE
1jym:G (VAL142) to (GLY188) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | PDF, MALARIA, PLASMODIUM, DEFORMYLATION, METALLOENZYME, HYDROLASE
1jym:J (VAL142) to (GLY188) CRYSTALS OF PEPTIDE DEFORMYLASE FROM PLASMODIUM FALCIPARUM WITH TEN SUBUNITS PER ASYMMETRIC UNIT REVEAL CRITICAL CHARACTERISTICS OF THE ACTIVE SITE FOR DRUG DESIGN | PDF, MALARIA, PLASMODIUM, DEFORMYLATION, METALLOENZYME, HYDROLASE
4n3l:H (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH A NOVEL GLUCOSE- CONJUGATED POTENT INHIBITOR | HYDROLASE(SERINE PROTEASE), COMPLEX THROMBIN-GLUCOSE-CONJUGATED INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3zcq:A (LEU198) to (THR240) RABBIT MUSCLE GLYCOGEN PHOSPHORYLASE B IN COMPLEX WITH N-(4- TRIFLUOROMETHYL-BENZOYL)-N-BETA-D-GLUCOPYRANOSYL UREA DETERMINED AT 2.15 A RESOLUTION | TRANSFERASE, INHIBITOR, HYPOGLYCAEMIC AGENTS, STRUCTURE-BASED LIGAND DESIGN
2jet:B (GLN30) to (LYS84) CRYSTAL STRUCTURE OF A TRYPSIN-LIKE MUTANT (S189D, A226G) CHYMOTRYPSIN. | SUBSTRATE SPECIFICITY, ZYMOGEN, PROTEASE, HYDROLASE, DIGESTION, SERINE PROTEASE, PROTEIN ENGINEERING
2jh5:D (GLN30) to (MET84) HUMAN THROMBIN HIRUGEN INHIBITOR COMPLEX | GLYCOPROTEIN, SERINE PROTEASE, KRINGLE, ZYMOGEN, THROMBIN, PROTEASE, DISEASE MUTATION, BLOOD COAGULATION, GAMMA-CARBOXYGLUTAMIC ACID, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, SULFATION, ACUTE PHASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2xvg:A (THR809) to (ALA850) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE (GH31) FROM CELLVIBRIO JAPONICUS | HYDROLASE, GLYCOSYL HYDROLASE FAMILY 31, BETA/ALPHA 8 BARREL
2xvk:A (THR809) to (ALA850) CRYSTAL STRUCTURE OF ALPHA-XYLOSIDASE (GH31) FROM CELLVIBRIO JAPONICUS IN COMPLEX WITH 5-FLUORO-ALPHA-D-XYLOPYRANOSYL FLUORIDE | HYDROLASE, GLYCOSYL HYDROLASE FAMILY 31, (BETA/ALPHA) 8 BARREL
1w8o:A (GLU584) to (ALA639) CONTRIBUTION OF THE ACTIVE SITE ASPARTIC ACID TO CATALYSIS IN THE BACTERIAL NEURAMINIDASE FROM MICROMONOSPORA VIRIDIFACIENS | 3D-STRUCTURE, GLYCOSIDASE, HYDROLASE, SIALIDASE, BETA- PROPELLER
2xwb:F (ALA472) to (HIS531) CRYSTAL STRUCTURE OF COMPLEMENT C3B IN COMPLEX WITH FACTORS B AND D | IMMUNE SYSTEM, PRO-CONVERTASE, HYDROLASE, SERINE PROTEASE, CONFORMATIONAL CHANGES, ALTERNATIVE PATHWAY
2xwb:H (ALA472) to (HIS531) CRYSTAL STRUCTURE OF COMPLEMENT C3B IN COMPLEX WITH FACTORS B AND D | IMMUNE SYSTEM, PRO-CONVERTASE, HYDROLASE, SERINE PROTEASE, CONFORMATIONAL CHANGES, ALTERNATIVE PATHWAY
1w9w:A (ASP21) to (ASP70) STRUCTURE OF A BETA-1,3-GLUCAN BINDING CBM6 FROM BACILLUS HALODURANS IN COMPLEX WITH LAMINARIHEXAOSE | CARBOHYDRATE-BINDING MODULE, LECTIN, BETA-GLUCAN, CARBOHYDRATE BINDING, GLYCOSIDE HYDROLASE
1k2i:1 (GLN30) to (LYS84) CRYSTAL STRUCTURE OF GAMMA-CHYMOTRYPSIN IN COMPLEX WITH 7- HYDROXYCOUMARIN | ENZYME-INHIBITOR COMPLEX, HYDROLASE
1k32:B (ASN145) to (ARG194) CRYSTAL STRUCTURE OF THE TRICORN PROTEASE | PROTEIN DEGRADATION, SUBSTRATE GATING, SERINE PROTEASE, BETA PROPELLER, PROTEASOME, HYDROLASE
2k1q:A (GLN34) to (GLN73) NMR STRUCTURE OF HEPATITIS C VIRUS NS3 SERINE PROTEASE COMPLEXED WITH THE NON-COVALENTLY BOUND PHENETHYLAMIDE INHIBITOR | SERINE PROTEASE, NS3, HEPATITIS C VIRUS, NON COVALENT INHIBITOR, ENVELOPE PROTEIN, HELICASE, HYDROLASE, NUCLEOTIDE-BINDING, RNA REPLICATION, TRANSMEMBRANE, VIRAL PROTEIN
4niy:A (GLN30) to (SER84) CRYSTAL STRUCTURE OF TRYPSILIGASE (K60E/N143H/Y151H/D189K TRYPSIN) COMPLEXED TO YRH-ECOTIN (M84Y/M85R/A86H ECOTIN) | TRYPSIN INHIBITOR, SERINE PROTEINASE, ENZYME DESIGN, ACTIVATION DOMAIN, PEPTIDE LIGATION, REVERSE PROTEOLYSIS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4niy:D (GLN30) to (SER84) CRYSTAL STRUCTURE OF TRYPSILIGASE (K60E/N143H/Y151H/D189K TRYPSIN) COMPLEXED TO YRH-ECOTIN (M84Y/M85R/A86H ECOTIN) | TRYPSIN INHIBITOR, SERINE PROTEINASE, ENZYME DESIGN, ACTIVATION DOMAIN, PEPTIDE LIGATION, REVERSE PROTEOLYSIS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2y4y:C (GLY106) to (THR169) STRUCTURE OF A DOMAIN FROM THE TYPE IV PILUS BIOGENESIS LIPOPROTEIN PILP, FROM PSEUDOMONAS AERUGINOSA | BIOSYNTHETIC PROTEIN
1kf9:F (GLN1565) to (PHE1623) PHAGE DISPLAY DERIVED VARIANT OF HUMAN GROWTH HORMONE COMPLEXED WITH TWO COPIES OF THE EXTRACELLULAR DOMAIN OF ITS RECEPTOR | CYTOKINE, HORMONE-RECEPTOR COMPLEX, PHAGE DISPLAY MOLECULAR PLASTICITY, RECEPTOR HOMODIMERIZATION, HUMAN GROWTH HORMONE, HORMONE/GROWTH FACTOR COMPLEX
1wsr:A (SER306) to (LYS363) CRYSTAL STRUCTURE OF HUMAN T-PROTEIN OF GLYCINE CLEAVAGE SYSTEM | GLYCINE-CLEAVAGE SYTEM, AMINOMETHYL TRANSFERASE
1wsv:B (SER306) to (LYS363) CRYSTAL STRUCTURE OF HUMAN T-PROTEIN OF GLYCINE CLEAVAGE SYSTEM | GLYCINE-CLEAVAGE SYTEM, AMINOMETHYL TRANSFERASE
1kj1:D (GLY52) to (SER100) MANNOSE-SPECIFIC AGGLUTININ (LECTIN) FROM GARLIC (ALLIUM SATIVUM) BULBS COMPLEXED WITH ALPHA-D-MANNOSE | BULB LECTIN, MANNOSE, PLANT PROTEIN
1kj1:Q (GLY52) to (SER100) MANNOSE-SPECIFIC AGGLUTININ (LECTIN) FROM GARLIC (ALLIUM SATIVUM) BULBS COMPLEXED WITH ALPHA-D-MANNOSE | BULB LECTIN, MANNOSE, PLANT PROTEIN
4nu3:B (ALA47) to (ASP84) CRYSTAL STRUCTURE OF MFFIBP, A CAPPING HEAD REGION SWAPPED MUTANT OF ICE-BINDING PROTEIN | BETA-HELICAL, ANTIFREEZE ACTIVITY, ICE-CRYSTAL, ANTIFREEZE PROTEIN
1kts:B (GLN30) to (MET84) THROMBIN INHIBITOR COMPLEX | BLOOD COAGULATION, INHIBITION, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4nzl:A (MET44) to (ALA100) EXTRACELLULAR PROTEINS OF STAPHYLOCOCCUS AUREUS INHIBIT THE NEUTROPHIL SERINE PROTEASES | PRIMARILY BETA, SERINE PROTEASE, PROTEASE INHIBITOR, INNATE IMMUNITY, AZUROPHILIC GRANULES, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1kyn:A (ALA31) to (THR84) CATHEPSIN-G | SERINE PROTEASE, HYDROLASE
4o03:A (GLN335) to (MET400) CRYSTAL STRUCTURE OF CA2+ BOUND PROTHROMBIN DELETION MUTANT RESIDUES 146-167 | PROTHROMBIN, KRINGLE, SERINE PROTEASE, COAGULATION, HYDROLASE
1xen:A (ASN74) to (GLY124) HIGH RESOLUTION CRYSTAL STRUCTURE OF ESCHERICHIA COLI IRON- PEPTIDE DEFORMYLASE BOUND TO FORMATE | IRON DEFORMYLASE, FORMATE, HYDROLASE
1xeo:A (ASN74) to (GLY124) HIGH RESOLUTION CRYSTALS STRUCTURE OF COBALT- PEPTIDE DEFORMYLASE BOUND TO FORMATE | COBALT DEFORMYLASE, FORMATE, HYDROLASE
1l1g:A (GLN15) to (GLY73) THE STRUCTURE OF PORCINE PANCREATIC ELASTASE COMPLEXED WITH XENON AND BROMIDE, CRYOPROTECTED WITH GLYCEROL | XENON, BROMIDE, PPE, HYDROLASE
1l2e:A (GLN30) to (SER84) HUMAN KALLIKREIN 6 (HK6) ACTIVE FORM WITH BENZAMIDINE INHIBITOR | SERINE PROTEASE, KALLIKREIN, HUMAN KALLIKREIN 6, BENZAMIDINE, PROTEASE, MYELENCEPHALON SPECIFIC PROTEASE, ZYME, PROTEASE M, NEUROSIN, HYDROLASE
4o3u:A (MET508) to (ASN566) ZYMOGEN HGF-BETA/MET WITH ZYMOGEN ACTIVATOR PEPTIDE ZAP2.3 | TRYPSIN HOMOLOY, RECEPTOR ACTIVATION, TRANSFERASE-GROWTH FACTOR COMPLEX
1l4z:A (GLN576) to (GLU634) X-RAY CRYSTAL STRUCTURE OF THE COMPLEX OF MICROPLASMINOGEN WITH ALPHA DOMAIN OF STREPTOKINASE IN THE PRESENCE CADMIUM IONS | PLASMINOGEN, STREPTOKINASE, PROTEIN COMPLEX, CRYSTAL STRUCTURE, HYDROLASE/BLOOD CLOTTING COMPLEX
4o9v:A (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MATRIPTASE IN COMPLEX WITH INHIBITOR | MATRIPTASE, TRYPSIN-LIKE SERINE PROTEINASE FOLD, PROTEASE, SMALL MOLECULE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1lhc:H (GLN30) to (MET84) HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BOROARG-OH | BLOOD COAGULATION, PLASMA, CALCIUM-BINDING, GLYCOPROTEIN, DUPLICATION, VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE, KRINGLE, SIGNAL, DISEASE MUTATION, COMPLEX (SERINE PROTEASE/INHIBITOR)
1lhf:H (GLN30) to (MET84) HUMAN ALPHA-THROMBIN COMPLEXED WITH AC-(D)PHE-PRO-BORO- HOMOLYS-OH | BLOOD COAGULATION, PLASMA, CALCIUM-BINDING, GLYCOPROTEIN, DUPLICATION, VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE, KRINGLE, SIGNAL, DISEASE MUTATION, COMPLEX (SERINE PROTEASE/INHIBITOR)
1lnh:A (SER57) to (VAL128) LIPOXYGENASE-3(SOYBEAN) NON-HEME FE(II) METALLOPROTEIN | OXIDOREDUCTASE, METALLOPROTEIN, FE(II) COMPLEX
1lo6:A (GLN30) to (SER84) HUMAN KALLIKREIN 6 (HK6) ACTIVE FORM WITH BENZAMIDINE INHIBITOR AT 1.56 A RESOLUTION | SERINE PROTEASE, KALLIKREIN, HUMAN KALLIKREIN 6, HK6, BENZAMIDINE, PROTEASE, BRAIN SERINE PROTEASE, MYELENCEPHALON SPECIFIC PROTEASE, MSP, ZYME, PROTEASE M, NEUROSIN, HYDROLASE
1lpa:B (HIS354) to (ALA417) INTERFACIAL ACTIVATION OF THE LIPASE-PROCOLIPASE COMPLEX BY MIXED MICELLES REVEALED BY X-RAY CRYSTALLOGRAPHY | HYDROLASE(CARBOXYLIC ESTERASE)
4a5t:S (GLN576) to (GLU634) STRUCTURAL BASIS FOR THE CONFORMATIONAL MODULATION | HYDROLASE, MULTI-DOMAIN CONFORMATIONAL CHANGE
2zcl:P (GLN30) to (GLN84) CRYSTAL STRUCTURE OF HUMAN PROSTATE SPECIFIC ANTIGEN COMPLEXED WITH AN ACTIVATING ANTIBODY | HUMAN PSA, ANTIBODIES, KALLIKREIN RELATED PEPTIDASES, PROSTATE CANCER, GLYCOPROTEIN, HYDROLASE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, IMMUNE SYSTEM
2o7i:A (MET37) to (TYR70) THE X-RAY CRYSTAL STRUCTURE OF A THERMOPHILIC CELLOBIOSE BINDING PROTEIN BOUND WITH CELLOBIOSE | PERIPLASMIC BINDING PROTEIN, CELLULOSE, THERMOPHILIC PROTEINS, CELLOBIOSE BINDING PROTEIN, SUGAR BINDING PROTEIN
2zf0:H (GLN30) to (MET84) EXPLORING THROMBIN S1 POCKET | BLOOD CLOTTING/HYDROLASE INHIBITORS, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
2zfp:H (GLN30) to (MET84) THROMBIN INIBITION | BLOOD CLOTTING/HYDROLASE INHIBITOR, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
2zfq:H (GLN30) to (MET84) EXPLORING THROMBIN S3 POCKET | BLOOD COAGULATION/HYDROLASE INHIBITORS, ACUTE PHASE, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, SULFATION, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
2zgb:H (GLN30) to (MET84) THROMBIN INHIBITION | BLOOD CLOTTING, HYDROLASE INHIBITOR, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2zhe:H (GLN30) to (MET84) EXPLORING THROMBIN S3 POCKET | BLOOD COAGULATION, HYDROLASE INHIBITORS, ACUTE PHASE, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, SULFATION, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3kcg:H (VAL31) to (ASN84) CRYSTAL STRUCTURE OF THE ANTITHROMBIN-FACTOR IXA- PENTASACCHARIDE COMPLEX | MICHAELIS COMPLEX, BLOOD COAGULATION, CALCIUM, DISULFIDE BOND, EGF-LIKE DOMAIN, GLYCOPROTEIN, HEMOPHILIA, HYDROLASE, PHARMACEUTICAL, PROTEASE, SECRETED, SERINE PROTEASE, SULFATION, ZYMOGEN, HEPARIN-BINDING, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, THROMBOPHILIA
4oqw:H (LEU138) to (ARG220) CRYSTAL STRUCTURE OF MCARDINAL FAR-RED FLUORESCENT PROTEIN | FLUORESCENT PROTEIN
1xug:A (GLN30) to (SER84) TRYPSIN-BABIM-ZN+2, PH 8.2 | COMPLEX, TRYPSIN-ZN+2-SMALL MOLECULE LIGAND, DESIGNED SMALL MOLECULE LIGAND WITH NANOMOLAR AFFINITY, SERINE PROTEASE
2znk:H (GLN30) to (MET84) THROMBIN INHIBITION | BLOOD CLOTTING, HYDROLASE INHIBITOR, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SERINE PROTEASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
2zo6:A (SER141) to (ALA212) CRYSTAL STRUCTURE OF KUSABIRA-CYAN (KCY), A CYAN-EMITTING GFP-LIKE PROTEIN | GFP-LIKE PROTEIN, LUMINESCENT PROTEIN, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES
2zo7:A (SER142) to (ALA213) CRYSTAL STRUCTURE OF A KUSABIRA-CYAN MUTANT (KCY-R1), A CYAN/GREEN- EMITTING GFP-LIKE PROTEIN | GFP-LIKE PROTEIN, LUMINESCENT PROTEIN, STRUCTURAL GENOMICS, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES
1xvm:A (ILE30) to (SER83) TRYPSIN FROM FUSARIUM OXYSPORUM- ROOM TEMPERATURE TO ATOMIC RESOLUTION | ATOMIC RESOLUTION, MOBILITY, ROOM TEMPERATURE, HYDROLASE
1xvo:A (ILE30) to (SER83) TRYPSIN FROM FUSARIUM OXYSPORUM AT PH 6 | TRYPSIN, ATOMIC RESOLUTION, HYDROLASE
2zp0:H (GLN30) to (ARG84) HUMAN FACTOR VIIA-TISSUE FACTOR COMPLEXED WITH BENZYLSULFONAMIDE-D- ILE-GLN-P-AMINOBENZAMIDINE | SERINE PROTEASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, EGF-LIKE DOMAIN, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, HYDROXYLATION, PROTEASE, ZYMOGEN, LIPOPROTEIN, MEMBRANE, PALMITATE, TRANSMEMBRANE, HYDROLASE-BLOOD CLOTTING COMPLEX
3khv:A (PHE30) to (GLU84) CRYSTAL STRUCTURES OF UROKINASE-TYPE PLASMINOGEN ACTIVATOR IN COMPLEX WITH 4-(AMINOMETHYL) BENZOIC ACID AND 4- (AMINOMETHYL-PHENYL)-METHANOL | PROTEIN-LIGAND COMPLEX, DISULFIDE BOND, FIBRINOLYSIS, HYDROLASE, PLASMINOGEN ACTIVATION, SERINE PROTEASE
4ab8:A (GLN30) to (SER84) FRAGMENTS BOUND TO BOVINE TRYPSIN FOR THE SAMPL CHALLENGE | HYDROLASE, FRAGMENT SCREENING, MODELLING
4abg:A (GLN30) to (SER84) FRAGMENTS BOUND TO BOVINE TRYPSIN FOR THE SAMPL CHALLENGE | HYDROLASE, FRAGMENT SCREENING, MODELLING
1max:A (GLN30) to (SER84) BETA-TRYPSIN PHOSPHONATE INHIBITED | HYDROLASE, SERINE PROTEASE, DIGESTION, PANCREAS, ZYMOGEN, HYDROLASE (SERINE PROTEASE)
1mbm:A (GLY13) to (THR57) NSP4 PROTEINASE FROM EQUINE ARTERITIS VIRUS | SERINE PROTEINASE, CHYMOTRYPSIN-LIKE PROTEINASE, COLLAPSED OXYANION HOLE, TRANSFERASE
1mbm:A (GLY91) to (THR139) NSP4 PROTEINASE FROM EQUINE ARTERITIS VIRUS | SERINE PROTEINASE, CHYMOTRYPSIN-LIKE PROTEINASE, COLLAPSED OXYANION HOLE, TRANSFERASE
1mbm:B (GLY13) to (THR57) NSP4 PROTEINASE FROM EQUINE ARTERITIS VIRUS | SERINE PROTEINASE, CHYMOTRYPSIN-LIKE PROTEINASE, COLLAPSED OXYANION HOLE, TRANSFERASE
1mbm:C (GLY13) to (THR57) NSP4 PROTEINASE FROM EQUINE ARTERITIS VIRUS | SERINE PROTEINASE, CHYMOTRYPSIN-LIKE PROTEINASE, COLLAPSED OXYANION HOLE, TRANSFERASE
1mbm:D (GLY13) to (LEU56) NSP4 PROTEINASE FROM EQUINE ARTERITIS VIRUS | SERINE PROTEINASE, CHYMOTRYPSIN-LIKE PROTEINASE, COLLAPSED OXYANION HOLE, TRANSFERASE
4afq:A (TYR14) to (GLU71) HUMAN CHYMASE - FYNOMER COMPLEX | HYDROLASE-DE NOVO PROTEIN COMPLEX, INHIBITOR, SERINE PROTEASE
4afs:A (TYR14) to (GLU71) HUMAN CHYMASE - FYNOMER COMPLEX | HYDROLASE-DE NOVO PROTEIN COMPLEX, INHIBITOR, SERINE PROTEASE
3kqd:A (GLN30) to (GLU84) FACTOR XA IN COMPLEX WITH THE INHIBITOR 1-(3-(5-OXO-4,5- DIHYDRO-1H-1, 2,4-TRIAZOL-3-YL)PHENYL)-6-(2'-(PYRROLIDIN-1- YLMETHYL)BIPHENYL-4- YL)-3-(TRIFLUOROMETHYL)-5,6-DIHYDRO- 1H-PYRAZOLO[3,4-C]PYRIDIN-7(4H)- ONE | GLYCOPROTEIN, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM- BINDING, BLOOD COAGULATION, CALCIUM, PROTEASE, SECRETED, EGF-LIKE DOMAIN, GAMMA-CARBOXYGLUTAMIC ACID, HYDROLASE
1yc0:A (ALA423) to (GLY478) SHORT FORM HGFA WITH FIRST KUNITZ DOMAIN FROM HAI-1 | HYDROLASE/INHIBITOR, HYDROLASE-INHIBITOR COMPLEX
1mtn:F (GLN30) to (LYS84) BOVINE ALPHA-CHYMOTRYPSIN:BPTI CRYSTALLIZATION | COMPLEX, PROTEASE INHIBITOR, TRYPSIN, HYDROLASE, SERINE, COMPLEX (HYDROLASE/INHIBITOR) COMPLEX
1mu6:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH L-378,622 | HYDROLASE, BLOOD CLOTTING, HYDROLASE-BLOOD CLOTTING COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, BLOOD CLOTTING,HYDROLASE- INHIBITOR COMPLEX
1mu8:B (GLN30) to (MET84) THROMBIN-HIRUGEN_L-378,650 | THROMBIN-HIRUGEN, BLOOD CLOTTING, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1mue:B (GLN30) to (MET84) THROMBIN-HIRUGEN-L405,426 | ALPHA THROMBIN-HIRUGEN, BLOOD CLOTTING COMPLEX,HYDROLASE INHIBITOR COMPLEX, HYDROLASE INHIBITOR
1ylc:A (GLN30) to (ASN84) TRYPSIN/BPTI COMPLEX MUTANT | TRYPSIN II, PANCREATIC TRYPSIN INHIBITOR, BPTI, HYDROLASE/INHIBITOR COMPLEX
1ynj:D (MET351) to (LYS397) TAQ RNA POLYMERASE-SORANGICIN COMPLEX | TRANSFERASE
1ype:H (GLN30) to (MET84) THROMBIN INHIBITOR COMPLEX | THROMBIN, INHIBITOR COMPLEX, BARREL, 6 STRANDED BETA-SHEET, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
1yph:C (GLN30) to (LYS84) HIGH RESOLUTION STRUCTURE OF BOVINE ALPHA-CHYMOTRYPSIN | SERINE PROTEASE, HYDROLASE
1yph:D (GLN30) to (LYS84) HIGH RESOLUTION STRUCTURE OF BOVINE ALPHA-CHYMOTRYPSIN | SERINE PROTEASE, HYDROLASE
1ypo:G (GLY205) to (GLU254) HUMAN OXIDIZED LOW DENSITY LIPOPROTEIN RECEPTOR LOX-1 P3 1 21 SPACE GROUP | OXIDIZED LOW DENSITY LIPOPROTEIN RECEPTOR, LOX-1,CTLD, C- TYPE LECTIN LIKE DOMAIN, NK CELL RECEPTOR, IMMUNE SYSTEM
5dgr:A (HIS30) to (ALA85) CRYSTAL STRUCTURE OF GH9 EXO-BETA-D-GLUCOSAMINIDASE PBPRA0520, GLUCOSAMINE COMPLEX | GLYCOSIDE HYDROLASE FAMILY 9, ALPHA-ALPHA-6 BARREL, EXO-D-BETA- GLUCOSAMINIDASE, HYDROLASE
5dgr:B (HIS30) to (ALA85) CRYSTAL STRUCTURE OF GH9 EXO-BETA-D-GLUCOSAMINIDASE PBPRA0520, GLUCOSAMINE COMPLEX | GLYCOSIDE HYDROLASE FAMILY 9, ALPHA-ALPHA-6 BARREL, EXO-D-BETA- GLUCOSAMINIDASE, HYDROLASE
5dgq:B (HIS30) to (ALA85) CRYSTAL STRUCTURE OF GH9 EXO-BETA-D-GLUCOSAMINIDASE PBPRA0520 | GLYCOSIDE HYDROLASE FAMILY 9, ALPHA-ALPHA-6 BARREL, EXO-D-BETA- GLUCOSAMINIDASE, HYDROLASE
3l33:D (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH AMYLOID PRECURSOR PROTEIN INHIBITOR(APPI) | HUMAN MESOTRYPSIN, ALZHEIMER'S AMYLOID PRECURSOR PROTEIN INHIBITOR, APPI, SERINE PROTEASE INHIBITOR, HYDROLASE-CELL ADHESION COMPLEX
3l5n:A (VAL365) to (VAL427) STAPHYLOCOCCAL COMPLEMENT INHIBITOR (SCIN) IN COMPLEX WITH HUMAN COMPLEMENT COMPONENT C3B | COMPLEMENT ALTERNATE PATHWAY, COMPLEMENT PATHWAY, CONVERSTASE, IMMUNE RESPONSE, INFLAMMATORY RESPONSE, INNATE IMMUNITY, SECRETED, VIRULENCE, IMMUNE EVASION, IMMUNE SYSTEM
1n6e:A (ASN145) to (ARG194) TRICORN PROTEASE IN COMPLEX WITH A TRIDECAPEPTIDE CHLOROMETHYL KETONE DERIVATIVE | TRICORN PROTEASE, HYDROLASE, PROPELLER
1n6e:C (ASN145) to (ARG194) TRICORN PROTEASE IN COMPLEX WITH A TRIDECAPEPTIDE CHLOROMETHYL KETONE DERIVATIVE | TRICORN PROTEASE, HYDROLASE, PROPELLER
1n6e:E (ASN145) to (ARG194) TRICORN PROTEASE IN COMPLEX WITH A TRIDECAPEPTIDE CHLOROMETHYL KETONE DERIVATIVE | TRICORN PROTEASE, HYDROLASE, PROPELLER
1n6e:G (ASN145) to (ARG194) TRICORN PROTEASE IN COMPLEX WITH A TRIDECAPEPTIDE CHLOROMETHYL KETONE DERIVATIVE | TRICORN PROTEASE, HYDROLASE, PROPELLER
1n6e:K (ASN145) to (ARG194) TRICORN PROTEASE IN COMPLEX WITH A TRIDECAPEPTIDE CHLOROMETHYL KETONE DERIVATIVE | TRICORN PROTEASE, HYDROLASE, PROPELLER
3lc3:A (GLN30) to (ASN84) BENZOTHIOPHENE INHIBITORS OF FACTOR IXA | PROTEIN-INHIBITOR COMPLEX, PEPTIDASE S1, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, EGF-LIKE DOMAIN, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HEMOPHILIA, HYDROLASE, HYDROXYLATION, PHARMACEUTICAL, PHOSPHOPROTEIN, POLYMORPHISM, PROTEASE, SECRETED, SERINE PROTEASE, SULFATION, ZYMOGEN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3lc3:C (GLN30) to (ASN84) BENZOTHIOPHENE INHIBITORS OF FACTOR IXA | PROTEIN-INHIBITOR COMPLEX, PEPTIDASE S1, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, EGF-LIKE DOMAIN, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HEMOPHILIA, HYDROLASE, HYDROXYLATION, PHARMACEUTICAL, PHOSPHOPROTEIN, POLYMORPHISM, PROTEASE, SECRETED, SERINE PROTEASE, SULFATION, ZYMOGEN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1z7k:A (GLN30) to (ASN84) CRYSTAL STRUCTURE OF TRYPSIN- OVOMUCOID TURKEY EGG WHITE INHIBITOR COMPLEX | SERINE PROTEASE, HYDROLASE, PROTEASE INHIBITOR, DI-NAG, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1z9s:A (GLY180) to (LYS231) CRYSTAL STRUCTURE OF THE NATIVE CHAPERONE:SUBUNIT:SUBUNIT CAF1M:CAF1:CAF1 COMPLEX | DONOR STRAND COMPLEMENTATION, NATIVE MINIMAL FIBER, CHAPERONE-USHER PATHWAY, CHAPERONE/IMMUNE SYSTEM COMPLEX
1zgi:A (GLN30) to (MET84) THROMBIN IN COMPLEX WITH AN OXAZOLOPYRIDINE INHIBITOR 21 | THROMBIN, THROMBIN INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1zgv:A (GLN30) to (MET84) THROMBIN IN COMPLEX WITH AN OXAZOLOPYRIDINE INHIBITOR 2 | THROMBIN, THROMBIN INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4arx:C (ASN480) to (VAL536) LEPIDOPTERA-SPECIFIC TOXIN CRY1AC FROM BACILLUS THURINGIENSIS SSP. KURSTAKI HD-73 | TOXIN, MEMBRANE PORE-FORMING TOXIN, INSECTICIDAL PROTEIN LEPIDOPTERAN SPECIFICITY, RECEPTOR BINDING SITE
4q2k:B (GLN30) to (LYS84) BOVINE ALPHA CHYMOTRYPSIN BOUND TO A CYCLIC PEPTIDE INHIBITOR, 5B | CHYMOTRYPSIN, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4q2k:C (GLN30) to (LYS84) BOVINE ALPHA CHYMOTRYPSIN BOUND TO A CYCLIC PEPTIDE INHIBITOR, 5B | CHYMOTRYPSIN, PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5dzx:B (ARG35) to (ASN99) PROTOCADHERIN BETA 6 EXTRACELLULAR CADHERIN DOMAINS 1-4 | CADHERIN, DIMER, EXTRACELLULAR, CELL ADHESION
1zrb:A (GLN30) to (MET84) THROMBIN IN COMPLEX WITH AN AZAFLUORENYL INHIBITOR 23B | THROMBIN; THROMBIN INHIBITOR COMPLEX, BLOOD CLOTTING, HYDROLASE- INHIBITOR COMPLEX, BLOOD CLOTTING,HYDROLASE-INHIBITOR COMPLEX
5e2o:A (GLN30) to (HIS91) FACTOR XIA IN COMPLEX WITH THE INHIBITOR 4-[(N-{(2E)-3-[5-CHLORO-2- (1H-TETRAZOL-1-YL)PHENYL]PROP-2-ENOYL}-L-PHENYLALANYL)AMINO]BENZOIC ACID | HYDROLASE, SERINE PROTEASE, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3lt3:B (LYS206) to (GLU253) CRYSTAL STRUCTURE OF RV3671C FROM M. TUBERCULOSIS H37RV, SER343ALA MUTANT, INACTIVE FORM | SERINE PROTEASE, H37RV, HTRA, HYDROLASE, PROTEASE
5e55:A (ILE630) to (LYS688) CRYSTAL STRUCTURE OF MOUSE CNTN6 FN1-FN3 DOMAINS | NEURAL CELL ADHESION MOLECULE, FIBRONECTIN TYPE III DOMAINS, CELL ADHESION
3arr:A (THR77) to (SER124) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH PENTOXIFYLLINE | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3arp:A (THR77) to (ALA125) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH DEQUALINIUM | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3ars:A (THR77) to (ALA125) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - APO STRUCTURE OF MUTANT W275G | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE
3arw:A (THR77) to (ALA125) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH CHELERYTHRINE | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1zyo:A (LEU152) to (ASP203) CRYSTAL STRUCTURE OF THE SERINE PROTEASE DOMAIN OF SESBANIA MOSAIC VIRUS POLYPROTEIN | VIRAL SERINE PROTEASE OF TRYPSIN FOLD, BETA-BARREL, GLUTAMYL ENDOPEPTIDASE, HYDROLASE
3ary:A (THR77) to (SER124) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH 2-(IMIDAZOLIN-2-YL)-5- ISOTHIOCYANATOBENZOFURAN | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3arz:A (THR77) to (SER124) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH 2-(IMIDAZOLIN-2-YL)-5- ISOTHIOCYANATOBENZOFURAN | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3lvt:A (GLU682) to (GLU730) THE CRYSTAL STRUCTURE OF A PROTEIN IN THE GLYCOSYL HYDROLASE FAMILY 38 FROM ENTEROCOCCUS FAECALIS TO 2.55A | GLYCOSYL, HYDROLASE, PSI, MCSG, STRUCTURAL GENOMICS, MIDWEST CENTER FOR STRUCTURAL GENOMICS, PROTEIN STRUCTURE INITIATIVE
4ayy:B (GLN15) to (MET80) HUMAN THROMBIN - INHIBITOR COMPLEX | HYDROLASE-INHIBITOR COMPLEX
2a0q:D (GLN30) to (MET84) STRUCTURE OF THROMBIN IN 400 MM POTASSIUM CHLORIDE | SERINE PROTEASE, HYDROLASE
2a2x:H (GLN30) to (MET84) ORALLY ACTIVE THROMBIN INHIBITORS IN COMPLEX WITH THROMBIN INH12 | BLOOD CLOTTING, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2a31:A (GLN30) to (ASN84) TRYPSIN IN COMPLEX WITH BORATE | HYDROLASE, TRYPSIN
2a32:A (GLN30) to (ASN84) TRYPSIN IN COMPLEX WITH BENZENE BORONIC ACID | HYDROLASE
5ec5:E (LYS21) to (MET130) CRYSTAL STRUCTURE OF LYSENIN PORE | INVERTEBRATE CYTOLYSIN, NONAMER, FUNCTIONAL PORE, NANOPORE, TOXIN
5ec5:G (LYS21) to (MET130) CRYSTAL STRUCTURE OF LYSENIN PORE | INVERTEBRATE CYTOLYSIN, NONAMER, FUNCTIONAL PORE, NANOPORE, TOXIN
5ec5:R (LYS21) to (MET130) CRYSTAL STRUCTURE OF LYSENIN PORE | INVERTEBRATE CYTOLYSIN, NONAMER, FUNCTIONAL PORE, NANOPORE, TOXIN
3m6o:A (LYS78) to (ARG125) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA PEPTIDE DEFORMYLASE 1B (ATPDF1B) | PEPTIDE DEFORMYLASE, 1B, PDF, N-TERMINAL EXCISION PATHWAY, NME, ARABIDOPSIS THALIANA, INDUCED-FIT, HYDROLASE, METAL-BINDING, MITOCHONDRION, PROTEIN BIOSYNTHESIS, TRANSIT PEPTIDE
5eg4:A (GLN30) to (SER84) BOVINE TRYPSIN IN COMPLEX WITH CYCLIC INHIBITOR | METAL-BINDING, DIGESTION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, HYDROLASE
3m9d:J (PRO98) to (PHE155) CRYSTAL STRUCTURE OF THE PROKARYOTIC UBIQUINTIN-LIKE PROTEIN PUP COMPLEXED WITH THE HEXAMERIC PROTEASOMAL ATPASE MPA WHICH INCLUDES THE AMINO TERMINAL COILED COIL DOMAIN AND THE INTER DOMAIN | ALPHA HELIX COIL COIL, 5 BETA-STRAND BARREL, ATP-BINDING, CHAPERONE, NUCLEOTIDE-BINDING, PROTEASOME, S-NITROSYLATION, VIRULENCE, ISOPEPTIDE BOND, UBL CONJUGATION PATHWAY
4b9i:A (GLY60) to (VAL146) STRUCTURE OF CSSA SUBUNIT COMPLEMENTED WITH DONOR STRAND FROM CSSB SUBUNIT OF ENTEROTOXIGENIC ESCHERICHIA COLI COLONIZATION FACTOR CS6 | CELL ADHESION, DIARRHEAL DISEASE, FIMBRIAE, FUSION PROTEIN
4b9j:A (GLY60) to (SER174) STRUCTURE OF SELF-COMPLEMENTED CSSA SUBUNIT OF ENTEROTOXIGENIC ESCHERICHIA COLI COLONIZATION FACTOR CS6 | CELL ADHESION, DIARRHEAL DISEASE, FIMBRIAE, FUSION PROTEIN
5ejb:D (VAL390) to (SER428) CRYSTAL STRUCTURE OF PREFUSION HENDRA VIRUS F PROTEIN | PREFUSION FORM, VIRAL GLYCOPROTEIN, ECTODOMAIN, VIRAL PROTEIN
3b8s:A (THR77) to (ALA125) CRYSTAL STRUCTURE OF WILD-TYPE CHITINASE A FROM VIBRIO HARVEYI | TIM-BARREL, GLYCOSIDASE, HYDROLASE
3b8s:B (THR77) to (ALA125) CRYSTAL STRUCTURE OF WILD-TYPE CHITINASE A FROM VIBRIO HARVEYI | TIM-BARREL, GLYCOSIDASE, HYDROLASE
3b9a:A (THR77) to (SER124) CRYSTAL STRUCTURE OF VIBRIO HARVEYI CHITINASE A COMPLEXED WITH HEXASACCHARIDE | TIM-BARREL, HEXASACCHARIDE COMPLEX, GLYCOSIDASE, HYDROLASE
3bcu:A (LEU198) to (THR240) GLUCOGEN PHOSPHORYLASE COMPLEX WITH THYMIDINE | GLYCOGENOLYSIS, TYPE 2 DIABETES, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHORYLATION, PYRIDOXAL PHOSPHATE, TRANSFERASE
5est:E (GLN30) to (GLY84) CRYSTALLOGRAPHIC ANALYSIS OF THE INHIBITION OF PORCINE PANCREATIC ELASTASE BY A PEPTIDYL BORONIC ACID: STRUCTURE OF A REACTION INTERMEDIATE | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4qt8:B (GLN608) to (ARG677) CRYSTAL STRUCTURE OF RON SEMA-PSI-IPT1 EXTRACELLULAR DOMAINS IN COMPLEX WITH MSP BETA-CHAIN | GROWTH FACTOR RECEPTOR/GROWTH FACTOR, RECEPTOR-LIGAND COMPLEX, RON RECEPTOR TYROSINE KINASE, MACROPHAGE STIMULATING PROTEIN, HYDROLASE- SIGNALING PROTEIN COMPLEX
4qt8:C (THR495) to (PRO556) CRYSTAL STRUCTURE OF RON SEMA-PSI-IPT1 EXTRACELLULAR DOMAINS IN COMPLEX WITH MSP BETA-CHAIN | GROWTH FACTOR RECEPTOR/GROWTH FACTOR, RECEPTOR-LIGAND COMPLEX, RON RECEPTOR TYROSINE KINASE, MACROPHAGE STIMULATING PROTEIN, HYDROLASE- SIGNALING PROTEIN COMPLEX
4qt8:D (THR495) to (PRO556) CRYSTAL STRUCTURE OF RON SEMA-PSI-IPT1 EXTRACELLULAR DOMAINS IN COMPLEX WITH MSP BETA-CHAIN | GROWTH FACTOR RECEPTOR/GROWTH FACTOR, RECEPTOR-LIGAND COMPLEX, RON RECEPTOR TYROSINE KINASE, MACROPHAGE STIMULATING PROTEIN, HYDROLASE- SIGNALING PROTEIN COMPLEX
3ms4:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE COMPLEXED WITH 4-TRIFLUOROMETHYLBENZALDEHYDE-4- (BETA-D-GLUCOPYRANOSYL)-THIOSEMICARBAZONE | GLYCOGENOLYSIS, TYPE 2 DIABETES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mt9:A (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE COMPLEXED WITH 4-NITROBENZALDEHYDE-4-(BETA-D- GLUCOPYRANOSYL)-THIOSEMICARBAZONE | GLYCOGENOLYSIS, TYPE 2 DIABETES, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3muj:A (LEU283) to (CYS327) EARLY B-CELL FACTOR 3 (EBF3) IPT/TIG AND DIMERIZATION HELICES | IMMUNOGLOBULIN LIKE FOLD, HELIX-LOOP-HELIX, STRUCTURAL GENOMICS CONSORTIUM, SGC, DNA BINDING PROTEIN
3bn9:B (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MT-SP1 IN COMPLEX WITH FAB INHIBITOR E2 | ANTIBODY-PROTEASE COMPLEX, PROTEIN-PROTEIN COMPLEX, ENZYME- INHIBITOR COMPLEX, DISEASE MUTATION, GLYCOPROTEIN, HYDROLASE, MEMBRANE, POLYMORPHISM, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
3bn9:A (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MT-SP1 IN COMPLEX WITH FAB INHIBITOR E2 | ANTIBODY-PROTEASE COMPLEX, PROTEIN-PROTEIN COMPLEX, ENZYME- INHIBITOR COMPLEX, DISEASE MUTATION, GLYCOPROTEIN, HYDROLASE, MEMBRANE, POLYMORPHISM, SERINE PROTEASE, SIGNAL- ANCHOR, TRANSMEMBRANE
4boh:H (GLN335) to (MET400) MADANINS (MEROPS I53) ARE CLEAVED BY THROMBIN AND FACTOR XA | HYDROLASE-INHIBITOR COMPLEX, COAGULATION INHIBITOR, PROTEASE, MACROMOLECULAR RECOGNITION
4bom:A (GLY205) to (THR249) STRUCTURE OF HERPESVIRUS FUSION GLYCOPROTEIN B-BILAYER COMPLEX REVEALING THE PROTEIN-MEMBRANE AND LATERAL PROTEIN-PROTEIN INTERACTION | VIRAL PROTEIN, MEMBRANE PROXIMAL REGION, PROTEIN COAT, PSEUDO-ATOMIC VIRUS-HOST INTERACTION
3bsq:A (GLN30) to (SER82) CRYSTAL STRUCTURE OF HUMAN KALLIKREIN 7 PRODUCED AS A SECRETION PROTEIN IN E.COLI | SERINE PROTEASES, KALLIKREINS, LD6, X-RAY CRYSTAL STRUCTURE, GLYCOPROTEIN, HYDROLASE, SECRETED, ZYMOGEN
4btt:B (GLN30) to (GLU84) FACTOR XA IN COMPLEX WITH THE DUAL THROMBIN-FXA INHIBITOR 31. | HYDROLASE, SAR107375, FACTOR XA INHIBITOR, THROMBIN INHIBITOR, CHLOROTHIOPHENE P1 FRAGMENT, S3 SUBSITE, MICROSOMES STABILITY, ORAL ANTITHROMBOTIC, DUAL INHIBITOR, IV ANTITHROMBOTIC
4btu:B (GLN30) to (GLU84) FACTOR XA IN COMPLEX WITH THE DUAL THROMBIN-FXA INHIBITOR 57. | HYDROLASE, SAR107375, FACTOR XA INHIBITOR, THROMBIN INHIBITOR, CHLOROTHIOPHENE P1 FRAGMENT, S3 SUBSITE, MICROSOMES STABILITY, ORAL ANTITHROMBOTIC, DUAL INHIBITOR, IV ANTITHROMBOTIC
4r0i:A (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MATRIPTASE IN COMPLEX WITH INHIBITOR | HYDROLASE, MATRIPTASE, COMPLEX STRUCTURE, TRYPSIN-LIKE SERINE PROTEINASE FOLD, PROTEASE, SMALL MOLECULE INHIBITOR
5fah:A (GLN30) to (LYS84) KALLIKREIN-7 IN COMPLEX WITH COMPOUND1 | HYDROLASE
3c1k:A (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH INHIBITOR 15 | THROMBIN, THROMBIN INHIBITOR COMPLEX, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, SULFATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5fcr:A (MET30) to (ASP84) MOUSE COMPLEMENT FACTOR D | HYDROLASE
3c2u:B (MET196) to (HIS263) STRUCTURE OF THE TWO SUBSITE D-XYLOSIDASE FROM SELENOMONAS RUMINANTIUM IN COMPLEX WITH 1,3-BIS[TRIS(HYDROXYMETHYL) METHYLAMINO]PROPANE | TETRAMER; GLYCOSIDE HYDROLASE; GH43; ALPHA-L- ARABINOFURANOSIDASE
4r5l:C (LEU397) to (ASP460) CRYSTAL STRUCTURE OF THE DNAK C-TERMINUS (DNAK-SBD-C) | HELICAL BUNDLE, BETA SHEETS, CHAPERONE, MEMBRANE
3c5m:A (TYR254) to (ASP303) CRYSTAL STRUCTURE OF OLIGOGALACTURONATE LYASE (VPA0088) FROM VIBRIO PARAHAEMOLYTICUS. NORTHEAST STRUCTURAL GENOMICS CONSORTIUM TARGET VPR199 | 7 BLADE-SHAPED BETA-PROPELLER, STRUCTURAL GENOMICS, PSI-2, PROTEIN STRUCTURE INITIATIVE, NORTHEAST STRUCTURAL GENOMICS CONSORTIUM, NESG, LYASE
3nbn:A (GLN84) to (LYS145) CRYSTAL STRUCTURE OF A DIMER OF NOTCH TRANSCRIPTION COMPLEX TRIMERS ON HES1 DNA | PROMOTER REGIONS, NOTCH1, CSL, RBPJ, MASTERMIND, TRANSCRIPTION FACTORS, TRANSCRIPTION, TRANSCRIPTIONAL ACTIVATION, TRANSCRIPTION- DNA COMPLEX
3nbn:D (GLN84) to (LYS145) CRYSTAL STRUCTURE OF A DIMER OF NOTCH TRANSCRIPTION COMPLEX TRIMERS ON HES1 DNA | PROMOTER REGIONS, NOTCH1, CSL, RBPJ, MASTERMIND, TRANSCRIPTION FACTORS, TRANSCRIPTION, TRANSCRIPTIONAL ACTIVATION, TRANSCRIPTION- DNA COMPLEX
4c91:A (TYR692) to (VAL748) EVIDENCE THAT GH115 ALPHA-GLUCURONIDASE ACTIVITY IS DEPENDENT ON CONFORMATIONAL FLEXIBILITY | HYDROLASE, XYLOSE, GLUCURONIC ACID
4c91:B (TYR692) to (VAL748) EVIDENCE THAT GH115 ALPHA-GLUCURONIDASE ACTIVITY IS DEPENDENT ON CONFORMATIONAL FLEXIBILITY | HYDROLASE, XYLOSE, GLUCURONIC ACID
3nps:A (GLN30) to (ARG84) CRYSTAL STRUCTURE OF MEMBRANE-TYPE SERINE PROTEASE 1 (MT-SP1) IN COMPLEX WITH THE FAB INHIBITOR S4 | HYDROLASE, ANTIBODY-PROTEASE COMPLEX, PROTEIN-PROTEIN COMPLEX, ENZYME-INHIBITOR COMPLEX, DISEASE MUTATION, GLYCOPROTEIN, MEMBRANE, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE, HYDROLASE - IMMUNE SYSTEM COMPLEX, HYDROLASE-IMMUNE SYSTEM COMPLEX
4rn6:A (GLN30) to (MET84) STRUCTURE OF PRETHROMBIN-2 MUTANT S195A BOUND TO THE ACTIVE SITE INHIBITOR ARGATROBAN | SERINE PROTEASE, PRETHROMBIN-2, AUTOACTIVATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3cuv:A (LEU198) to (THR240) TRACKING STRUCTURE ACTIVITY RELATIONSHIPS OF GLYCOGEN PHOSPHORYLASE INHIBITORS: SYNTHESIS, KINETIC AND CRYSTALLOGRAPHIC EVALUATION OF ANALOGUES OF N-(-D- GLUCOPYRANOSYL)-N'-OXAMIDES | GLYCOGEN PHOSPHORYLASE, STRUCTURE, CATALYTIC SITE, RATIONAL INHIBITOR DESIGN, ACETYLATION, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
3d12:A (GLN450) to (GLY523) CRYSTAL STRUCTURES OF NIPAH VIRUS G ATTACHMENT GLYCOPROTEIN IN COMPLEX WITH ITS RECEPTOR EPHRIN-B3 | BETA PROPELLER, PROTEIN-RECEPTOR COMPLEX, ENVELOPE PROTEIN, GLYCOPROTEIN, HEMAGGLUTININ, HYDROLASE, MEMBRANE, SIGNAL-ANCHOR, TRANSMEMBRANE, VIRION, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, NEUROGENESIS, HYDROLASE-MEMBRANE PROTEIN COMPLEX
4ctn:A (LEU198) to (THR240) GLUCOPYRANOSYLIDENE-SPIRO-IMINOTHIAZOLIDINONE, A NEW BICYCLIC RING SYSTEM: SYNTHESIS, DERIVATIZATION, AND EVALUATION AS GLYCOGEN PHOSPHORYLASE INHIBITORS BY ENZYME KINETIC AND CRYSTALLOGRAPHIC METHODS | TRANSFERASE, TYPE 2 DIABETES, INHIBITOR, STRUCTURE-BASED DRUG DESIGN
3da9:B (GLN51) to (MET116) CRYSTAL STRUCTURE OF THROMBIN IN COMPLEX WITH INHIBITOR | THROMBIN, INHIBITOR COMPLEX, ACUTE PHASE, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PHARMACEUTICAL, POLYMORPHISM, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN
5gch:F (GLN30) to (LYS84) CHEMISTRY OF CAGED ENZYMES /II$. PHOTOACTIVATION OF INHIBITED CHYMOTRYPSIN | HYDROLASE (SERINE PROTEINASE)
3ooc:A (GLN263) to (PRO328) CRYSTAL STRUCTURE OF THE MEMBRANE FUSION PROTEIN CUSB FROM ESCHERICHIA COLI | THREE-HELIX BUNDLE, BETA BARREL, COPPER TRANSPORT, ION TRANSPORT, TRANSPORT, TRANSPORT PROTEIN, CUSA,CUSC
5gxp:A (GLN30) to (SER84) CATIONIC TRYPSIN WITH GOL/PGE AS DIMER AT PH 4.6 | CATIONIC TRYPSIN, GOL, PGE, HYDROLASE
4d8n:A (GLN30) to (SER84) HUMAN KALLIKREIN 6 INHIBITORS WITH A PARA-AMIDOBENZYLANMINE P1 GROUP CARRY A HIGH BINDING EFFICIENCY | HUMAN KALLIKREIN 6, HK6, SERINE PROTEASE, PROTEIN-LIGAND COMPLEX, AMIDINOTHIOPHENE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3dt0:H (GLN30) to (MET84) UNDERSTANDING THROMBIN INHIBITION | BLOOD CLOTTING, HYDROLASE INHIBITOR, ACUTE PHASE, BLOOD COAGULATION, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4u30:C (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH BIKUNIN KUNITZ DOMAIN 2 | SERINE PROTEASE, PROTEASE INHIBITOR, PROTEIN-PROTEIN INTERACTION, PROTEIN DEGRADATION, PROTEOLYSIS, SUBSTRATE SPECIFICITY, ENZYME KINETICS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4u32:A (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH HAI-2 KUNITZ DOMAIN 1 | SERINE PROTEASE, PROTEASE INHIBITOR, PROTEIN-PROTEIN INTERACTION, PROTEIN DEGRADATION, PROTEOLYSIS, SUBSTRATE SPECIFICITY, ENZYME KINETICS, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3owr:C (THR40) to (PRO120) CRYSTAL STRUCTURE OF A PUTATIVE SECRETED PROTEIN (BF4250) FROM BACTEROIDES FRAGILIS NCTC 9343 AT 1.81 A RESOLUTION | CARBOHYDRATE METABOLISM, PUTATIVE GLYCOSIDE HYDROLASE, IG-LIKE, STRUCTURAL GENOMICS, JOINT CENTER FOR STRUCTURAL GENOMICS, JCSG, PROTEIN STRUCTURE INITIATIVE, PSI-BIOLOGY, UNKNOWN FUNCTION
4dii:H (GLN30) to (MET84) X-RAY STRUCTURE OF THE COMPLEX BETWEEN HUMAN ALPHA THROMBIN AND THROMBIN BINDING APTAMER IN THE PRESENCE OF POTASSIUM IONS | PROTEIN-DNA COMPLEX, SERINE PROTEASE, BLOOD COAGULATION, APTAMER, HYDROLASE-HYDROLASE INHIBITOR-DNA COMPLEX, SERINE PROTEASE FOLD, DNA APTAMER, BLOOD, G-QUADRUPLEX
4u5z:A (MET151) to (VAL249) TRICHODYSPLASIA SPINULOSA-ASSOCIATED POLYOMAVIRUS (TSPYV) VP1 | VIRAL COAT PROTEIN, JELLY-ROLL FOLD, GLYCAN BINDING, VIRAL PROTEIN
4u5z:G (GLY150) to (LEU250) TRICHODYSPLASIA SPINULOSA-ASSOCIATED POLYOMAVIRUS (TSPYV) VP1 | VIRAL COAT PROTEIN, JELLY-ROLL FOLD, GLYCAN BINDING, VIRAL PROTEIN
4u61:A (GLY150) to (VAL249) TRICHODYSPLASIA SPINULOSA-ASSOCIATED POLYOMAVIRUS (TSPYV) VP1 IN COMPLEX WITH 6'-SIALYLLACTOSE | VIRAL COAT PROTEIN, JELLY-ROLL FOLD, GLYCAN BINDING, VIRAL PROTEIN
3e0p:B (GLN30) to (THR84) THE X-RAY STRUCTURE OF HUMAN PROSTASIN IN COMPLEX WITH A COVALENT BENZOXAZOLE INHIBITOR | PROSTASIN, PROTEASE, BENZOXAZOLE, WARHEAD, CHANNEL, ENAC, CELL MEMBRANE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, SECRETED, SERINE PROTEASE, TRANSMEMBRANE, ZYMOGEN
3p6z:B (GLN378) to (MET443) STRUCTURAL BASIS OF THROMBIN MEDIATED FACTOR V ACTIVATION: ESSENTIAL ROLE OF THE HIRUDIN-LIKE SEQUENCE GLU666-GLU672 FOR PROCESSING AT THE HEAVY CHAIN-B DOMAIN JUNCTION | TRYPSIN-LIKE SERINE PROTEINASE, BLOOD COAGULATION, N-GLYCOSYLATION, BLOOD PLASMA, PPACK, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3e1f:3 (LEU651) to (ARG721) E.COLI (LACZ) BETA-GALACTOSIDASE (H418E) IN COMPLEX WITH GALACTOSE | HIS-418-GLU BETA-GALACTOSIDASE HYDROLASE TIM BARREL (ALPHA/BETA BARREL) JELLY-ROLL BARREL IMMUNOGLOBULIN BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
3e1f:4 (LEU651) to (ARG721) E.COLI (LACZ) BETA-GALACTOSIDASE (H418E) IN COMPLEX WITH GALACTOSE | HIS-418-GLU BETA-GALACTOSIDASE HYDROLASE TIM BARREL (ALPHA/BETA BARREL) JELLY-ROLL BARREL IMMUNOGLOBULIN BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
5hoo:A (LYS158) to (LYS209) CRYSTAL STRUCTURE OF THE MOS1 STRAND TRANSFER COMPLEX | PROTEIN-DNA COMPLEX, DNA TRANSPOSASE, RECOMBINASE, INTEGRASE, HELIX- TURN-HELIX, BASE FLIPPING, DNA
3e3l:C (LEU198) to (THR240) THE R-STATE GLYCOGEN PHOSPHORYLASE | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
3pa1:A (GLY332) to (PHE434) CRYSTAL STRUCTURE OF P DOMAIN FROM NORWALK VIRUS STRAIN VIETNAM 026 IN COMPLEX WITH HBGA TYPE A | NOROVIRUS, P-DOMAIN, CAPSID, RECEPTOR, HISTO BLOOD GROUP ANTIGEN (HBGA), VIRAL PROTEIN
3e3o:C (LEU198) to (THR240) GLYCOGEN PHOSPHORYLASE R STATE-IMP COMPLEX | GLYCOGENOLYSIS, INHIBITION, TYPE 2 DIABETES, ALLOSTERIC ENZYME, CARBOHYDRATE METABOLISM, GLYCOGEN METABOLISM, GLYCOSYLTRANSFERASE, NUCLEOTIDE-BINDING, PHOSPHOPROTEIN, PYRIDOXAL PHOSPHATE, TRANSFERASE
4dt7:D (GLN30) to (MET84) CRYSTAL STRUCTURE OF THROMBIN BOUND TO THE ACTIVATION DOMAIN QEDQVDPRLIDGKMTRRGDS OF PROTEIN C | SERINE PROTEASE, HYDROLASE
5hza:B (GLY332) to (PHE434) CRYSTAL STRUCTURE OF GII.10 P DOMAIN IN COMPLEX WITH 3-FUCOSYLLACTOSE (3 FL) | NOROVIRUS, P DOMAIN, HMO, 3-FUCOSYLLACTOSE, HUMAN MILK, VIRUS, VIRAL PROTEIN
5hzb:B (GLY332) to (PHE434) CRYSTAL STRUCTURE OF GII.10 P DOMAIN IN COMPLEX WITH 2-FUCOSYLLACTOSE (2'FL) | NOROVIRUS CAPSID, P DOMAIN, HMO, HUMAN MILK, 2-FUCOSYLLACTOSE, VIRUS, VIRAL PROTEIN
4uff:H (GLN30) to (MET84) THROMBIN IN COMPLEX WITH (2R)-2-(BENZYLSULFONYLAMINO)-N-(2-( (4-CARBAMIMIDOYLPHENYL)METHYLAMINO)-2-OXO-ETHYL)-N-METHYL- 3-PHENYL-PROPANAMIDE | HYDROLASE, HYDROLASE INHIBITOR COMPLEX, SERINE PROTEASE, BLOOD COAGULATION, BLOOD CLOTTING, CONVERTION OF FIBRINOGEN TO FIBRIN, BLOOD CLOTTING INHIBITOR, THROMBIN INHIBITOR, PREORGANIZATION, GLYCOSYLATION, BLOOD
4ufg:H (GLN30) to (MET84) THROMBIN IN COMPLEX WITH (2R)-2-(BENZYLSULFONYLAMINO)-N-(( 1S)-2-((4-CARBAMIMIDOYLPHENYL)METHYLAMINO)-1-METHYL-2-OXO- ETHYL)-N-METHYL-3-PHENYL-PROPANAMIDE ETHANE | HYDROLASE, HYDROLASE INHIBITOR COMPLEX, SERINE PROTEASE, BLOOD COAGULATION, BLOOD CLOTTING, CONVERTION OF FIBRINOGEN TO FIBRIN, BLOOD CLOTTING INHIBITOR, THROMBIN INHIBITOR, PREORGANIZATION, GLYCOSYLATION, BLOOD
4dur:A (GLN576) to (GLU634) THE X-RAY CRYSTAL STRUCTURE OF FULL-LENGTH TYPE II HUMAN PLASMINOGEN | SERINE PROTEASE, FIBRINOLYSIS, HYDROLASE
5i46:H (GLN30) to (ARG84) FACTOR VIIA IN COMPLEX WITH THE INHIBITOR (2R,15R)-2-[(1- AMINOISOQUINOLIN-6-YL)AMINO]-8-FLUORO-7-HYDROXY-4,15,17-TRIMETHYL-13- OXA-4,11-DIAZATRICYCLO[14.2.2.1~6,10~]HENICOSA-1(18),6(21),7,9,16,19- HEXAENE-3,12-DIONE | GLYCOPROTEIN, HYDROLASE, SERINE PROTEASE, PLASMA, BLOOD COAGULATION FACTOR, PROTEIN INHIBITOR COMPLEX, CALCIUM-BINDING, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3pj5:B (LEU138) to (ALA219) CRYSTAL STRUCTURE OF FAR-RED FLUORESCENT PROTEIN KATUSHKA CRYSTALLIZED AT PH 5.0 | KATUSHKA, FAR-RED FLUORESCENT PROTEIN, BETA-BARREL, BIOMARKER, MUTANT VARIANT OF EQFP578, MET-TYR-GLY CHROMOPHORE, FLUORESCENT PROTEIN
3pjb:A (LEU138) to (ALA219) CRYSTAL STRUCTURE OF RED FLUORESCENT PROTEIN EQFP578 CRYSTALLIZED AT PH 4.0 | EQFP578, RED FLUORESCENT PROTEIN, BETA-BARREL, BIOMARKER, MET-TYR-GLY CHROMOPHORE, FLUORESCENT PROTEIN
3pjb:B (LEU138) to (ALA219) CRYSTAL STRUCTURE OF RED FLUORESCENT PROTEIN EQFP578 CRYSTALLIZED AT PH 4.0 | EQFP578, RED FLUORESCENT PROTEIN, BETA-BARREL, BIOMARKER, MET-TYR-GLY CHROMOPHORE, FLUORESCENT PROTEIN
3pma:B (GLN30) to (SER83) 2.2 ANGSTROM CRYSTAL STRUCTURE OF THE COMPLEX BETWEEN BOVINE THROMBIN AND SUCROSE OCTASULFATE | PROTEASE, THROMBOSIS, FIBRINOLYSIS, AGONIST, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4e7n:A (LEU30) to (VAL84) CRYSTAL STRUCTURE OF AHV_TL-I, A GLYCOSYLATED SNAKE-VENOM THROMBIN- LIKE ENZYME FROM AGKISTRODON HALYS | BETA-BARREL, HYDROLASE, ARGININE ESTERASE, GLYCOSYLATION, EXTRACELLULAR
4e7r:H (GLN30) to (MET84) THROMBIN IN COMPLEX WITH 3-AMIDINOPHENYLALANINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEASE, KRINGLE, HYDROLASE, BLOOD COAGULATION, BLOOD CLOTTING, CONVERTION OF FIBRINOGEN TO FIBRIN, BLOOD CLOTTING INHIBITOR, THROMBIN INHIBITOR, GLYCOSYLATION, BLOOD
4e7r:G (GLN1030) to (MET1084) THROMBIN IN COMPLEX WITH 3-AMIDINOPHENYLALANINE INHIBITOR | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEASE, KRINGLE, HYDROLASE, BLOOD COAGULATION, BLOOD CLOTTING, CONVERTION OF FIBRINOGEN TO FIBRIN, BLOOD CLOTTING INHIBITOR, THROMBIN INHIBITOR, GLYCOSYLATION, BLOOD
4edo:A (LEU138) to (ALA219) CRYSTAL STRUCTURE OF FAR-RED FLUORESCENT PROTEIN EQFP650 | BETA BARREL, FLUORESCENT PROTEIN
4eds:A (LEU138) to (ALA219) CRYSTAL STRUCTURE OF FAR-RED FLUORESCENT PROTEIN EQFP670 | BETA BARREL, FLUORESCENT PROTEIN
4eke:A (LEU198) to (THR240) CRYSTAL STRUCTURE OF GPB IN COMPLEX WITH DK11 | ALPHA/BETA PROTEIN, TRANSFERASE
4eky:A (LEU198) to (THR240) CRYSTAL STRUCTURE OF GPB IN COMPLEX WITH DK15 | ALPHA/BETA PROTEIN, TRANSFERASE
3q39:A (GLY332) to (PHE434) CRYSTAL STRUCTURE OF P DOMAIN FROM NORWALK VIRUS STRAIN VIETNAM 026 IN COMPLEX WITH HBGA TYPE H2 (DIGLYCAN) | NOROVIRUS, P-DOMAIN, CAPSID, RECEPTOR, HISTO BLOOD GROUP ANTIGEN (HBGA), VIRAL PROTEIN
3q6r:A (GLY332) to (PHE434) CRYSTAL STRUCTURE OF P DOMAIN FROM NORWALK VIRUS STRAIN VIETNAM 026 IN COMPLEX WITH DISORDERED HBGA TYPE LEX | NOROVIRUS, P-DOMAIN, CAPSID, RECEPTOR, HISTO BLOOD GROUP ANTIGEN (HBGA), VIRAL PROTEIN
4est:E (GLN30) to (GLY84) CRYSTAL STRUCTURE OF THE COVALENT COMPLEX FORMED BY A PEPTIDYL ALPHA, ALPHA-DIFLUORO-BETA-KETO AMIDE WITH PORCINE PANCREATIC ELASTASE AT 1.78-ANGSTROMS RESOLUTION | SERINE PROTEINASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3qum:P (GLN30) to (GLN84) CRYSTAL STRUCTURE OF HUMAN PROSTATE SPECIFIC ANTIGEN (PSA) IN FAB SANDWICH WITH A HIGH AFFINITY AND A PCA SELECTIVE ANTIBODY | KALLIKREIN FOLD, PROSTATE-SPECIFIC ANTIGEN, SERINE PROTEASE, NEGATIVE REGULATION OF ANGIOGENESIS, NATURAL POST-TRANSDUCTIONAL MODIFICATION, N-LINKED AND O-LINKED GLYCOSYLATION, IMMUNE SYSTEM
3qum:Q (GLN30) to (GLN84) CRYSTAL STRUCTURE OF HUMAN PROSTATE SPECIFIC ANTIGEN (PSA) IN FAB SANDWICH WITH A HIGH AFFINITY AND A PCA SELECTIVE ANTIBODY | KALLIKREIN FOLD, PROSTATE-SPECIFIC ANTIGEN, SERINE PROTEASE, NEGATIVE REGULATION OF ANGIOGENESIS, NATURAL POST-TRANSDUCTIONAL MODIFICATION, N-LINKED AND O-LINKED GLYCOSYLATION, IMMUNE SYSTEM
5jb8:S (GLN30) to (ASN84) CRYSTAL STRUCTURE OF FACTOR IXA VARIANT K98T IN COMPLEX WITH EGR- CHLOROMETHYLKETONE | BLOOD CLOTTING, HYDROLASE, GLYCOPROTEIN, HAEMOSTASIS
5jba:S (GLN30) to (ASN84) CRYSTAL STRUCTURE OF FACTOR IXA VARIANT V16I K98T Y177T I212V IN COMPLEX WITH PPACK | BLOOD CLOTTING, HYDROLASE, GLYCOPROTEIN, HAEMOSTASIS
5jbb:S (VAL31) to (ASN84) CRYSTAL STRUCTURE OF FACTOR IXA VARIANT V16I K98T Y177T I213V IN COMPLEX WITH EGR-CHLOROMETHYLKETONE | BLOOD CLOTTING, HYDROLASE, GLYCOPROTEIN, HAEMOSTASIS
5jbc:S (GLN30) to (ASN84) CRYSTAL STRUCTURE OF FACTOR IXA VARIANT V16I K98T Y177T I213V IN COMPLEX WITH PPACK | CRYSTAL STRUCTURE OF FACTOR IXA VARIANT K98T IN COMPLEX WITH EGR- CHLOROMETHYLKETONE, HYDROLASE
5jbt:A (GLN30) to (ASN84) MESOTRYPSIN IN COMPLEX WITH CLEAVED AMYLOID PRECURSOR LIKE PROTEIN 2 INHIBITOR (APLP2) | INHIBITOR PROTEASE SERINE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3rgb:I (LYS120) to (ASP179) CRYSTAL STRUCTURE OF PARTICULATE METHANE MONOOXYGENASE FROM METHYLOCOCCUS CAPSULATUS (BATH) | MEMBRANE, OXIDOREDUCTASE
4fs9:B (ALA289) to (ASN337) COMPLEX STRUCTURE OF A BROAD SPECIFICITY AMINO ACID RACEMASE (BAR) WITHIN THE REACTIVE INTERMEDIATE | ISOMERASE, PLP BINDING, RACEMIZATION
4gaw:H (MET30) to (PRO85) CRYSTAL STRUCTURE OF ACTIVE HUMAN GRANZYME H | SERINE PROTEASE, CYTOLYSIS, HYDROLASE, CYTOTOXIC GRANULES
4gaw:J (TYR29) to (PRO85) CRYSTAL STRUCTURE OF ACTIVE HUMAN GRANZYME H | SERINE PROTEASE, CYTOLYSIS, HYDROLASE, CYTOTOXIC GRANULES
4gch:F (GLN30) to (LYS84) STRUCTURE AND ACTIVITY OF TWO PHOTOREVERSIBLE CINNAMATES BOUND TO CHYMOTRYPSIN | HYDROLASE (SERINE PROTEINASE)
5l56:A (ASN1185) to (SER1227) PLEXIN A1 FULL EXTRACELLULAR REGION, DOMAINS 1 TO 10, TO 4 ANGSTROM | RECEPTOR, SIGNALING, AXON GUIDANCE, SIGNALING PROTEIN
5l59:A (ASN1185) to (SER1227) PLEXIN A1 FULL EXTRACELLULAR REGION, DOMAINS 1 TO 10, TO 6 ANGSTROM, SPACEGROUP P2(1) | RECEPTOR, SIGNALING, AXON GUIDANCE, SIGNALING PROTEIN
5l59:B (ASN1185) to (SER1227) PLEXIN A1 FULL EXTRACELLULAR REGION, DOMAINS 1 TO 10, TO 6 ANGSTROM, SPACEGROUP P2(1) | RECEPTOR, SIGNALING, AXON GUIDANCE, SIGNALING PROTEIN
5l5c:A (ASN1185) to (SER1227) PLEXIN A1 FULL EXTRACELLULAR REGION, DOMAINS 1 TO 10, TO 6 ANGSTROM, SPACEGROUP P4(3)2(1)2 | RECEPTOR, SIGNALING, AXON GUIDANCE, SIGNALING PROTEIN
5la2:B (TYR390) to (ILE452) THE MECHANISM BY WHICH ARABINOXYLANASES CAN RECOGNISE HIGHLY DECORATED XYLANS | ARABINOXYLANASE, GLYCOSIDE HYDROLASE, CARBOHYDRATE BINDING MODULE, ARABINOSE, CLOSTRIDIUM THERMOCELLUM, CELLULOSOME, HYDROLASE
5lpe:B (GLN30) to (ARG84) KALLIKREIN-RELATED PEPTIDASE 10 COMPLEX WITH ZN2+ | SERINE PROTEASE, ZYMOGEN-LIKE ENZYME, ZN2+ INHIBITION, TUMOR SUPPRESSOR, HYDROLASE
5lpf:A (GLN30) to (ARG84) KALLIKREIN-RELATED PEPTIDASE 10 | SERINE PROTEASE, ZYMOGEN-LIKE ENZYME, ZN2+ INHIBITION, TUMOR SUPPRESSOR, HYDROLASE
5lpf:B (GLN30) to (ARG84) KALLIKREIN-RELATED PEPTIDASE 10 | SERINE PROTEASE, ZYMOGEN-LIKE ENZYME, ZN2+ INHIBITION, TUMOR SUPPRESSOR, HYDROLASE
6cha:B (GLN30) to (LYS84) STRUCTURE OF A TETRAHEDRAL TRANSITION STATE COMPLEX OF ALPHA-*CHYMOTRYPSIN AT 1.8-*ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
6cha:F (GLN30) to (LYS84) STRUCTURE OF A TETRAHEDRAL TRANSITION STATE COMPLEX OF ALPHA-*CHYMOTRYPSIN AT 1.8-*ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
7kme:H (GLN30) to (MET84) CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN INHIBITED WITH SEL2711. | SELECTIDE INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
8gch:F (GLN30) to (LYS84) GAMMA-CHYMOTRYPSIN IS A COMPLEX OF ALPHA-CHYMOTRYPSIN WITH ITS OWN AUTOLYSIS PRODUCTS | HYDROLASE, SERINE PROTEINASE, HYDROLASE-PEPTIDE COMPLEX
8gpb:A (LEU198) to (THR240) STRUCTURAL MECHANISM FOR GLYCOGEN PHOSPHORYLASE CONTROL BY PHOSPHORYLATION AND AMP | GLYCOGEN PHOSPHORYLASE
8kme:2 (GLN30) to (MET84) CRYSTAL STRUCTURE OF HUMAN ALPHA-THROMBIN INHIBITED WITH SEL2770. | THROMBIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SELECTIDE
1a0h:B (GLN335) to (MET400) THE X-RAY CRYSTAL STRUCTURE OF PPACK-MEIZOTHROMBIN DESF1: KRINGLE/THROMBIN AND CARBOHYDRATE/KRINGLE/THROMBIN INTERACTIONS AND LOCATION OF THE LINKER CHAIN | SERINE PROTEASE, COAGULATION, THROMBIN, PROTHROMBIN, MEIZOTHROMBIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1a0h:E (GLN335) to (MET400) THE X-RAY CRYSTAL STRUCTURE OF PPACK-MEIZOTHROMBIN DESF1: KRINGLE/THROMBIN AND CARBOHYDRATE/KRINGLE/THROMBIN INTERACTIONS AND LOCATION OF THE LINKER CHAIN | SERINE PROTEASE, COAGULATION, THROMBIN, PROTHROMBIN, MEIZOTHROMBIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3edx:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF THE W215A/E217A MUTANT OF MURINE THROMBIN | SERINE PROTEASE, ACUTE PHASE, BLOOD COAGULATION, CLEAVAGE ON PAIR OF BASIC RESIDUES, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HYDROLASE, KRINGLE, PROTEASE, ZYMOGEN
1ae8:H (GLN30) to (MET84) HUMAN ALPHA-THROMBIN INHIBITION BY EOC-D-PHE-PRO-AZALYS-ONP | COMPLEX (SERINE PROTEASE-INHIBITOR), BLOOD COAGULATION, N- ETHOXYCARBONYL-D-PHE-PRO-ALFA-AZALYS-P-NITROPHENYLESTER, SERINE PROTEINASE INHIBITION, GLYCOSYLATED PROTEIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2oua:A (LEU33) to (VAL87) CRYSTAL STRUCTURE OF NOCARDIOPSIS PROTEASE (NAPASE) | SERINE PROTEASE; KINETIC STABILITY; ACID STABILITY; ELECTROSTATICS, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1ny2:2 (GLN30) to (MET84) HUMAN ALPHA THROMBIN INHIBITED BY RPPGF AND HIRUGEN | THROMBOSIS, RETRO BINDING, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1bjv:A (GLN30) to (SER84) BETA-TRYPSIN COMPLEXED WITH APPU | HYDROLASE, SERINE PROTEASE, DIGESTION, PANCREAS, ZYMOGEN
1o2o:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2p:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2r:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o2x:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o36:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o38:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3b:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3h:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1o3o:A (GLN30) to (SER84) ELABORATE MANIFOLD OF SHORT HYDROGEN BOND ARRAYS MEDIATING BINDING OF ACTIVE SITE-DIRECTED SERINE PROTEASE INHIBITORS | SERINE PROTEASE, SHORT HYDROGEN BOND, INHIBITION MECHANISM, SHIFT OF PKA, TRYPSIN, THROMBIN, UROKINASE, FACTOR XA, HYDROLASE
1bs5:B (GLU579) to (GLY624) PEPTIDE DEFORMYLASE AS ZN2+ CONTAINING FORM | HYDROLASE, IRON METALLOPROTEASE; PROTEIN SYNTHESIS
2bvx:H (GLN30) to (MET84) DESIGN AND DISCOVERY OF NOVEL, POTENT THROMBIN INHIBITORS WITH A SOLUBILIZING CATIONIC P1-P2-LINKER | SERINE PROTEINASE, COAGULATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1p:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c1t:A (GLN30) to (SER84) RECRUITING ZINC TO MEDIATE POTENT, SPECIFIC INHIBITION OF SERINE PROTEASES | ZN(II)-MEDIATED SERINE PROTEASE INHIBITORS, PH DEPENDENCE, ZN(II) AFFINITY STUCTURE-BASED DRUG DESIGN, SERINE PROTEASE/INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1c5p:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c5r:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1- BINDING, SUB-MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
1c5u:A (GLN30) to (SER84) STRUCTURAL BASIS FOR SELECTIVITY OF A SMALL MOLECULE, S1-BINDING, SUB- MICROMOLAR INHIBITOR OF UROKINASE TYPE PLASMINOGEN ACTIVATOR | SELECTIVE, S1 SITE INHIBITOR, STRUCTURE-BASED DRUG DESIGN, UROKINASE, TRYPSIN, THROMBIN, HYDROLASE
2pr3:A (GLN30) to (GLU84) FACTOR XA INHIBITOR | FXA COAGULATION FACTOR INHIBITOR, BLOOD CLOTTING
1cbw:B (GLN30) to (LYS84) BOVINE CHYMOTRYPSIN COMPLEXED TO BPTI | SERINE PROTEASE, INHIBITOR, PROTEASE-SUBSTRATE INTERACTIONS, COMPLEX (SERINE PROTEASE/INHIBITOR)
1os8:A (PHE29) to (ARG84) RECOMBINANT STREPTOMYCES GRISEUS TRYPSIN | TRYPSIN, SERINE PROTEASE, HYDROLASE
1pjp:A (TYR29) to (GLU84) THE 2.2 A CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH SUCCINYL- ALA-ALA-PRO-PHE-CHLOROMETHYLKETONE | HUMAN CHYMASE, SERINE PROTEINASE, DIPEPTIDYL CARBOXYPEPTIDASE, ANGIOTENSIN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
4iw4:F (LEU447) to (ALA518) CRYSTAL STRUCTURE OF THE SERINE PROTEASE DOMAIN OF MASP-3 IN COMPLEX WITH ECOTIN | TRYPSIN-LIKE FOLD, PROTEASE, INHIBITOR, EXTRACELLULAR, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1pq8:A (ILE30) to (SER83) TRYPSIN AT PH 4 AT ATOMIC RESOLUTION | TRYPSIN, ATOMIC RESOLUTION, CATALYSIS, HYDROLASE
2r9p:A (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR(BPTI) | HUMAN MESOTRYPSIN, SERINE PROTEASE, BOVINE PANCREATIC TRYPSIN INHIBITOR, BPTI, ALTERNATIVE SPLICING, CALCIUM, DIGESTION, HYDROLASE, METAL-BINDING, SECRETED, SULFATION, ZYMOGEN, PHARMACEUTICAL, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
2r9p:C (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR(BPTI) | HUMAN MESOTRYPSIN, SERINE PROTEASE, BOVINE PANCREATIC TRYPSIN INHIBITOR, BPTI, ALTERNATIVE SPLICING, CALCIUM, DIGESTION, HYDROLASE, METAL-BINDING, SECRETED, SULFATION, ZYMOGEN, PHARMACEUTICAL, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
2r9p:D (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH BOVINE PANCREATIC TRYPSIN INHIBITOR(BPTI) | HUMAN MESOTRYPSIN, SERINE PROTEASE, BOVINE PANCREATIC TRYPSIN INHIBITOR, BPTI, ALTERNATIVE SPLICING, CALCIUM, DIGESTION, HYDROLASE, METAL-BINDING, SECRETED, SULFATION, ZYMOGEN, PHARMACEUTICAL, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
1elb:A (GLN30) to (GLY88) ANALOGOUS INHIBITORS OF ELASTASE DO NOT ALWAYS BIND ANALOGOUSLY | HYDROLASE-HYDROLASE INHIBITOR COMPLEX, SERINE PROTEINASE
1qj1:B (GLN30) to (MET84) NOVEL COVALENT ACTIVE SITE THROMBIN INHIBITORS | BLOOD COAGULATION-INHIBITOR, PROTEINASE, TRYPSIN LIKE PROTEINASE, PROTEASE-INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
2snw:B (PHE188) to (GLY232) SINDBIS VIRUS CAPSID PROTEIN, TYPE3 CRYSTAL FORM | SINDBIS, VIRUS, PROTEINASE, ALPHAVIRUS, CAPSID, CHYMOTRYPSIN, VIRUS COAT PROTEIN, VIRAL PROTEIN
4k2y:A (TYR29) to (GLU84) CRYSTAL STRUCTURE OF HUMAN CHYMASE IN COMPLEX WITH FRAGMENT INHIBITOR 6-CHLORO-1,3-DIHYDRO-2H-INDOL-2-ONE | SERINE PROTEASE, GLYCOSYLATED, MAST CELLS, SECRETED, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3uir:B (GLN576) to (GLU634) CRYSTAL STRUCTURE OF THE PLASMIN-TEXTILININ-1 COMPLEX | SERINE PROTEASE, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1rjx:B (GLN576) to (GLU634) HUMAN PLASMINOGEN CATALYTIC DOMAIN, K698M MUTANT | MICROPLASMINOGEN, PLASMINOGEN ACTIVATION, STREPTOKINASE, HYDROLASE
1fy8:E (GLN30) to (ASN84) CRYSTAL STRUCTURE OF THE DELTAILE16VAL17 RAT ANIONIC TRYPSINOGEN-BPTI COMPLEX | PROTEIN-PROTEIN COMPLEX, PROTEASE-INHIBITOR COMPLEX, BETA BARREL, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3utu:H (GLN30) to (MET84) HIGH AFFINITY INHIBITOR OF HUMAN THROMBIN | SERINE PROTEASE, BLOOD CLOTTING, FIBRINOPEPTIDE A, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3uwa:A (ASN75) to (LYS123) CRYSTAL STRUCTURE OF A PROBABLE PEPTIDE DEFORMYLASE FROM SYNECHOCOCCUS PHAGE S-SSM7 | SYNECHOCOCCUS PHAGE, PROBABLE PEPTIDE DEFORMYLASE, HYDROLASE
4zae:A (TRP29) to (ASN84) DEVELOPMENT OF A NOVEL CLASS OF POTENT AND SELECTIVE FIXA INHIBITORS | SERINE PROTEINASE, BLOOD COAGULATION, COAGULATION FACTOR, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
1ghz:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI- CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gi0:A (GLN30) to (SER84) A NOVEL SERINE PROTEASE INHIBITION MOTIF INVOLVING A MULTI-CENTERED SHORT HYDROGEN BONDING NETWORK AT THE ACTIVE SITE | THREE-CENTERED, VERY SHORT HYDROGEN BOND, OXYANION HOLE WATER, SHIFT OF PKA OF HIS57, STRUCTURE-BASED DRUG DESIGN, SPECIFICITY, UROKINASE, TRYPSIN, THROMBIN, ZN+2-MEDIATED INHIBITION, HYDROLASE
1gmc:F (GLN30) to (LYS84) THE X-RAY CRYSTAL STRUCTURE OF THE TETRAHEDRAL INTERMEDIATE OF GAMMA- CHYMOTRYPSIN IN HEXANE | HYDROLASE, SERINE PROTEASE
1sg8:E (GLN30) to (MET84) CRYSTAL STRUCTURE OF THE PROCOAGULANT FAST FORM OF THROMBIN | THROMBIN, ALLOSTERY, HYDROLASE
2vnt:A (PHE24) to (GLU86) UROKINASE-TYPE PLASMINOGEN ACTIVATOR INHIBITOR COMPLEX WITH A 1-(7-SULPHOAMIDOISOQUINOLINYL)GUANIDINE | UPA, INHIBITOR COMPLEX, HYDROLASE
2vnt:F (PHE24) to (GLU86) UROKINASE-TYPE PLASMINOGEN ACTIVATOR INHIBITOR COMPLEX WITH A 1-(7-SULPHOAMIDOISOQUINOLINYL)GUANIDINE | UPA, INHIBITOR COMPLEX, HYDROLASE
3vd5:B (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (N460S) | TRANSITION STATE STABILIZATION, SUBSTRATE BINDING, 2-STAGE BINDING, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
3vd7:A (LEU651) to (ALA716) E. COLI (LACZ) BETA-GALACTOSIDASE (N460S) IN COMPLEX WITH GALACTOTETRAZOLE | TRANSITION STATE STABILIZATION, SUBSTRATE BINDING, 2-STAGE BINDING, TIM BARREL (ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN, BETA SUPERSANDWICH, GLYCOSIDASE, HYDROLASE
1gvz:A (GLN30) to (GLN84) PROSTATE SPECIFIC ANTIGEN (PSA) FROM STALLION SEMINAL PLASMA | ANTIGEN, PROSTATE SPECIFIC ANTIGEN, HYDROLASE
1h1b:A (MET30) to (ALA84) CRYSTAL STRUCTURE OF HUMAN NEUTROPHIL ELASTASE COMPLEXED WITH AN INHIBITOR (GW475151) | HYDROLASE, SERINE PROTEASE,
1h1b:B (MET30) to (ALA84) CRYSTAL STRUCTURE OF HUMAN NEUTROPHIL ELASTASE COMPLEXED WITH AN INHIBITOR (GW475151) | HYDROLASE, SERINE PROTEASE,
1t31:A (TYR29) to (GLU84) A DUAL INHIBITOR OF THE LEUKOCYTE PROTEASES CATHEPSIN G AND CHYMASE WITH THERAPEUTIC EFFICACY IN ANIMALS MODELS OF INFLAMMATION | HUMAN CHYMASE, SERINE PROTEINASE, HYDROLASE
1tgt:A (GLN30) to (SER84) ON THE DISORDERED ACTIVATION DOMAIN IN TRYPSINOGEN. CHEMICAL LABELLING AND LOW-TEMPERATURE CRYSTALLOGRAPHY | HYDROLASE ZYMOGEN (SERINE PROTEINASE)
1toc:B (GLN30) to (MET84) STRUCTURE OF SERINE PROTEINASE | VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE KUNITZ-LIKE INHIBITOR, KRINGLE, SIGNAL, COMPLEX (HYDROLASE/INHIBITOR) COMPLEX
1toc:D (GLN30) to (MET84) STRUCTURE OF SERINE PROTEINASE | VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE KUNITZ-LIKE INHIBITOR, KRINGLE, SIGNAL, COMPLEX (HYDROLASE/INHIBITOR) COMPLEX
1toc:F (GLN30) to (MET84) STRUCTURE OF SERINE PROTEINASE | VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE KUNITZ-LIKE INHIBITOR, KRINGLE, SIGNAL, COMPLEX (HYDROLASE/INHIBITOR) COMPLEX
1toc:H (GLN30) to (MET84) STRUCTURE OF SERINE PROTEINASE | VITAMIN K, ZYMOGEN, GAMMA-CARBOXYGLUTAMIC ACID, ACUTE PHASE, LIVER, HYDROLASE, SERINE PROTEASE KUNITZ-LIKE INHIBITOR, KRINGLE, SIGNAL, COMPLEX (HYDROLASE/INHIBITOR) COMPLEX
1tx6:B (GLN30) to (ASN84) TRYPSIN:BBI COMPLEX | ANTICARCINOGENIC ACTIVITY, DOUBLE-HEADED INHIBITOR, GENE DUPLICATION, MONOCOTYLEDONOUS PLANT, INHIBITORY LOOP, HYDROLASE/PROTEIN BINDING COMPLEX
1tx6:D (GLN30) to (ASN84) TRYPSIN:BBI COMPLEX | ANTICARCINOGENIC ACTIVITY, DOUBLE-HEADED INHIBITOR, GENE DUPLICATION, MONOCOTYLEDONOUS PLANT, INHIBITORY LOOP, HYDROLASE/PROTEIN BINDING COMPLEX
1hyl:A (TYR29) to (ASN84) THE 1.8 A STRUCTURE OF COLLAGENASE FROM HYPODERMA LINEATUM | HYDROLASE (SERINE PROTEASE)
2hvx:A (TYR29) to (GLU84) DISCOVERY OF POTENT, ORALLY ACTIVE, NONPEPTIDE INHIBITORS OF HUMAN MAST CELL CHYMASE BY USING STRUCTURE-BASED DRUG DESIGN | SERINE PROTEASE, HYDROLASE
1id5:H (GLN30) to (SER83) CRYSTAL STRUCTURE OF BOVINE THROMBIN COMPLEX WITH PROTEASE INHIBITOR ECOTIN | THROMBIN, ECOTIN M84R, CONFORMATIONAL CHANGES, HYDROLASE
1ijq:B (ALA378) to (SER423) CRYSTAL STRUCTURE OF THE LDL RECEPTOR YWTD-EGF DOMAIN PAIR | BETA-PROPELLER, LIPID TRANSPORT
1ik3:A (SER57) to (VAL128) LIPOXYGENASE-3 (SOYBEAN) COMPLEX WITH 13(S)-HYDROPEROXY- 9(Z),11(E)-OCTADECADIENOIC ACID | OXIDOREDUCTASE, PURPLE LIPOXYGENASE, FE(III) COMPLEX, INTERM
5a8z:A (MET30) to (ALA84) CRYSTAL STRUCTURE OF HUMAN NEUTROPHIL ELASTASE IN COMPLEX WITH A DIHYDROPYRIMIDONE INHIBITOR | TRYPSIN FAMILY FOLD, PROTEASE, HYDROLASE, HYDROLASE- INHIBITOR COMPLEX
1iqf:A (GLN30) to (GLU84) HUMAN COAGULATION FACTOR XA IN COMPLEX WITH M55165 | HYDROLASE, SERINE PROTEASE, BLOOD COAGULATION FACTOR, COMPLEX
1utp:A (GLN30) to (SER84) TRYPSIN SPECIFICITY AS ELUCIDATED BY LIE CALCULATIONS, X-RAY STRUCTURES AND ASSOCIATION CONSTANT MEASUREMENTS | HYDROLASE, TRYPSIN, INHIBITOR SPECIFICITY, ELECTROSTATIC INTERACTIONS, COLD-ADAPTATION, MOLECULAR DYNAMICS, BINDING FREE ENERGY HYDROLASE
1uw7:A (CYS14) to (GLU68) NSP9 PROTEIN FROM SARS-CORONAVIRUS. | VIRUS, VIRAL PROTEIN, REPLICASE PROTEIN, SARS, CORONAVIRUS, RNA-BINDING
1v2r:T (GLN30) to (SER84) TRYPSIN INHIBITOR IN COMPLEX WITH BOVINE TRYPSIN VARIANT X(SSRI)BT.B4 | SERINE PROTEASE, HYDROLASE, SERINE PROTEINASE
1w8n:A (GLU584) to (ALA639) CONTRIBUTION OF THE ACTIVE SITE ASPARTIC ACID TO CATALYSIS IN THE BACTERIAL NEURAMINIDASE FROM MICROMONOSPORA VIRIDIFACIENS. | GLYCOSIDASE, HYDROLASE, NEURAMINIDASE, BETA- PROPELLER FOLD.
2mqh:A (GLU14) to (ALA78) SOLUTION STRUCTURE OF THE CHLAMYDOMONAS REINHARDTII NAB1 COLD SHOCK DOMAIN, CSD1 | PROTEIN, COLD SHOCK DOMAIN, RNA-BINDING, CHLAMYDOMONAS REINHARDTII, ALGAE, DNA BINDING PROTEIN
5c67:B (GLN30) to (ASN84) HUMAN MESOTRYPSIN IN COMPLEX WITH AMYLOID PRECURSOR PROTEIN INHIBITOR VARIANT APPI-M17G/I18F/F34V | APPI, KUNITZ DOMAIN, TRYPSIN, HYRDOLASE-HYDROLASE INHIBITOR COMPLEX
1xem:A (ASN74) to (GLY124) HIGH RESOLUTION CRYSTAL STRUCTURE OF ESCHERICHIA COLI ZINC- PEPTIDE DEFORMYLASE BOUND TO FORMATE | ZINC DEFORMYLASE, FORMATE, HYDROLASE
5cha:B (GLN30) to (LYS84) THE REFINEMENT AND THE STRUCTURE OF THE DIMER OF ALPHA- *CHYMOTRYPSIN AT 1.67-*ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
5cha:F (GLN30) to (LYS84) THE REFINEMENT AND THE STRUCTURE OF THE DIMER OF ALPHA- *CHYMOTRYPSIN AT 1.67-*ANGSTROMS RESOLUTION | HYDROLASE (SERINE PROTEINASE)
1lxk:A (SER704) to (PHE746) STREPTOCOCCUS PNEUMONIAE HYALURONATE LYASE IN COMPLEX WITH TETRASACCHARIDE HYALURONAN SUBSTRATE | PROTEIN-CARBOHYDRATE COMPLEX, LYASE
2zhf:H (GLN30) to (MET84) EXPLORING THROMBIN S3 POCKET | BLOOD COAGULATION, HYDROLASE INHIBITORS, ACUTE PHASE, CLEAVAGE ON PAIR OF BASIC RESIDUES, GAMMA-CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, KRINGLE, PROTEASE, SECRETED, SERINE PROTEASE, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, SULFATION, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
1mcv:A (GLN30) to (GLY84) CRYSTAL STRUCTURE ANALYSIS OF A HYBRID SQUASH INHIBITOR IN COMPLEX WITH PORCINE PANCREATIC ELASTASE | ELASTASE-INHIBITOR COMPLEX, HYBRID SQUASH INHIBITOR, HYDROLASE
1mh0:B (GLN30) to (MET84) CRYSTAL STRUCTURE OF THE ANTICOAGULANT SLOW FORM OF THROMBIN | THROMBIN, ALLOSTERY, SODIUM BINDING, SERINE PROTEASE, BLOOD CLOTTING
4afz:A (TYR14) to (GLU71) HUMAN CHYMASE - FYNOMER COMPLEX | HYDROLASE-DE NOVO PROTEIN COMPLEX, INHIBITOR, SERINE PROTEASE
3kwf:B (HIS66) to (GLU117) HUMAN DPP-IV WITH CARMEGLIPTIN (S)-1-((2S,3S,11BS)-2-AMINO- 9,10-DIMETHOXY-1,3,4,6,7,11B-HEXAHYDRO-2H-PYRIDO[2,1- A]ISOQUINOLIN-3-YL)-4-FLUOROMETHYL-PYRROLIDIN-2-ONE | DIABETES TYPE II, AMINOPEPTIDASE, CELL MEMBRANE, DISULFIDE BOND, GLYCOPROTEIN, HYDROLASE, MEMBRANE, PROTEASE, SECRETED, SERINE PROTEASE, SIGNAL-ANCHOR, TRANSMEMBRANE
1ypm:H (GLN30) to (MET84) X-RAY CRYSTAL STRUCTURE OF THROMBIN INHIBITED BY SYNTHETIC CYANOPEPTIDE ANALOGUE RA-1014 | THROMBIN, INHIBITOR COMPLEX, BARREL, 6 STRANDED BETA-SHEET, BLOOD CLOTTING-HYDROLASE INHIBITOR COMPLEX
3l3t:D (GLN30) to (ASN84) HUMAN MESOTRYPSIN COMPLEXED WITH AMYLOID PRECURSOR PROTEIN INHIBITOR VARIANT (APPIR15K) | HUMAN MESOTRYPSIN, CANONICAL INHIBITOR, ALZHEIMER'S AMYLOID PRECURSOR PROTEIN INHIBITOR,APPI, APPI-R15K, HYDROLASE-CELL ADHESION COMPLEX
3lc5:A (VAL31) to (ASN84) SELECTIVE BENZOTHIOPHINE INHIBITORS OF FACTOR IXA | PROTEIN-INHIBITOR COMPLEX, PEPTIDASE S1, BLOOD COAGULATION, CALCIUM, CLEAVAGE ON PAIR OF BASIC RESIDUES, DISEASE MUTATION, DISULFIDE BOND, EGF-LIKE DOMAIN, GAMMA- CARBOXYGLUTAMIC ACID, GLYCOPROTEIN, HEMOPHILIA, HYDROLASE, HYDROXYLATION, PHARMACEUTICAL, PHOSPHOPROTEIN, POLYMORPHISM, PROTEASE, SECRETED, SERINE PROTEASE, SULFATION, ZYMOGEN, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
3arq:A (THR77) to (ALA125) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH IDARUBICIN | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
3arv:A (THR77) to (SER124) CRYSTAL STRUCTURE ANALYSIS OF CHITINASE A FROM VIBRIO HARVEYI WITH NOVEL INHIBITORS - COMPLEX STRUCTURE WITH SANGUINARINE | TIM BARREL, INHIBITOR COMPLEX, GLYCOSIDASE, HYDROLASE, HYDROLASE- HYDROLASE INHIBITOR COMPLEX
4b30:A (VAL140) to (VAL219) STRUCTURE OF THE MUTANT V44A OF THE FLUORESCENT PROTEIN KILLERRED | FLUORESCENT PROTEIN, PHOTOBLEACHING, PHOTOCONVERSION, ROS
4b30:B (ASP141) to (VAL219) STRUCTURE OF THE MUTANT V44A OF THE FLUORESCENT PROTEIN KILLERRED | FLUORESCENT PROTEIN, PHOTOBLEACHING, PHOTOCONVERSION, ROS
3m6p:A (LYS78) to (ARG125) CRYSTAL STRUCTURE OF ARABIDOPSIS THALIANA PEPTIDE DEFORMYLASE 1B (ATPDF1B) IN COMPLEX WITH ACTINONIN | PEPTIDE DEFORMYLASE, 1B, PDF, N-TERMINAL EXCISION PATHWAY, NME, ARABIDOPSIS THALIANA, INDUCED-FIT, HYDROLASE, METAL-BINDING, MITOCHONDRION, PROTEIN BIOSYNTHESIS, TRANSIT PEPTIDE, HYDROLASE- ANTIBIOTIC COMPLEX
5egm:A (TRP29) to (ASN84) DEVELOPMENT OF A NOVEL TRICYCLIC CLASS OF POTENT AND SELECTIVE FIXA INHIBITORS | SERINE PROTEINASE, BLOOD COAGULATION, COAGULATION FACTOR, HYDROLASE-2 HYDROLASE INHIBITOR COMPLEX, HYDROLASE-HYDROLASE INHIBITOR COMPLEX
5ek5:A (PRO43) to (PRO109) STRUCTURAL CHARACTERIZATION OF IRMA FROM ESCHERICHIA COLI | FIBRONECTIN FOLD, VIRULENCE, SECRETED PROTEIN, UNKNOWN FUNCTION
3bg4:B (GLN30) to (LYS84) THE CRYSTAL STRUCTURE OF GUAMERIN IN COMPLEX WITH CHYMOTRYPSIN AND THE DEVELOPMENT OF AN ELASTASE-SPECIFIC INHIBITOR | GUAMERIN, CHYMOTRYPSIN, ELASTASE, INHIBITOR, DIGESTION, HYDROLASE, PROTEASE, SECRETED, SERINE PROTEASE, ZYMOGEN, PROTEASE INHIBITOR, SERINE PROTEASE INHIBITOR, HYDROLASE/HYDROLASE INHIBITOR COMPLEX
3muz:3 (LEU651) to (ALA716) E.COLI (LACZ) BETA-GALACTOSIDASE (R599A) IN COMPLEX WITH IPTG | ARG-599-ALA, BETA-GALACTOSIDASE, HYDROLASE TIM BARREL(ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3mv1:3 (ASN649) to (ALA716) E.COLI (LACZ) BETA-GALACTOSIDASE (R599A) IN COMPLEX WITH GUANIDINIUM | ARG-599-ALA, BETA-GALACTOSIDASE, HYDROLASE TIM BARREL(ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3mv1:4 (ASN649) to (ALA716) E.COLI (LACZ) BETA-GALACTOSIDASE (R599A) IN COMPLEX WITH GUANIDINIUM | ARG-599-ALA, BETA-GALACTOSIDASE, HYDROLASE TIM BARREL(ALPHA/BETA BARREL), JELLY-ROLL BARREL, IMMUNOGLOBULIN BETA SUPERSANDWHICH, GLYCOSIDASE, HYDROLASE
3brf:A (GLU285) to (GLN361) CSL (LAG-1) BOUND TO DNA WITH LIN-12 RAM PEPTIDE, C2221 | PROTEIN-DNA COMPLEX, SIGNALING, TRANSCRIPTION, NOTCH, DNA- BINDING, ANK REPEAT, DEVELOPMENTAL PROTEIN, DIFFERENTIATION, EGF-LIKE DOMAIN, GLYCOPROTEIN, MEMBRANE, TRANSMEMBRANE, DNA BINDING PROTEIN/DNA COMPLEX
3n50:A (LEU283) to (CYS327) HUMAN EARLY B-CELL FACTOR 3 (EBF3) IPT/TIG AND HLHLH DOMAINS | BETA-BARREL, HELIX-LOOP-HELIX-LOOP-HELIX, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
3n50:D (GLN284) to (CYS327) HUMAN EARLY B-CELL FACTOR 3 (EBF3) IPT/TIG AND HLHLH DOMAINS | BETA-BARREL, HELIX-LOOP-HELIX-LOOP-HELIX, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
3n50:F (GLY282) to (CYS327) HUMAN EARLY B-CELL FACTOR 3 (EBF3) IPT/TIG AND HLHLH DOMAINS | BETA-BARREL, HELIX-LOOP-HELIX-LOOP-HELIX, STRUCTURAL GENOMICS CONSORTIUM, SGC, TRANSCRIPTION
4r5g:B (PRO396) to (ASP460) CRYSTAL STRUCTURE OF THE DNAK C-TERMINUS WITH THE INHIBITOR PET-16 | HELICAL BUNDLE, BETA SHEETS, CHAPERONE, HSP70/DNAK INHIBITORS, MEMBRANE, CHAPERONE-CHAPERONE INHIBITOR COMPLEX
3nwf:B (GLY205) to (THR249) GLYCOPROTEIN B FROM HERPES SIMPLEX VIRUS TYPE 1, LOW-PH | COILED-COIL, ENVELOPE GLYCOPROTEIN, MEMBRANE FUSION, VIRAL PROTEIN, GLYCOPROTEIN B, HERPESVIRUS 1, HSV-1, MEMBRANE
3nwf:C (GLY205) to (THR249) GLYCOPROTEIN B FROM HERPES SIMPLEX VIRUS TYPE 1, LOW-PH | COILED-COIL, ENVELOPE GLYCOPROTEIN, MEMBRANE FUSION, VIRAL PROTEIN, GLYCOPROTEIN B, HERPESVIRUS 1, HSV-1, MEMBRANE
4ci8:B (VAL247) to (VAL291) CRYSTAL STRUCTURE OF THE TANDEM ATYPICAL BETA-PROPELLER DOMAIN OF EML1 | STRUCTURAL PROTEIN, EML1, EML4-ALK, HSP90 INHIBITORS, TUBULIN-BINDING, BETA PROPELLER
3dfj:A (GLN59) to (THR116) CRYSTAL STRUCTURE OF HUMAN PROSTASIN | PROSTASIN, SERINE PROTEASE, GLYCOPROTEIN, HYDROLASE, MEMBRANE, SECRETED, TRANSMEMBRANE, ZYMOGEN
3p70:F (GLN378) to (MET443) STRUCTURAL BASIS OF THROMBIN-MEDIATED FACTOR V ACTIVATION: ESSENTIAL ROLE OF THE HIRUDIN-LIKE SEQUENCE GLU666-GLU672 FOR PROCESSING AT THE HEAVY CHAIN-B DOMAIN JUNCTION | TRYPSIN-LIKE SERINE PROTEINASE, BLOOD COAGULATION, N-GLYCOSYLATION, BLOOD PLASMA, HYDROLASE
3p70:H (GLN378) to (MET443) STRUCTURAL BASIS OF THROMBIN-MEDIATED FACTOR V ACTIVATION: ESSENTIAL ROLE OF THE HIRUDIN-LIKE SEQUENCE GLU666-GLU672 FOR PROCESSING AT THE HEAVY CHAIN-B DOMAIN JUNCTION | TRYPSIN-LIKE SERINE PROTEINASE, BLOOD COAGULATION, N-GLYCOSYLATION, BLOOD PLASMA, HYDROLASE
3pa2:B (GLY332) to (PHE434) CRYSTAL STRUCTURE OF P DOMAIN FROM NORWALK VIRUS STRAIN VIETNAM 026 IN COMPLEX WITH HBGA TYPE LEY | NOROVIRUS, P-DOMAIN, CAPSID, RECEPTOR, HISTO BLOOD GROUP ANTIGEN (HBGA), VIRAL PROTEIN
4vgc:B (GLN30) to (LYS84) GAMMA-CHYMOTRYPSIN D-NAPHTHYL-1-ACETAMIDO BORONIC ACID INHIBITOR COMPLEX | HYDROLASE, SERINE PROTEASE
5k0h:A (GLN30) to (GLU84) HUMAN FACTOR XA IN COMPLEX WITH SYNTHETIC INHIBITOR BENZYLSULFONYL- DSER(BENZYL)-GLY-4-AMIDINOBENZYLAMIDE | HUMAN FACTOR XA, INHIBITOR COMPLEX, BENZAMIDINE INHIBITOR, HYDROLASE, CLOTTING FACTOR
5kai:B (HIS343) to (ASP413) NH3-BOUND RT XFEL STRUCTURE OF PHOTOSYSTEM II 500 MS AFTER THE 2ND ILLUMINATION (2F) AT 2.8 A RESOLUTION | PHOTOSYSTEMS, TRANSMEMBRANE, ROOM TEMPERATURE, ELECTRON TRANSPORT
5knd:F (LEU29) to (ASP91) CRYSTAL STRUCTURE OF THE PI-BOUND V1 COMPLEX | P-LOOP, HYDROLASE, NA(+)-ATPASE, ATP BINDING