4gsy:A (ILE5) to (ALA119) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS BOUND TO INHIBITOR. | TRANSFERASE, NUCLEOTIDE BINDING, THYMIDYLATE KINASE ACTIVITY, ATP BINDING, KINASE ACTIVITY, TRANSFERASE ACTIVITY, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4gsy:B (SER2) to (ILE120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS BOUND TO INHIBITOR. | TRANSFERASE, NUCLEOTIDE BINDING, THYMIDYLATE KINASE ACTIVITY, ATP BINDING, KINASE ACTIVITY, TRANSFERASE ACTIVITY, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4hdc:B (SER2) to (ILE120) DISCOVERY OF SELECTIVE AND POTENT INHIBITORS OF GRAM-POSITIVE BACTERIAL THYMIDYLATE KINASE (TMK: COMPOUND 41) | KINASE, TMP, ACTIVE SITE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4hej:B (SER2) to (ALA119) DISCOVERY OF SELECTIVE AND POTENT INHIBITORS OF GRAM-POSITIVE BACTERIAL THYMIDYLATE KINASE (TMK): COMPUND 16 | TMK, INHIBITOR, TMP, ANTIBACTERIAL, DNA REPAIR, KINASE, DTMP ATP, PHOSPHORYLATION, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2pbr:A (MET1) to (THR118) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE (AQ_969) FROM AQUIFEX AEOLICUS VF5 | KINASE, TRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TMP-BINDING, ATP- BINDING, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
4hlc:B (SER2) to (ILE120) SULFONYLPIPERIDINES AS NOVEL, ANTIBACTERIAL INHIBITORS OF GRAM- POSITIVE THYMIDYLATE KINASE (TMK): COMPOUND 5 | TMK, KINASE, THYMIDYLATE KINASE, MRSA, PIPIRIDINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4hld:B (SER2) to (ILE120) SULFONYLPIPERIDINES AS NOVEL, ANTIBACTERIAL INHIBITORS OF GRAM- POSITIVE THYMIDYLATE KINASE (TMK): COMPOUND 11 | TMK, KINASE, THYMIDYLATE KINASE, MRSA, PIPIRIDINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
2plr:B (LYS3) to (SER117) CRYSTAL STRUCTURE OF DTMP KINASE (ST1543) FROM SULFOLOBUS TOKODAII STRAIN7 | TMP-BINDING, ATP-BINDING, THYMIDYLATE KINASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI, TRANSFERASE
2ccj:B (ILE5) to (ALA119) CRYSTAL STRUCTURE OF S. AUREUS THYMIDYLATE KINASE COMPLEXED WITH THYMIDINE MONOPHOSPHATE | KINASE, TRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TMP-BINDING, ATP-BINDING, THYMIDYLATE KINASE
2cck:A (SER2) to (ALA119) CRYSTAL STRUCTURE OF UNLIGANDED S. AUREUS THYMIDYLATE KINASE | KINASE, TRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TMP-BINDING, ATP-BINDING, THYMIDYLATE KINASE
2cck:B (ILE5) to (ALA119) CRYSTAL STRUCTURE OF UNLIGANDED S. AUREUS THYMIDYLATE KINASE | KINASE, TRANSFERASE, NUCLEOTIDE BIOSYNTHESIS, TMP-BINDING, ATP-BINDING, THYMIDYLATE KINASE
1p60:B (LYS22) to (PHE166) STRUCTURE OF HUMAN DCK COMPLEXED WITH 2'-DEOXYCYTIDINE AND ADP, SPACE GROUP C 2 2 21 | NUCLEOSIDE KINASE, P-LOOP, DEOXYCYTIDINE, TRANSFERASE
1p62:B (LYS22) to (PHE166) STRUCTURE OF HUMAN DCK COMPLEXED WITH GEMCITABINE AND ADP-MG | NUCLEOSIDE KINASE, P-LOOP, GEMCITABINE, TRANSFERASE
1p6x:A (HIS21) to (LEU170) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH THY AND SO4 | P-LOOP, LID, TRANSFERASE
1p72:A (HIS21) to (LEU170) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH THY AND ADP | P-LOOP, LID, TRANSFERASE
1p72:B (THR24) to (LEU170) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH THY AND ADP | P-LOOP, LID, TRANSFERASE
1p73:A (THR24) to (GLY156) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH TP4A | P-LOOP, LID, TRANSFERASE
1p73:B (THR24) to (LEU170) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH TP4A | P-LOOP, LID, TRANSFERASE
1p75:A (THR24) to (LEU170) CRYSTAL STRUCTURE OF EHV4-TK COMPLEXED WITH TP5A | P-LOOP, LID, TRANSFERASE
1p7c:A (PRO47) to (ILE194) CRYSTAL STRUCTURE OF HSV1-TK COMPLEXED WITH TP5A | P-LOOP, LID, BISUBSTRATE INHIBITOR, TRANSFERASE
4xwa:A (PHE4) to (ILE120) TMK FROM S.AUREUS IN COMPLEX WITH THE PIPERIDINYL THYMINE CLASS INHIBITOR WITH A C5 ETHYL-AMINE | TMK, KINASE, ANTIBACTERIAL, PIPERIDINE, THYMIDINE, TRANSFERASE
4xwa:B (SER2) to (ILE120) TMK FROM S.AUREUS IN COMPLEX WITH THE PIPERIDINYL THYMINE CLASS INHIBITOR WITH A C5 ETHYL-AMINE | TMK, KINASE, ANTIBACTERIAL, PIPERIDINE, THYMIDINE, TRANSFERASE
2qrn:A (LYS22) to (PHE137) HUMAN DEOXYCYTIDINE KINASE DCMP, UDP, MG ION PRODUCT COMPLEX | DEOXYCYTIDINE KINASE, DEOXYCYTIDINE MONOPHOSPHATE, URIDINE DIPHOSPHATE, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSFERASE
2qrn:B (LYS22) to (PHE137) HUMAN DEOXYCYTIDINE KINASE DCMP, UDP, MG ION PRODUCT COMPLEX | DEOXYCYTIDINE KINASE, DEOXYCYTIDINE MONOPHOSPHATE, URIDINE DIPHOSPHATE, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSFERASE
2qrn:C (LYS22) to (PHE137) HUMAN DEOXYCYTIDINE KINASE DCMP, UDP, MG ION PRODUCT COMPLEX | DEOXYCYTIDINE KINASE, DEOXYCYTIDINE MONOPHOSPHATE, URIDINE DIPHOSPHATE, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSFERASE
2qrn:D (LYS22) to (PHE137) HUMAN DEOXYCYTIDINE KINASE DCMP, UDP, MG ION PRODUCT COMPLEX | DEOXYCYTIDINE KINASE, DEOXYCYTIDINE MONOPHOSPHATE, URIDINE DIPHOSPHATE, ATP-BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHORYLATION, TRANSFERASE
4ivq:A (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH IN43/5 | DNA SYNTHESIS, PET IMAGING TRACER, ATP BINDING, NUCLEOTIDE BINDING, TRANSFERASE
1e2j:B (PRO47) to (ILE194) THE NUCLEOSIDE BINDING SITE OF HERPES SIMPLEX TYPE 1 THYMIDINE KINASE ANALYZED BY X-RAY CRYSTALLOGRAPHY | TRANSFERASE, ADENINE ANALOG, ENZYME-PRODRUG GENE THERAPY, NUCLEOSIDE- BINDING, THYMIDINE KINASE, X-RAY CRYSTALLOGRAPHY
3tmk:A (MET1) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:B (LYS6) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:C (GLY5) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:D (LYS6) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:E (MET2) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:F (MET1) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:G (MET2) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
3tmk:H (LYS6) to (VAL121) CRYSTAL STRUCTURE OF YEAST THYMIDYLATE KINASE COMPLEXED WITH THE BISUBSTRATE INHIBITOR TP5A AT 2.0 A RESOLUTION: IMPLICATIONS FOR CATALYSIS AND AZT ACTIVATION | KINASE, PHOSPHOTRANSFERASE
4jlj:A (ARG20) to (PHE166) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE F2.1.1 INHIBITOR (2-[({2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-1,3-THIAZOL-4- YL}METHYL)SULFANYL]PYRIMIDINE-4,6-DIAMINE) | PHOSPHORYL TRANSFER, PHOSPHORYLATION, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jlj:B (LYS22) to (PHE166) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE F2.1.1 INHIBITOR (2-[({2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-1,3-THIAZOL-4- YL}METHYL)SULFANYL]PYRIMIDINE-4,6-DIAMINE) | PHOSPHORYL TRANSFER, PHOSPHORYLATION, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jlk:A (LYS22) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE F2.2.1 INHIBITOR (2-[({2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-5-METHYL-1,3-THIAZOL-4- YL}METHYL)SULFANYL]PYRIMIDINE-4,6-DIAMINE) | PHOSPHORYL TRANSFER, PHOSPHORYLATION, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jlm:A (LYS22) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE F2.3.1 INHIBITOR (2-[({5-ETHYL-2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-1,3-THIAZOL-4- YL}METHYL)SULFANYL]PYRIMIDINE-4,6-DIAMINE) | PHOSPHORYL TRANSFER, PHOSPHORYLATION, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4jlm:B (LYS22) to (GLY167) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE F2.3.1 INHIBITOR (2-[({5-ETHYL-2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-1,3-THIAZOL-4- YL}METHYL)SULFANYL]PYRIMIDINE-4,6-DIAMINE) | PHOSPHORYL TRANSFER, PHOSPHORYLATION, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
2tmk:A (LYS6) to (VAL121) YEAST THYMIDYLATE KINASE COMPLEXED WITH 3'-AZIDO-3'- DEOXYTHYMIDINE MONOPHOSPHATE (AZT-MP) | TRANSFERASE (PHOSPHOTRANSFERASE), KINASE, THYMIDINE ACTIVATION PATHWAY, ENZYME, AZT
2tmk:B (LYS6) to (VAL121) YEAST THYMIDYLATE KINASE COMPLEXED WITH 3'-AZIDO-3'- DEOXYTHYMIDINE MONOPHOSPHATE (AZT-MP) | TRANSFERASE (PHOSPHOTRANSFERASE), KINASE, THYMIDINE ACTIVATION PATHWAY, ENZYME, AZT
3hjn:A (MET1) to (ASP118) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE IN COMPLEX WITH DTDP AND ADP FROM THERMOTOGA MARITIMA | THYMIDYLATE KINASE, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
3hjn:B (MET1) to (ALA116) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE IN COMPLEX WITH DTDP AND ADP FROM THERMOTOGA MARITIMA | THYMIDYLATE KINASE, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, NPPSFA, NATIONAL PROJECT ON PROTEIN STRUCTURAL AND FUNCTIONAL ANALYSES, RIKEN STRUCTURAL GENOMICS/PROTEOMICS INITIATIVE, RSGI
4kcg:A (LYS22) to (PHE166) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE DI-39 INHIBITOR | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
4kcg:B (ARG20) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE DI-39 INHIBITOR | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3ipx:A (LYS22) to (PHE137) X-RAY STRUCTURE OF HUMAN DEOXYCYTIDINE KINASE IN COMPLEX WITH ADP AND AN INHIBITOR | HUMAN DEOXYCYTIDINE KINASE, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
1tmk:A (LYS6) to (VAL121) YEAST THYMIDYLATE KINASE COMPLEXED WITH THYMIDINE MONOPHOSPHATE (DTMP) | TRANSFERASE (PHOSPHOTRANSFERASE), KINASE, THYMIDINE ACTIVATION PATHWAY, ENZYME
1tmk:B (LYS6) to (VAL121) YEAST THYMIDYLATE KINASE COMPLEXED WITH THYMIDINE MONOPHOSPHATE (DTMP) | TRANSFERASE (PHOSPHOTRANSFERASE), KINASE, THYMIDINE ACTIVATION PATHWAY, ENZYME
2wwf:A (LYS9) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH TMP AND ADP | TRANSFERASE, KINASE, MALARIA
2wwf:B (GLY8) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH TMP AND ADP | TRANSFERASE, KINASE, MALARIA
2wwf:C (GLY8) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH TMP AND ADP | TRANSFERASE, KINASE, MALARIA
2wwh:B (LYS9) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH AP5DT | TRANSFERASE, MALARIA
4mqb:B (SER2) to (ALA119) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS IN COMPLEX WITH 2-(N-MORPHOLINO)ETHANESULFONIC ACID | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS, MTBI, THYMIDYLATE KINASE, TRANSFERASE
2jas:B (MET1) to (VAL112) STRUCTURE OF DEOXYADENOSINE KINASE FROM M.MYCOIDES WITH BOUND DATP | KINASE, TRANSFERASE
2jat:A (MET1) to (LEU113) STRUCTURE OF DEOXYADENOSINE KINASE FROM M.MYCOIDES WITH PRODUCTS DCMP AND A FLEXIBLE DCDP BOUND | KINASE, TRANSFERASE, DEOXYRIBONUCLEOSIDE KINASE
2jat:B (MET1) to (LEU113) STRUCTURE OF DEOXYADENOSINE KINASE FROM M.MYCOIDES WITH PRODUCTS DCMP AND A FLEXIBLE DCDP BOUND | KINASE, TRANSFERASE, DEOXYRIBONUCLEOSIDE KINASE
1ki3:B (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH PENCICLOVIR | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, ANTIVIRAL DRUG PENCICLOVIR
1ki4:B (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE I COMPLEXED WITH 5-BROMOTHIENYLDEOXYURIDINE | PHOSPHOTRANSFERASE, THYMIDINE KINASE, VIRIDAE, DS-DNA ENVELOPED VIRUSES, HERPESVIRIDAE, ALPHAHERPESVIRINAE, SUBSTRATE ANALOG, 5-BROMOTHIENYLDEOXYURIDINE
1ko8:A (ASP7) to (PRO103) CRYSTAL STRUCTURE OF GLUCONATE KINASE | ALFA/BETA, TRANSFERASE
2no0:B (LYS22) to (PHE137) C4S DCK VARIANT OF DCK IN COMPLEX WITH GEMCITABINE+ADP | DCK, GEMCITABINE, HUMAN DEOXYCYTIDINE KINASE, TRANSFERASE
2no1:B (LYS22) to (PHE137) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DC+ADP | DCK, HUMAN DEOXYCYTIDINE KINASE, D-DC, TRANSFERASE
2no6:B (LYS22) to (PHE166) C4S DCK VARIANT OF DCK IN COMPLEX WITH FTC+ADP | DCK, EMTRICITABINE, HUMAN DEOXYCYTIDINE KINASE, FTC, ENANTIOMER, ANTIVIRAL, TRANSFERASE
2no7:B (LYS22) to (PHE137) C4S DCK VARIANT OF DCK IN COMPLEX WITH L-DC+ADP | DCK, HUMAN DEOXYCYTIDINE KINASE, L-DC, ENANTIOMER, ENANTIOSELECTIVITY, TRANSFERASE
2no9:B (ARG20) to (GLY167) THE STRUCTURE OF DEOXYCYTIDINE KINASE COMPLEXED WITH TROXACITABINE AND ADP. | DCK, TROXACITABINE, HUMAN DEOXYCYTIDINE KINASE, L-DC, ENANTIOMER, ANTICANCER, TRANSFERASE
2noa:B (LYS22) to (PHE137) THE STRUCTURE OF DEOXYCYTIDINE KINASE COMPLEXED WITH LAMIVUDINE AND ADP. | DCK, 3TC, HUMAN DEOXYCYTIDINE KINASE, L-DC, ENANTIOMER, ANTIVIRAL, LAMIVUDINE, EPIVIR, TRANSFERASE
2yog:A (GLY8) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH A (THIO)UREA-ALPHA-DEOXYTHYMIDINE INHIBITOR | TRANSFERASE, MALARIA, INHIBITOR
2yoh:A (GLY8) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH A UREA-ALPHA-DEOXYTHYMIDINE INHIBITOR | TRANSFERASE, MALARIA, INHIBITOR
2yoh:B (PHE10) to (GLN124) PLASMODIUM FALCIPARUM THYMIDYLATE KINASE IN COMPLEX WITH A UREA-ALPHA-DEOXYTHYMIDINE INHIBITOR | TRANSFERASE, MALARIA, INHIBITOR
2zi4:A (LYS22) to (PHE166) C4S DCK VARIANT OF DCK IN COMPLEX WITH L-DA+ADP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, L-DA, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi5:B (ARG2020) to (GLU2145) C4S DCK VARIANT OF DCK IN COMPLEX WITH L-DA+UDP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, L-DA, UDP, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi5:D (ARG4020) to (GLY4167) C4S DCK VARIANT OF DCK IN COMPLEX WITH L-DA+UDP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, L-DA, UDP, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi6:A (LYS1022) to (PHE1166) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DA+UDP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, D-DA, UDP, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi6:B (ARG2020) to (GLN2165) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DA+UDP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, D-DA, UDP, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi6:D (ARG4020) to (GLU4145) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DA+UDP | DCK, PURINE, DEOXYADENOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, D-DA, UDP, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi7:B (LYS22) to (PHE137) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DG+UDP | DCK, PURINE, DEOXYGUANOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, D-DG, DG, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zi7:A (LYS22) to (PHE166) C4S DCK VARIANT OF DCK IN COMPLEX WITH D-DG+UDP | DCK, PURINE, DEOXYGUANOSINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, ENANTIOMER, D-DG, DG, ATP-BINDING, NUCLEOTIDE- BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zia:A (LYS22) to (PHE166) C4S DCK VARIANT OF DCK IN COMPLEX WITH CLADRIBINE+UDP | DCK, PURINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, CLADRIBINE, 2-CHLORO-2'-DEOXYADENOSINE, DEOXYADENOSINE ANALOG, UDP, ATP- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
2zia:B (LYS22) to (GLY167) C4S DCK VARIANT OF DCK IN COMPLEX WITH CLADRIBINE+UDP | DCK, PURINE, DEOXYCYTIDINE KINASE, NUCLEOSIDE, CLADRIBINE, 2-CHLORO-2'-DEOXYADENOSINE, DEOXYADENOSINE ANALOG, UDP, ATP- BINDING, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
4oql:B (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH DF-EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
4oqm:B (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH F-ARA-EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
4oqn:B (PRO47) to (ILE194) CRYSTAL STRUCTURE OF THYMIDINE KINASE FROM HERPES SIMPLEX VIRUS TYPE 1 IN COMPLEX WITH EDU | DNA SYNTHESIS, THYMIDINE KINASE, ATP-BINDING, NUCLEOTIDE-BINDING, TRANSFERASE, 5-ETHYNYLURIDINE NUCLEOSIDE DERIVATIVE
3kfx:A (LYS22) to (PHE166) HUMAN DCK COMPLEX WITH 5-ME DC AND ADP | HUMAN DCK, NUCLEOTIDE KINASE, P-LOOP, 5-ME DC, ATP-BINDING, KINASE, NUCLEOTIDE-BINDING, NUCLEUS, PHOSPHOPROTEIN, TRANSFERASE
3ld9:A (SER0) to (VAL120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM EHRLICHIA CHAFFEENSIS AT 2.15A RESOLUTION | SSGCID, NIH, NIAID, SBRI, UW, EMERALD BIOSTRUCTURES, EHRLICHIA CHAFFEENSIS, THYMIDYLATE KINASE, ALS COLLABORATIVE CRYSTALLOGRAPHY, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
3ld9:C (SER0) to (VAL120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM EHRLICHIA CHAFFEENSIS AT 2.15A RESOLUTION | SSGCID, NIH, NIAID, SBRI, UW, EMERALD BIOSTRUCTURES, EHRLICHIA CHAFFEENSIS, THYMIDYLATE KINASE, ALS COLLABORATIVE CRYSTALLOGRAPHY, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
3ld9:D (SER0) to (VAL120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM EHRLICHIA CHAFFEENSIS AT 2.15A RESOLUTION | SSGCID, NIH, NIAID, SBRI, UW, EMERALD BIOSTRUCTURES, EHRLICHIA CHAFFEENSIS, THYMIDYLATE KINASE, ALS COLLABORATIVE CRYSTALLOGRAPHY, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, STRUCTURAL GENOMICS, SEATTLE STRUCTURAL GENOMICS CENTER FOR INFECTIOUS DISEASE
4q1b:A (LYS22) to (GLU145) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 7 {N- (2-(3-(4-(((4,6-DIAMINOPYRIMIDIN-2-YL)THIO)METHYL)-5-PROPYLTHIAZOL-2- YL)PHENOXY)ETHYL)METHANESULFONAMIDE} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q18:A (LYS22) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 4 [1- [5-(4-{[(2,6-DIAMINOPYRIMIDIN-4-YL)SULFANYL]METHYL}-5-PROPYL-1,3- THIAZOL-2-YL)-2-METHOXYPHENOXY]-2-METHYLPROPAN-2-OL] | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q18:B (LYS22) to (GLU145) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 4 [1- [5-(4-{[(2,6-DIAMINOPYRIMIDIN-4-YL)SULFANYL]METHYL}-5-PROPYL-1,3- THIAZOL-2-YL)-2-METHOXYPHENOXY]-2-METHYLPROPAN-2-OL] | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q19:B (ARG20) to (GLY167) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 5 {5- (4-{[(4,6-DIAMINOPYRIMIDIN-2-YL)SULFANYL]METHYL}-5-PROPYL-1,3- THIAZOL-2-YL)-2-METHOXYPHENOL} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1a:A (LYS22) to (PHE166) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 6 {2- [5-(4-{[(4,6-DIAMINOPYRIMIDIN-2-YL)SULFANYL]METHYL}-5-PROPYL-1,3- THIAZOL-2-YL)-2-METHOXYPHENOXY]ETHANOL} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1a:B (ARG20) to (SER144) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 6 {2- [5-(4-{[(4,6-DIAMINOPYRIMIDIN-2-YL)SULFANYL]METHYL}-5-PROPYL-1,3- THIAZOL-2-YL)-2-METHOXYPHENOXY]ETHANOL} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1e:A (LYS22) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 10 {2- {[(1R/S)-1-{2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-5-METHYL-1,3- THIAZOL 4-YL}ETHYL]SULFANYL}PYRIMIDINE-4,6-DIAMINE} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1e:B (LYS22) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 10 {2- {[(1R/S)-1-{2-[3-(2-FLUOROETHOXY)-4-METHOXYPHENYL]-5-METHYL-1,3- THIAZOL 4-YL}ETHYL]SULFANYL}PYRIMIDINE-4,6-DIAMINE} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1f:B (ARG20) to (PHE137) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 12R {N-{2-[5-(4-{(1R)-1-[(4,6-DIAMINOPYRIMIDIN-2-YL)SULFANYL]ETHYL}-5- METHYL-1,3-THIAZOL-2-YL)-2-METHOXYPHENOXY]ETHYL}METHANESULFONAMIDE} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qg7:A (PHE4) to (ILE120) S.AUREUS TMK IN COMPLEX WITH A POTENT INHIBITOR COMPOUND 18, 2-(3- CHLOROPHENOXY)-3-METHOXY-4-{[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]METHYL}BENZOIC ACID | TRANSFERASE/TRANSFERASE INHIBITOR KINASE, THYMIDINE MONPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qg7:B (SER2) to (ILE120) S.AUREUS TMK IN COMPLEX WITH A POTENT INHIBITOR COMPOUND 18, 2-(3- CHLOROPHENOXY)-3-METHOXY-4-{[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]METHYL}BENZOIC ACID | TRANSFERASE/TRANSFERASE INHIBITOR KINASE, THYMIDINE MONPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qga:A (PHE4) to (ILE120) S.AUREUS TMK IN COMPLEX WITH POTENT INHIBITOR COMPOUND 19, 2-(3- CHLOROPHENOXY)-3-FLUORO-4-{[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]METHYL}BENZOIC ACID | TRANSFERASE/TRANSFERASE INHIBITOR KINASE, THYMIDINE MONPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qga:B (ILE5) to (ILE120) S.AUREUS TMK IN COMPLEX WITH POTENT INHIBITOR COMPOUND 19, 2-(3- CHLOROPHENOXY)-3-FLUORO-4-{[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]METHYL}BENZOIC ACID | TRANSFERASE/TRANSFERASE INHIBITOR KINASE, THYMIDINE MONPHOSPHATE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgf:A (PHE4) to (ILE120) S.AUREUS TMK IN COMPLEX WITH THE POTENT INHIBITOR COMPOUND 38, 2-(3- CHLOROPHENOXY)-3-METHOXY-4-{(1R)-1-[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]PROPYL}BENZOIC ACID | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgf:B (ILE5) to (ILE120) S.AUREUS TMK IN COMPLEX WITH THE POTENT INHIBITOR COMPOUND 38, 2-(3- CHLOROPHENOXY)-3-METHOXY-4-{(1R)-1-[(3S)-3-(5-METHYL-2,4-DIOXO-3,4- DIHYDROPYRIMIDIN-1(2H)-YL)PIPERIDIN-1-YL]PROPYL}BENZOIC ACID | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgg:A (ILE5) to (ASN121) TMK IN COMPLEX WITH COMPOUND 46, 2-(3-CHLOROPHENOXY)-3-FLUORO-4-{(1R)- 3-METHYL-1-[(3S)-3-(5-METHYL-2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1(2H)- YL)PIPERIDIN-1-YL]BUTYL}BENZOIC ACID | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgg:B (SER2) to (ILE120) TMK IN COMPLEX WITH COMPOUND 46, 2-(3-CHLOROPHENOXY)-3-FLUORO-4-{(1R)- 3-METHYL-1-[(3S)-3-(5-METHYL-2,4-DIOXO-3,4-DIHYDROPYRIMIDIN-1(2H)- YL)PIPERIDIN-1-YL]BUTYL}BENZOIC ACID | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgh:A (SER2) to (ILE120) S.AUREUS TMK IN COMPLEX WITH POTENT INHIBITOR COMPOUND 47 | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4qgh:B (ALA3) to (ILE120) S.AUREUS TMK IN COMPLEX WITH POTENT INHIBITOR COMPOUND 47 | THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
3mjr:C (ARG20) to (GLN156) HUMAN DCK COMPLEX WITH ACYCLIC NUCLEOSIDE | ACV,GCV,DCK,KINASE,UDP,P-LOOP,KINASE ACTIVITY,NUCLEOSIDE KINASE, TRANSFERASE
3mjr:D (ARG20) to (GLY167) HUMAN DCK COMPLEX WITH ACYCLIC NUCLEOSIDE | ACV,GCV,DCK,KINASE,UDP,P-LOOP,KINASE ACTIVITY,NUCLEOSIDE KINASE, TRANSFERASE
3n2i:B (ASN2) to (ALA125) 2.25 ANGSTROM RESOLUTION CRYSTAL STRUCTURE OF A THYMIDYLATE KINASE (TMK) FROM VIBRIO CHOLERAE O1 BIOVAR ELTOR STR. N16961 IN COMPLEX WITH THYMIDINE | THYMIDYLATE KINASE, VIBRIO CHOLERAE, STRUCTURAL GENOMICS, INFECTIOUS DISEASES, CENTER FOR STRUCTURAL GENOMICS OF INFECTIOUS DISEASES, ATP-BINDING, KINASE, NUCLEOTIDE BIOSYNTHESIS, NUCLEOTIDE-BINDING, TRANSFERASE, CSGID
4rzx:A (LYS3) to (SER117) CRYSTAL STRUCTURE (TYPE-3) OF DTMP KINASE (ST1543) FROM SULFOLOBUS TOKODAII STRAIN7 | TRANSFERASE
4dwj:E (SER2) to (ASN121) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS IN COMPLEX WITH THYMIDINE MONOPHOSPHATE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURES OF MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS, MTBI, THYMIDYLATE KINASE, TRANSFERASE
4dwj:G (PHE4) to (ASN121) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS IN COMPLEX WITH THYMIDINE MONOPHOSPHATE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURES OF MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS, MTBI, THYMIDYLATE KINASE, TRANSFERASE
4eaq:B (ILE5) to (ILE120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS IN COMPLEX WITH 3'-AZIDO-3'-DEOXYTHYMIDINE-5'-MONOPHOSPHATE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, MTBI, THYMIDYLATE KINASE, TRANSFERASE, TRANSFERASE- TRANSFERASE INHIBITOR COMPLEX
3qej:A (LYS22) to (PHE166) S74E-DCK MUTANT IN COMPLEX WITH UDP | ALPHA/BETA, PHOSPHORYL TRANSFER, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3qej:B (LYS22) to (PHE166) S74E-DCK MUTANT IN COMPLEX WITH UDP | ALPHA/BETA, PHOSPHORYL TRANSFER, ATP BINDING, PHOSPHORYLATION, TRANSFERASE
3qeo:A (LYS22) to (GLY167) S74E-R104M-D133A DCK VARIANT IN COMPLEX WITH L-DEOXYTHYMIDINE AND UDP | ALPHA/BETA, PHOSPHORYL TRANSFER, TRANSFERASE
3qeo:B (LYS22) to (PHE166) S74E-R104M-D133A DCK VARIANT IN COMPLEX WITH L-DEOXYTHYMIDINE AND UDP | ALPHA/BETA, PHOSPHORYL TRANSFER, TRANSFERASE
3qen:A (LYS22) to (PHE166) S74E DCK IN COMPLEX WITH 5-BROMODEOXYCYTIDINE AND UDP | ALPHA/BETA, PHOSPHORYL TRANSFER, PHOSPHORYLATION, TRANSFERASE
4f4i:B (ALA3) to (ILE120) CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM STAPHYLOCOCCUS AUREUS IN APO-FORM | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, MIDWEST CENTER FOR STRUCTURAL GENOMICS (MCSG), STRUCTURES OF MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS (MTBI), THYMIDYLATE KINASE, TRANSFERASE
4gmd:B (LEU4) to (GLY125) THE CRYSTAL STRUCTURE OF THYMIDYLATE KINASE FROM PSEUDOMONAS AERUGINOSA PAO1 IN COMPLEX WITH AZT MONOPHOSPHATE | STRUCTURAL GENOMICS, PSI-BIOLOGY, MIDWEST CENTER FOR STRUCTURAL GENOMICS, MCSG, STRUCTURES OF MTB PROTEINS CONFERRING SUSCEPTIBILITY TO KNOWN MTB INHIBITORS, MTBI, PROTEIN STRUCTURE INITIATIVE, TRANSFERASE, TRANSFERASE-INHIBITOR COMPLEX
4l5b:B (ARG20) to (GLY167) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE DI-43 INHIBITOR | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4q1c:A (ARG20) to (PHE166) HUMAN DCK C4S-S74E MUTANT IN COMPLEX WITH UDP AND THE INHIBITOR 8 {2, 2'-[{4-[(2R)-4-{[(4,6-DIAMINOPYRIMIDIN-2-YL)SULFANYL]METHYL}-5- PROPYL-2,3-DIHYDRO-1,3-THIAZOL-2-YL]BENZENE-1,2-DIYL}BIS(OXY) ]DIETHANOL} | PHOSPHORYL TRANSFER, PHOSPHORYLATION, DEOXYCYTIDINE, TRANSFERASE, INHIBITOR COMPLEX, KINASE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gfd:A (PHE4) to (ALA119) THYMIDYLATE KINASE (TMK) FROM S. AUREUS IN COMPLEX WITH TK-666 | KINASE, THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX
4gfd:B (ALA3) to (ILE120) THYMIDYLATE KINASE (TMK) FROM S. AUREUS IN COMPLEX WITH TK-666 | KINASE, THYMIDINE MONPHOSPHATE, SOLUBLE, TRANSFERASE-TRANSFERASE INHIBITOR COMPLEX